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New thienopyrimidine and quinazoline derivatives as potential 5-HT7 receptor ligands. 1-gen-2013 Modica, Maria Nunziata; Intagliata, S; Romeo, Giuseppe; Pittala', Valeria; Salerno, Loredana; Siracusa, Maria Angela; Cagnotto, A. file da validare
New alkylpiperazines as 5-HT7R ligands 1-gen-2014 Intagliata, S; Modica, Maria Nunziata; Romeo, Giuseppe; Pittalà, V; Salerno, Loredana; Siracusa, Maria Angela; Cagnotto, A. file da validare
Thieno[3,2-d]pyrimidine as a scaffold for 5-HT7 receptor ligands 1-gen-2014 Romeo, Giuseppe; Modica, Maria Nunziata; Salerno, Loredana; Pittala', Valeria; Intagliata, S; Cagnotto, A; Salmona, M; Siracusa, Maria Angela file da validare
Structure-activity relationships and molecular modeling studies of novel arylpiperazinylalkyl 2-benzoxazolones and 2-benzothiazolones as 5-HT7 and 5-HT1A receptor ligands 1-gen-2014 Salerno, Loredana; Pittala', Valeria; Modica, Maria Nunziata; Siracusa, Maria Angela; Intagliata, S; Cagnotto, A; Salmona, M; Kurczab, R; Bojarski, A. J.; Romeo, Giuseppe
Synthesis and binding properties of new long-chain 4-substituted piperazine derivatives as 5-HT1A and 5-HT7 receptor ligands 1-gen-2015 Modica, Maria Nunziata; Intagliata, S; Pittala', Valeria; Salerno, Loredana; Siracusa, Maria Angela; Cagnotto, A; Salmona, M; Romeo, Giuseppe
New 5-Ht7 Receptor Ligands As Potential Antidepressant Agents. 1-gen-2015 Romeo, Giuseppe; Modica, Maria Nunziata; Salerno, Loredana; Pittala', Valeria; Siracusa, Maria Angela; Intagliata, Sebastiano; Marrazzo, Agostino; Prezzavento, Orazio; Amata, Emanuele; Cagnotto, Alfredo; Salmona, Mario file da validare
New alkylpiperazines as 5-HT7R ligands 8-dic-2015 Intagliata, Sebastiano
Novel selective ligands for the serotonergic 5-HT7 receptor: tricyclic derivatives Bearing the pyrimido-4(3H)-one ring 1-gen-2016 Romeo, Giuseppe; Pittala', Valeria; Salerno, Loredana; MODICA Maria, N; Candido, Margherita; Intagliata, Sebastiano; Marrazzo, Agostino; Amata, Emanuele; Cagnotto, A; Salmona, M; Siracusa, Maria Angela file da validare
Design and synthesis of new homo and hetero bis-piperazinyl-1- propanone derivatives as 5-HT7R selective ligands over 5-HT1AR 1-gen-2016 Intagliata, S; Modica, Maria Nunziata; Pittala', Valeria; Salerno, Loredana; Siracusa, Maria Angela; Cagnotto, A; Salmona, M; Romeo, Giuseppe
ATTIVITÀ ANTIOSSIDANTE IN VITRO DI DERIVATI DELL’IDEBENONE 1-gen-2017 Modica, Maria Nunziata; Salerno, Loredana; Intagliata, S; Romeo, Giuseppe; Pittala', Valeria; Panico, Anna Maria; Crascì, L; Puglisi, Giovanni; Montenegro, Lucia file da validare
New N- and O-arylpiperazinylalkyl pyrimidines and 2-methylquinazolines derivatives as 5-HT7 and 5-HT1A receptor ligands: Synthesis, structure-activity relationships, and molecular modeling studies 1-gen-2017 Intagliata, Sebastiano; Modica, Maria Nunziata; Pittala', Valeria; Salerno, Loredana; Siracusa, Maria Angela; Cagnotto, A; Salmona, M; Kurczab, R; Romeo, Giuseppe
New homo and hetero bis-arylpiperazine and bis-benzylpiperazine derivatives as 5-HT7R selective ligands: design and synthesis 1-gen-2018 Intagliata, Sebastiano; Pittalà, Valeria; Salerno, Loredana; Cagnotto, Alfredo; Romeo, Giuseppe; Amata, Emanuele; Marrazzo, Agostino; Modica Maria, N. file da validare
Design, synthesis, and pharmacological evaluation of NO donor-sigma receptors hybrids for the treatment of cancer 1-gen-2018 Dichiara, Maria; Barbaraci, Carla; Gentile, Davide; Intagliata, Sebastiano; Pittalà, Valeria; Arena, Emanuelea; Fraix, Aurore; Farina, Giuseppe; Prezzavento, Orazio; Amata, Emanuele; Marrazzo, Agostino.
Synthesis and in vitro antioxidant activity of a novel idebenone ester with pyroglutamic acid. 1-gen-2018 Montenegro, L; Intagliata, S; Salerno, L; Romeo, G; Pittalà, V; Siciliano, E; Panico, Am; Modica, Mn. file da validare
Structure-Activity Relationships and Therapeutic Potentials of 5-HT7 Receptor Ligands: An Update 1-gen-2018 Modica, Maria N.; Lacivita, Enza; Intagliata, Sebastiano; Salerno, Loredana; Romeo, Giuseppe; Pittalà, Valeria; Leopoldo, Marcello
Novel structural insight into inhibitors of heme oxygenase-1 (ho-1) by new imidazole-based compounds: Biochemical and in vitro anticancer activity evaluation 1-gen-2018 Greish F., Khaled; Salerno, Loredana; Zahrani Reem, Al; Amata, Emanuele; Modica, Maria Nunziata; Romeo, Giuseppe; Marrazzo, Agostino; Prezzavento, Orazio; Sorrenti, Valeria; Rescifina, Antonio; Floresta, Giuseppe; Intagliata, Sebastiano; Pittalà, Valeria
Targeting heme Oxygenase-1 with hybrid compounds to overcome Imatinib resistance in chronic myeloid leukemia cell lines 1-gen-2018 Sorrenti, Valeria; Pittalà, Valeria; Romeo, Giuseppe; Amata, Emanuele; Dichiara, Maria; Marrazzo, Agostino; Turnaturi, Rita; Prezzavento, Orazio; Barbagallo, Ignazio; Vanella, Luca; Rescifina, Antonio; Floresta, Giuseppe; Tibullo, Daniele; DI RAIMONDO, Francesco; Intagliata, Sebastiano; Salerno, Loredana
Solid lipid nanoparticles loading idebenone ester with pyroglutamic acid: In vitro antioxidant activity and in vivo topical efficacy 1-gen-2019 Montenegro, Lucia; Panico, Anna Maria; Santagati, Ludovica Maria; Siciliano, EDY ANGELA; Intagliata, Sebastiano; Modica, Maria N.
Synthesis, in vitro and in silico studies of HO-1 inducers and lung antifibrotic agents 1-gen-2019 Pittalà, Valeria; Vanella, Luca; Platania, CHIARA BIANCA MARIA; Salerno, Loredana; Raffaele, Marco; Amata, Emanuele; Marrazzo, Agostino; Floresta, Giuseppe; Romeo, Giuseppe; Greish F., Khaled; Intagliata, Sebastiano; Bucolo, Claudio; Sorrenti, Valeria
Protective Effects of Caffeic Acid Phenethyl Ester (CAPE) and Novel Cape Analogue as Inducers of Heme Oxygenase-1 in Streptozotocin-Induced Type 1 Diabetic Rats 1-gen-2019 Sorrenti, Valeria; Raffaele, Marco; Vanella, Luca; Acquaviva, Rosaria; Salerno, Loredana; Pittalà, Valeria; Intagliata, Sebastiano; Di Giacomo, Claudia
Mostrati risultati da 1 a 20 di 59
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