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Mostrati risultati da 1 a 20 di 145
Titolo Data di pubblicazione Autore(i) File
Synthesis of piperazinyl-alkylthiothieno[2,3-d]pyrimidine derivatives and serotonergic activity avaluation 1-gen-1992 Modica, Maria Nunziata; Santagati, M; Santagati, A; Russo, F. file da validare
A new heterocyclic ring system: synthesis of pyrazolo[3',4':4,5]pyrimido-[2,1-a]phthalazine derivatives 1-gen-1992 Santagati, M; Santagati, A; Modica, Maria Nunziata; Russo, F. file da validare
Synthesis of 2,3,5,6,7,8-hexahydro-3-amino-thioxo[1]benzothieno[2,3-d]-pyrimidin-4(1H)-one and derivatives of the new heterocyclic system 7,8,9,10-tetrahydro-3H,11H-[1]benzothieno[2',3':4,5]pyrimido[2,1-b][1,3,4]-thiadiazin-11-one 1-gen-1993 Santagati, A; Santagati, M; Modica, Maria Nunziata file da validare
Synthesis of 2,3-dihydro-3-amino-6-phenyl-2-thioxothieno[2,3-d]pyrimidin-4(1H)-one and of potential antiinflammatory agents 2-aryl-7-phenyl-3H,9H-pyrimido[2,1-b]thieno[2',3':4,5][1,3,4]thiadiazin-9-ones 1-gen-1994 Santagati, A; Modica, Maria Nunziata; Santagati, M; Caruso, A; Cutuli, V. file da validare
Synthesis and pharmacological properties of benzothiazole, 1,3,4-oxadiazole and 1,3,4-thiadiazole derivatives 1-gen-1994 Santagati, M; Modica, Maria Nunziata; Santagati, A; Russo, F; Caruso, A; Cutuli, V; DI PIETRO, E; AMICO ROXAS, M. file da validare
Study on the tachykinins antagonist effect of combinatorial functionalized heterocycle replacements in tryciclic pyrimidine derivatives 1-gen-1994 Guccione, Salvatore; Modica, Maria Nunziata; Shaw, D; UCCELLO BARRETTA, G; Santagati, A; Santagati, M. file da validare
Bridgehead nitrogen heterocycles derived from the potassium salt of 2,3,5,6,7,8-hexahydro-3-amino-2-thioxo-[1]benzothieno[2,3-d]pyrimidin-4(1H)-one 1-gen-1994 Santagati, A; Modica, Maria Nunziata; Santagati, M. file da validare
Synthesis and pharmacological properties of thieno[2',3':4,5]pyrimido[2,1-b][1,3,4]thiadiazine derivatives 1-gen-1995 Santagati, A; Modica, Maria Nunziata; Santagati, M; Cutuli, V; Amore, D; Caruso, A. file da validare
CoMFA contributions to a binding mode for NK2 receptor antagonists 1-gen-1995 Guccione, Salvatore; Santagati, M; Santagati, A; Modica, Maria Nunziata; UCCELLO BARRETTA, G; Langer, T; Russo, F. file da validare
Potential of indole skeleton containing heterocycles as antagonists at the neurokinin (NK) receptor system 1-gen-1995 Modica, Maria Nunziata; Santagati, A; Santagati, M; MONSU’ SCOLARO, L; Guccione, Salvatore; Russo, F. file da validare
Synthesis and NK-2 antagonist effect of 1,6-diphenyl-pyrazolo [3, 4-d]-thiazolo[3,2-a]4H-pyrimidin-4-one 1-gen-1996 Guccione, Salvatore; Modica, Maria Nunziata; J., Longmore; D., Shaw; G., UCCELLO BARRETTA; A., Santagati; M., Santagati; F., Russo file da validare
Synthesis of aminothienopyrimidine and thienotriazolopyrimidine derivatives as potential anticonvulsant agents 1-gen-1996 Santagati, M; Modica, Maria Nunziata; Santagati, A; Russo, F; Spampinato, S. file da validare
Synthesis of 1-phenyl-6-arilsubstituted pyrazolopyrimidothiazole as antagonists at the NK-2 receptors 1-gen-1997 Russo, F; Longmore, J; Modica, Maria Nunziata; Santagati, M; Santagati, A; Guccione, Salvatore file da validare
[[(Arylpiperazinyl)alkylthio]thieno[2,3-d]pyrimidinone derivatives as high-affinity, selective 5-HT1A receptor ligands 1-gen-1997 Modica, Maria Nunziata; Santagati, M; Russo, F; Parotti, L; DE GIOIA, L; Selvaggini, C; Salmona, M; Mennini, T. file da validare
5-HT1A receptors mapping by conformational analysis (2D NOESY/MM) and ”three way modelling” (HASL, CoMFA, PARM) 1-gen-1998 Santagati, M; Doweyko, A; Santagati, A; Modica, Maria Nunziata; Guccione, Salvatore; Chen, H. M.; Uccello Barretta, G; Balzano, F. file da validare
5-HT1A receptors mapping by conformational analysis (2D NOESY/MM) and "tree way modelling" (HASL, CoMFA, PARM) 1-gen-1998 Santagati, M; Doweyko, A; Santagati, A; Modica, Maria Nunziata; Guccione, Salvatore; Chen, H; Russo, F; UCCELLO BARRETTA, G; Balzano, F. file da validare
Application of PARM to constructing and comparing 5-HT1A and alfa1 receptor models 1-gen-1998 Santagati, M; Chen, H; Santagati, A; Modica, Maria Nunziata; Guccione, Salvatore; Uccello Barretta, G; Balzano, F. file da validare
Building a model of interaction at the NK-2 receptors: polycondensed heterocycles containing the pyrimidoindole skeleton 1-gen-1998 Santagati, A; Longmore, J; Guccione, Salvatore; Langer, T; Tonnel, E; Modica, Maria Nunziata; Santagati, M; MONSU’ SCOLARO, L; Russo, F. file da validare
Application of Parm to constructing and comparing 5-HT1A and alfa1 receptor models 1-gen-1998 Santagati, M; Chen, H; Santagati, A; Modica, Maria Nunziata; Guccione, Salvatore; Russo, F; UCCELLO BARRETTA, G; Balzano, F. file da validare
Design and synthesis of new high-affinity, selective 5-HT1A receptor ligands 1-gen-1999 Modica, Maria Nunziata; Santagati, M; Santagati, A; Russo, F; Cagnotto, A; Goegan, M; Mennini, T. file da validare
Mostrati risultati da 1 a 20 di 145
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