Sfoglia per Autore
New selective Sigma-1/HDACi prodrugs for neurodegenerative disorders
2018-01-01 Barbaraci, Carla; Dichiara, Maria; Turnaturi, Rita; Fallica Antonino, N; Arena, Emanuela; Prezzavento, Orazio; Amata, Emanuele; Marrazzo, Agostino
A structure-and ligand-based virtual screening of a database of “small” marine natural products for the identification of “blue” sigma-2 receptor ligands
2018-01-01 Floresta, Giuseppe; Amata, Emanuele; Barbaraci, Carla; Gentile, Davide; Turnaturi, Rita; Marrazzo, Agostino; Rescifina, Antonio
Design, synthesis, and pharmacological evaluation of NO donor-sigma receptors hybrids for the treatment of cancer
2018-01-01 Dichiara, Maria; Barbaraci, Carla; Gentile, Davide; Intagliata, Sebastiano; Pittalà, Valeria; Arena, Emanuelea; Fraix, Aurore; Farina, Giuseppe; Prezzavento, Orazio; Amata, Emanuele; Marrazzo, Agostino.
Synthesis of “no-light activated” Ciprofloxacin and Norfloxacin derivatives as potential biofilm dispersant agents
2019-01-01 Fallica, Antonino N.; Ciaffaglione, Valeria; Leonardi, Carmen; Dichiara, Maria; Barbaraci, Carla; Catalfo, Alfio; Finocchiaro, GUGLIELMO MARTINO; DE GUIDI, Guido; Amata, Emanuele; Marrazzo, Agostino
Development of novel H2S-donor sigma receptor hybrids for the management of pain.
2019-01-01 Dichiara, Maria; Pitino, Cristina; Barbaraci, Carla; Artacho-Cordón, A.; Cobos Enrique, J; Marrazzo, Agostino; Amata, Emanuele
Nitric Oxide Photo-Donor Hybrids of Ciprofloxacin and Norfloxacin: A Shift in Activity from Antimicrobial to Anticancer Agents
2021-01-01 Fallica, A. N.; Barbaraci, C.; Amata, E.; Pasquinucci, L.; Turnaturi, R.; Dichiara, M.; Intagliata, S.; Gariboldi, M. B.; Marras, E.; Orlandi, V. T.; Ferroni, C.; Martini, C.; Rescifina, A.; Gentile, D.; Varchi, G.; Marrazzo, A.
Haloperidol Metabolite II Valproate Ester ( S)-(-)-MRJF22: Preliminary Studies as a Potential Multifunctional Agent Against Uveal Melanoma
2021-01-01 Barbaraci, Carla; Giurdanella, Giovanni; Leotta, CLAUDIA GIOVANNA; Longo, ANNA MARIA; Amata, Emanuele; Dichiara, Maria; Pasquinucci, Lorella Giuseppina; Turnaturi, Rita; Prezzavento, Orazio; Cacciatore, Ivana; Zuccarello, Elisa; Lupo, Gabriella; Mario Pitari, Giovanni; Anfuso, CARMELINA DANIELA; Marrazzo, Agostino
Interaction of new sigma ligands with biomembrane models evaluated by differential scanning calorimetry and Langmuir-Blodgett studies
2021-01-01 Marrazzo, A.; Torrisi, C.; Barbaraci, C.; Amata, E.; Castelli, F.; Sarpietro, M. G.
Dual Sigma-1 receptor antagonists and hydrogen sulfide-releasing compounds for pain treatment: Design, synthesis, and pharmacological evaluation
2022-01-01 Dichiara, Maria; Artacho-Cordon, Antonia; Turnaturi, Rita; Santos-Caballero, Miriam; Gonzalez-Cano, Rafael; Pasquinucci, Lorella; Barbaraci, Carla; Rodriguez-Gomez, Isabel; Gomez-Guzman, Manuel; Marrazzo, Agostino; Cobos Enrique, J.; Amata, Emanuele.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
New selective Sigma-1/HDACi prodrugs for neurodegenerative disorders | 1-gen-2018 | Barbaraci, Carla; Dichiara, Maria; Turnaturi, Rita; Fallica Antonino, N; Arena, Emanuela; Prezzavento, Orazio; Amata, Emanuele; Marrazzo, Agostino | |
A structure-and ligand-based virtual screening of a database of “small” marine natural products for the identification of “blue” sigma-2 receptor ligands | 1-gen-2018 | Floresta, Giuseppe; Amata, Emanuele; Barbaraci, Carla; Gentile, Davide; Turnaturi, Rita; Marrazzo, Agostino; Rescifina, Antonio | |
Design, synthesis, and pharmacological evaluation of NO donor-sigma receptors hybrids for the treatment of cancer | 1-gen-2018 | Dichiara, Maria; Barbaraci, Carla; Gentile, Davide; Intagliata, Sebastiano; Pittalà, Valeria; Arena, Emanuelea; Fraix, Aurore; Farina, Giuseppe; Prezzavento, Orazio; Amata, Emanuele; Marrazzo, Agostino. | |
Synthesis of “no-light activated” Ciprofloxacin and Norfloxacin derivatives as potential biofilm dispersant agents | 1-gen-2019 | Fallica, Antonino N.; Ciaffaglione, Valeria; Leonardi, Carmen; Dichiara, Maria; Barbaraci, Carla; Catalfo, Alfio; Finocchiaro, GUGLIELMO MARTINO; DE GUIDI, Guido; Amata, Emanuele; Marrazzo, Agostino | |
Development of novel H2S-donor sigma receptor hybrids for the management of pain. | 1-gen-2019 | Dichiara, Maria; Pitino, Cristina; Barbaraci, Carla; Artacho-Cordón, A.; Cobos Enrique, J; Marrazzo, Agostino; Amata, Emanuele | |
Nitric Oxide Photo-Donor Hybrids of Ciprofloxacin and Norfloxacin: A Shift in Activity from Antimicrobial to Anticancer Agents | 1-gen-2021 | Fallica, A. N.; Barbaraci, C.; Amata, E.; Pasquinucci, L.; Turnaturi, R.; Dichiara, M.; Intagliata, S.; Gariboldi, M. B.; Marras, E.; Orlandi, V. T.; Ferroni, C.; Martini, C.; Rescifina, A.; Gentile, D.; Varchi, G.; Marrazzo, A. | |
Haloperidol Metabolite II Valproate Ester ( S)-(-)-MRJF22: Preliminary Studies as a Potential Multifunctional Agent Against Uveal Melanoma | 1-gen-2021 | Barbaraci, Carla; Giurdanella, Giovanni; Leotta, CLAUDIA GIOVANNA; Longo, ANNA MARIA; Amata, Emanuele; Dichiara, Maria; Pasquinucci, Lorella Giuseppina; Turnaturi, Rita; Prezzavento, Orazio; Cacciatore, Ivana; Zuccarello, Elisa; Lupo, Gabriella; Mario Pitari, Giovanni; Anfuso, CARMELINA DANIELA; Marrazzo, Agostino | |
Interaction of new sigma ligands with biomembrane models evaluated by differential scanning calorimetry and Langmuir-Blodgett studies | 1-gen-2021 | Marrazzo, A.; Torrisi, C.; Barbaraci, C.; Amata, E.; Castelli, F.; Sarpietro, M. G. | |
Dual Sigma-1 receptor antagonists and hydrogen sulfide-releasing compounds for pain treatment: Design, synthesis, and pharmacological evaluation | 1-gen-2022 | Dichiara, Maria; Artacho-Cordon, Antonia; Turnaturi, Rita; Santos-Caballero, Miriam; Gonzalez-Cano, Rafael; Pasquinucci, Lorella; Barbaraci, Carla; Rodriguez-Gomez, Isabel; Gomez-Guzman, Manuel; Marrazzo, Agostino; Cobos Enrique, J.; Amata, Emanuele. |
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