Sfoglia per Autore
New thienopyrimidine and quinazoline derivatives as potential 5-HT7 receptor ligands.
file da validare2013-01-01 Modica, Maria Nunziata; Intagliata, S; Romeo, Giuseppe; Pittala', Valeria; Salerno, Loredana; Siracusa, Maria Angela; Cagnotto, A.
New alkylpiperazines as 5-HT7R ligands
file da validare2014-01-01 Intagliata, S; Modica, Maria Nunziata; Romeo, Giuseppe; Pittalà, V; Salerno, Loredana; Siracusa, Maria Angela; Cagnotto, A.
Thieno[3,2-d]pyrimidine as a scaffold for 5-HT7 receptor ligands
file da validare2014-01-01 Romeo, Giuseppe; Modica, Maria Nunziata; Salerno, Loredana; Pittala', Valeria; Intagliata, S; Cagnotto, A; Salmona, M; Siracusa, Maria Angela
Structure-activity relationships and molecular modeling studies of novel arylpiperazinylalkyl 2-benzoxazolones and 2-benzothiazolones as 5-HT7 and 5-HT1A receptor ligands
2014-01-01 Salerno, Loredana; Pittala', Valeria; Modica, Maria Nunziata; Siracusa, Maria Angela; Intagliata, S; Cagnotto, A; Salmona, M; Kurczab, R; Bojarski, A. J.; Romeo, Giuseppe
Synthesis and binding properties of new long-chain 4-substituted piperazine derivatives as 5-HT1A and 5-HT7 receptor ligands
2015-01-01 Modica, Maria Nunziata; Intagliata, S; Pittala', Valeria; Salerno, Loredana; Siracusa, Maria Angela; Cagnotto, A; Salmona, M; Romeo, Giuseppe
New 5-Ht7 Receptor Ligands As Potential Antidepressant Agents.
file da validare2015-01-01 Romeo, Giuseppe; Modica, Maria Nunziata; Salerno, Loredana; Pittala', Valeria; Siracusa, Maria Angela; Intagliata, Sebastiano; Marrazzo, Agostino; Prezzavento, Orazio; Amata, Emanuele; Cagnotto, Alfredo; Salmona, Mario
New alkylpiperazines as 5-HT7R ligands
2015-12-08 Intagliata, Sebastiano
Novel selective ligands for the serotonergic 5-HT7 receptor: tricyclic derivatives Bearing the pyrimido-4(3H)-one ring
file da validare2016-01-01 Romeo, Giuseppe; Pittala', Valeria; Salerno, Loredana; MODICA Maria, N; Candido, Margherita; Intagliata, Sebastiano; Marrazzo, Agostino; Amata, Emanuele; Cagnotto, A; Salmona, M; Siracusa, Maria Angela
Design and synthesis of new homo and hetero bis-piperazinyl-1- propanone derivatives as 5-HT7R selective ligands over 5-HT1AR
2016-01-01 Intagliata, S; Modica, Maria Nunziata; Pittala', Valeria; Salerno, Loredana; Siracusa, Maria Angela; Cagnotto, A; Salmona, M; Romeo, Giuseppe
ATTIVITÀ ANTIOSSIDANTE IN VITRO DI DERIVATI DELL’IDEBENONE
file da validare2017-01-01 Modica, Maria Nunziata; Salerno, Loredana; Intagliata, S; Romeo, Giuseppe; Pittala', Valeria; Panico, Anna Maria; Crascì, L; Puglisi, Giovanni; Montenegro, Lucia
New N- and O-arylpiperazinylalkyl pyrimidines and 2-methylquinazolines derivatives as 5-HT7 and 5-HT1A receptor ligands: Synthesis, structure-activity relationships, and molecular modeling studies
2017-01-01 Intagliata, Sebastiano; Modica, Maria Nunziata; Pittala', Valeria; Salerno, Loredana; Siracusa, Maria Angela; Cagnotto, A; Salmona, M; Kurczab, R; Romeo, Giuseppe
New homo and hetero bis-arylpiperazine and bis-benzylpiperazine derivatives as 5-HT7R selective ligands: design and synthesis
file da validare2018-01-01 Intagliata, Sebastiano; Pittalà, Valeria; Salerno, Loredana; Cagnotto, Alfredo; Romeo, Giuseppe; Amata, Emanuele; Marrazzo, Agostino; Modica Maria, N.
Design, synthesis, and pharmacological evaluation of NO donor-sigma receptors hybrids for the treatment of cancer
2018-01-01 Dichiara, Maria; Barbaraci, Carla; Gentile, Davide; Intagliata, Sebastiano; Pittalà, Valeria; Arena, Emanuelea; Fraix, Aurore; Farina, Giuseppe; Prezzavento, Orazio; Amata, Emanuele; Marrazzo, Agostino.
Synthesis and in vitro antioxidant activity of a novel idebenone ester with pyroglutamic acid.
file da validare2018-01-01 Montenegro, L; Intagliata, S; Salerno, L; Romeo, G; Pittalà, V; Siciliano, E; Panico, Am; Modica, Mn.
Structure-Activity Relationships and Therapeutic Potentials of 5-HT7 Receptor Ligands: An Update
2018-01-01 Modica, Maria N.; Lacivita, Enza; Intagliata, Sebastiano; Salerno, Loredana; Romeo, Giuseppe; Pittalà, Valeria; Leopoldo, Marcello
Novel structural insight into inhibitors of heme oxygenase-1 (ho-1) by new imidazole-based compounds: Biochemical and in vitro anticancer activity evaluation
2018-01-01 Greish F., Khaled; Salerno, Loredana; Zahrani Reem, Al; Amata, Emanuele; Modica, Maria Nunziata; Romeo, Giuseppe; Marrazzo, Agostino; Prezzavento, Orazio; Sorrenti, Valeria; Rescifina, Antonio; Floresta, Giuseppe; Intagliata, Sebastiano; Pittalà, Valeria
Targeting heme Oxygenase-1 with hybrid compounds to overcome Imatinib resistance in chronic myeloid leukemia cell lines
2018-01-01 Sorrenti, Valeria; Pittalà, Valeria; Romeo, Giuseppe; Amata, Emanuele; Dichiara, Maria; Marrazzo, Agostino; Turnaturi, Rita; Prezzavento, Orazio; Barbagallo, Ignazio; Vanella, Luca; Rescifina, Antonio; Floresta, Giuseppe; Tibullo, Daniele; DI RAIMONDO, Francesco; Intagliata, Sebastiano; Salerno, Loredana
Solid lipid nanoparticles loading idebenone ester with pyroglutamic acid: In vitro antioxidant activity and in vivo topical efficacy
2019-01-01 Montenegro, Lucia; Panico, Anna Maria; Santagati, Ludovica Maria; Siciliano, EDY ANGELA; Intagliata, Sebastiano; Modica, Maria N.
Synthesis, in vitro and in silico studies of HO-1 inducers and lung antifibrotic agents
2019-01-01 Pittalà, Valeria; Vanella, Luca; Platania, CHIARA BIANCA MARIA; Salerno, Loredana; Raffaele, Marco; Amata, Emanuele; Marrazzo, Agostino; Floresta, Giuseppe; Romeo, Giuseppe; Greish F., Khaled; Intagliata, Sebastiano; Bucolo, Claudio; Sorrenti, Valeria
Protective Effects of Caffeic Acid Phenethyl Ester (CAPE) and Novel Cape Analogue as Inducers of Heme Oxygenase-1 in Streptozotocin-Induced Type 1 Diabetic Rats
2019-01-01 Sorrenti, Valeria; Raffaele, Marco; Vanella, Luca; Acquaviva, Rosaria; Salerno, Loredana; Pittalà, Valeria; Intagliata, Sebastiano; Di Giacomo, Claudia
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
New thienopyrimidine and quinazoline derivatives as potential 5-HT7 receptor ligands. | 1-gen-2013 | Modica, Maria Nunziata; Intagliata, S; Romeo, Giuseppe; Pittala', Valeria; Salerno, Loredana; Siracusa, Maria Angela; Cagnotto, A. | file da validare |
New alkylpiperazines as 5-HT7R ligands | 1-gen-2014 | Intagliata, S; Modica, Maria Nunziata; Romeo, Giuseppe; Pittalà, V; Salerno, Loredana; Siracusa, Maria Angela; Cagnotto, A. | file da validare |
Thieno[3,2-d]pyrimidine as a scaffold for 5-HT7 receptor ligands | 1-gen-2014 | Romeo, Giuseppe; Modica, Maria Nunziata; Salerno, Loredana; Pittala', Valeria; Intagliata, S; Cagnotto, A; Salmona, M; Siracusa, Maria Angela | file da validare |
Structure-activity relationships and molecular modeling studies of novel arylpiperazinylalkyl 2-benzoxazolones and 2-benzothiazolones as 5-HT7 and 5-HT1A receptor ligands | 1-gen-2014 | Salerno, Loredana; Pittala', Valeria; Modica, Maria Nunziata; Siracusa, Maria Angela; Intagliata, S; Cagnotto, A; Salmona, M; Kurczab, R; Bojarski, A. J.; Romeo, Giuseppe | |
Synthesis and binding properties of new long-chain 4-substituted piperazine derivatives as 5-HT1A and 5-HT7 receptor ligands | 1-gen-2015 | Modica, Maria Nunziata; Intagliata, S; Pittala', Valeria; Salerno, Loredana; Siracusa, Maria Angela; Cagnotto, A; Salmona, M; Romeo, Giuseppe | |
New 5-Ht7 Receptor Ligands As Potential Antidepressant Agents. | 1-gen-2015 | Romeo, Giuseppe; Modica, Maria Nunziata; Salerno, Loredana; Pittala', Valeria; Siracusa, Maria Angela; Intagliata, Sebastiano; Marrazzo, Agostino; Prezzavento, Orazio; Amata, Emanuele; Cagnotto, Alfredo; Salmona, Mario | file da validare |
New alkylpiperazines as 5-HT7R ligands | 8-dic-2015 | Intagliata, Sebastiano | |
Novel selective ligands for the serotonergic 5-HT7 receptor: tricyclic derivatives Bearing the pyrimido-4(3H)-one ring | 1-gen-2016 | Romeo, Giuseppe; Pittala', Valeria; Salerno, Loredana; MODICA Maria, N; Candido, Margherita; Intagliata, Sebastiano; Marrazzo, Agostino; Amata, Emanuele; Cagnotto, A; Salmona, M; Siracusa, Maria Angela | file da validare |
Design and synthesis of new homo and hetero bis-piperazinyl-1- propanone derivatives as 5-HT7R selective ligands over 5-HT1AR | 1-gen-2016 | Intagliata, S; Modica, Maria Nunziata; Pittala', Valeria; Salerno, Loredana; Siracusa, Maria Angela; Cagnotto, A; Salmona, M; Romeo, Giuseppe | |
ATTIVITÀ ANTIOSSIDANTE IN VITRO DI DERIVATI DELL’IDEBENONE | 1-gen-2017 | Modica, Maria Nunziata; Salerno, Loredana; Intagliata, S; Romeo, Giuseppe; Pittala', Valeria; Panico, Anna Maria; Crascì, L; Puglisi, Giovanni; Montenegro, Lucia | file da validare |
New N- and O-arylpiperazinylalkyl pyrimidines and 2-methylquinazolines derivatives as 5-HT7 and 5-HT1A receptor ligands: Synthesis, structure-activity relationships, and molecular modeling studies | 1-gen-2017 | Intagliata, Sebastiano; Modica, Maria Nunziata; Pittala', Valeria; Salerno, Loredana; Siracusa, Maria Angela; Cagnotto, A; Salmona, M; Kurczab, R; Romeo, Giuseppe | |
New homo and hetero bis-arylpiperazine and bis-benzylpiperazine derivatives as 5-HT7R selective ligands: design and synthesis | 1-gen-2018 | Intagliata, Sebastiano; Pittalà, Valeria; Salerno, Loredana; Cagnotto, Alfredo; Romeo, Giuseppe; Amata, Emanuele; Marrazzo, Agostino; Modica Maria, N. | file da validare |
Design, synthesis, and pharmacological evaluation of NO donor-sigma receptors hybrids for the treatment of cancer | 1-gen-2018 | Dichiara, Maria; Barbaraci, Carla; Gentile, Davide; Intagliata, Sebastiano; Pittalà, Valeria; Arena, Emanuelea; Fraix, Aurore; Farina, Giuseppe; Prezzavento, Orazio; Amata, Emanuele; Marrazzo, Agostino. | |
Synthesis and in vitro antioxidant activity of a novel idebenone ester with pyroglutamic acid. | 1-gen-2018 | Montenegro, L; Intagliata, S; Salerno, L; Romeo, G; Pittalà, V; Siciliano, E; Panico, Am; Modica, Mn. | file da validare |
Structure-Activity Relationships and Therapeutic Potentials of 5-HT7 Receptor Ligands: An Update | 1-gen-2018 | Modica, Maria N.; Lacivita, Enza; Intagliata, Sebastiano; Salerno, Loredana; Romeo, Giuseppe; Pittalà, Valeria; Leopoldo, Marcello | |
Novel structural insight into inhibitors of heme oxygenase-1 (ho-1) by new imidazole-based compounds: Biochemical and in vitro anticancer activity evaluation | 1-gen-2018 | Greish F., Khaled; Salerno, Loredana; Zahrani Reem, Al; Amata, Emanuele; Modica, Maria Nunziata; Romeo, Giuseppe; Marrazzo, Agostino; Prezzavento, Orazio; Sorrenti, Valeria; Rescifina, Antonio; Floresta, Giuseppe; Intagliata, Sebastiano; Pittalà, Valeria | |
Targeting heme Oxygenase-1 with hybrid compounds to overcome Imatinib resistance in chronic myeloid leukemia cell lines | 1-gen-2018 | Sorrenti, Valeria; Pittalà, Valeria; Romeo, Giuseppe; Amata, Emanuele; Dichiara, Maria; Marrazzo, Agostino; Turnaturi, Rita; Prezzavento, Orazio; Barbagallo, Ignazio; Vanella, Luca; Rescifina, Antonio; Floresta, Giuseppe; Tibullo, Daniele; DI RAIMONDO, Francesco; Intagliata, Sebastiano; Salerno, Loredana | |
Solid lipid nanoparticles loading idebenone ester with pyroglutamic acid: In vitro antioxidant activity and in vivo topical efficacy | 1-gen-2019 | Montenegro, Lucia; Panico, Anna Maria; Santagati, Ludovica Maria; Siciliano, EDY ANGELA; Intagliata, Sebastiano; Modica, Maria N. | |
Synthesis, in vitro and in silico studies of HO-1 inducers and lung antifibrotic agents | 1-gen-2019 | Pittalà, Valeria; Vanella, Luca; Platania, CHIARA BIANCA MARIA; Salerno, Loredana; Raffaele, Marco; Amata, Emanuele; Marrazzo, Agostino; Floresta, Giuseppe; Romeo, Giuseppe; Greish F., Khaled; Intagliata, Sebastiano; Bucolo, Claudio; Sorrenti, Valeria | |
Protective Effects of Caffeic Acid Phenethyl Ester (CAPE) and Novel Cape Analogue as Inducers of Heme Oxygenase-1 in Streptozotocin-Induced Type 1 Diabetic Rats | 1-gen-2019 | Sorrenti, Valeria; Raffaele, Marco; Vanella, Luca; Acquaviva, Rosaria; Salerno, Loredana; Pittalà, Valeria; Intagliata, Sebastiano; Di Giacomo, Claudia |
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