Sfoglia per Autore
Development of new benzomorphan LP1 analogues
file da validare2008-01-01 Pasquinucci, Lorella Giuseppina; Amata, Emanuele; Ronsisvalle, Giuseppe
In-vitro evaluation of a new benzomorphan-based ligand
2009-01-01 Pasquinucci, Lorella Giuseppina; Prezzavento, Orazio; Amata, Emanuele; Ronsisvalle, Simone; Parenti, Carmela; Aricò, Giuseppina; Iemolo, Attilio; SCOTO Giovanna, M; Georgoussi, Zafiroula; Ronsisvalle, Giuseppe
Design and synthesis of new benzomorphan LP1 analogues, an opioid ligand with low development of tolerance
file da validare2009-01-01 Amata, Emanuele
Pain management: new long-acting opioid ligands
file da validare2009-01-01 Prezzavento, Orazio; Amata, Emanuele; Ronsisvalle, Simone; Parenti, Carmela; Aricò, Giuseppina; Scoto Giovanna, M.; Ronsisvalle, Giuseppe
Synthesis and in vitro opioid receptor studies on benzomorphan-based compounds: LP1, a potent and long-acting antinociceptive
2009-01-01 Pasquinucci, Lorella Giuseppina; Prezzavento, Orazio; Amata, Emanuele; Arena, Emanuela; Ronsisvalle, Simone; Parenti, Carmela; Arico, Giuseppina; Scoto, Giovanna M; Ronsisvalle, Giuseppe
In vitro and in vivo pharmacological evaluation of LP1, a benzomorphan-based compound
file da validare2009-01-01 Iemolo, Attilio; Parenti, Carmela; Aricò, Giuseppina; Al-Khrasani, Mahmoud; Amata, Emanuele; Scoto Giovanna, M.; Ronsisvalle, Giuseppe; Pasquinucci, Lorella
Evaluation of N-substitution in 6,7-benzomorphan compounds
2010-01-01 Pasquinucci, Lorella; Prezzavento, Orazio; Marrazzo, Agostino; Amata, Emanuele; Ronsisvalle, Simone; Georgoussi, Zafiroula; Fourla, Danai-Dionysia; Scoto M., Giovanna; Parenti, Carmela; Aricò, Giuseppina; Ronsisvalle, Giuseppe
Synthesis and pharmacological evaluation of indole-based sigma receptor ligands
2011-01-01 Mesangeau, Christophe; Amata, Emanuele; Alsharif, Walid; Seminerio J., Michael; Robson J., Matthew; Matsumoto R., Rae; Poupaert H., Jacques; McCurdy R., Christopher
Evaluation of human PDE4 inhibitors cilomilast and piclamilast as lead compounds for the treatment of human African trypanosomiasis (HAT)
file da validare2012-01-01 Amata, Emanuele; Woodring, J; Ochiana, So; Bland, Nd; Gustafson, A; Campbell, Rk; Pollastri, Mp
Preparation and Evaluation of a Series of Indoles as Sigma Receptor Ligands
file da validare2012-01-01 Alsharif, W; Mesangeau, C; Matsumoto, Rr; Seminerio, Mj; M., Robson M; Poupaert, Jh; Amata, Emanuele; Mccurdy, Cr
Neglected disease lead discovery: Profiling analogs of Lapatinib against the protozoan parasites that cause Chagas disease, leishmaniasis, and malaria
file da validare2012-01-01 Amata, Emanuele; Devine, W; Mehta, N; Swaminathan, U; Rodriguez, A; Erath, J.; Andriani, G; Sciotti, R; Pollastri, Mp
Targeting Neglected Parasitic Diseases with Human EGFR Inhibitor Chemotypes
file da validare2013-01-01 Woodring, J. L.; Patel, G.; Amata, Emanuele; Sciotti, R.; Rodriguez, A.; Pollastri, M. P.
Antitrypanosomal lead discovery: Identification of a ligand-efficient inhibitor of Trypanosoma cruzi CYP51 and parasite growth
2013-01-01 Andriani, Grasiella; Amata, Emanuele; Beatty, Joel; Clements, Zeke; Coffey J., Brian; Courtemanche, Gilles; Devine, William; Erath, Jessey; Juda E., Cristin; Wawrzak, Zdzislaw; Wood T., Jodianne; Lepesheva L., Galina; Rodriguez, Ana; Pollastri P., Michael
Involvement of sigma 2 receptor on motor disorder
file da validare2014-01-01 Aricò, G; Ronsisvalle, N; Cova, Am; Blanco, P; Amata, Emanuele; Parenti, Carmela; Ronsisvalle, Simone
Repurposing human PDE4 inhibitors for neglected tropical diseases: design, synthesis and evaluation of cilomilast analogues as Trypanosoma brucei PDEB1 inhibitors
file da validare2014-01-01 Amata, Emanuele; Bland D., Nicholas; Hoyt T., Charles; Settimo, Luca; Campbell K., Robert; Pollastri P., Michael
Identification and characterization of hundreds of potent and selective inhibitors of Trypanosoma brucei growth from a kinase-targeted library screening campaign
2014-01-01 Diaz, Rosario; Luengo-Arratta A., Sandra; Seixas D., João; Amata, Emanuele; Devine, William; Cordon-Obras, Carlos; Rojas-Barros L., Domingo; Jimenez, Elena; Ortega, Fatima; Crouch, Sabrinia; Colmenarejo, Gonzalo; Fiandor Jose, Maria; Martin Jose, Julio; Berlanga, Manuela; Gonzalez, Silvia; Manzano, Pilar; Navarro, Miguel; Pollastri P., Michael
Antioxidant activity of (+)-Pentazocine on activated microglia
file da validare2015-01-01 Marrazzo, Agostino; Heiss, Kathrin; Prezzavento, Orazio; Arena, Emanuela; Amata, Emanuele; LI VOLTI, Giovanni
New 5-Ht7 Receptor Ligands As Potential Antidepressant Agents.
file da validare2015-01-01 Romeo, Giuseppe; Modica, Maria Nunziata; Salerno, Loredana; Pittala', Valeria; Siracusa, Maria Angela; Intagliata, Sebastiano; Marrazzo, Agostino; Prezzavento, Orazio; Amata, Emanuele; Cagnotto, Alfredo; Salmona, Mario
Antioxidant properties and pharmacokinetic studies of new selective σ1 bifunctional ligands
file da validare2015-01-01 Marrazzo, Agostino; Arena, Emanuela; Cacciatore, Ivana; Cerasa Laura, S.; Amata, Emanuele; Pittala', Valeria; Pasquinucci, Lorella Giuseppina; Turkez, Hasan; Di Stefano, Antonio; Prezzavento, Orazio
C-5'-Triazolyl-2'-oxa-3'-aza-4'a-carbanucleosides: Synthesis and biological evaluation
2015-01-01 Romeo, Roberto; Carnovale, Caterina; Giofrè V., Salvatore; Chiacchio, MARIA ASSUNTA ROSSELLA; Garozzo, Adriana; Amata, Emanuele; Romeo, Giovanni; Chiacchio, Ugo
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Development of new benzomorphan LP1 analogues | 1-gen-2008 | Pasquinucci, Lorella Giuseppina; Amata, Emanuele; Ronsisvalle, Giuseppe | file da validare |
In-vitro evaluation of a new benzomorphan-based ligand | 1-gen-2009 | Pasquinucci, Lorella Giuseppina; Prezzavento, Orazio; Amata, Emanuele; Ronsisvalle, Simone; Parenti, Carmela; Aricò, Giuseppina; Iemolo, Attilio; SCOTO Giovanna, M; Georgoussi, Zafiroula; Ronsisvalle, Giuseppe | |
Design and synthesis of new benzomorphan LP1 analogues, an opioid ligand with low development of tolerance | 1-gen-2009 | Amata, Emanuele | file da validare |
Pain management: new long-acting opioid ligands | 1-gen-2009 | Prezzavento, Orazio; Amata, Emanuele; Ronsisvalle, Simone; Parenti, Carmela; Aricò, Giuseppina; Scoto Giovanna, M.; Ronsisvalle, Giuseppe | file da validare |
Synthesis and in vitro opioid receptor studies on benzomorphan-based compounds: LP1, a potent and long-acting antinociceptive | 1-gen-2009 | Pasquinucci, Lorella Giuseppina; Prezzavento, Orazio; Amata, Emanuele; Arena, Emanuela; Ronsisvalle, Simone; Parenti, Carmela; Arico, Giuseppina; Scoto, Giovanna M; Ronsisvalle, Giuseppe | |
In vitro and in vivo pharmacological evaluation of LP1, a benzomorphan-based compound | 1-gen-2009 | Iemolo, Attilio; Parenti, Carmela; Aricò, Giuseppina; Al-Khrasani, Mahmoud; Amata, Emanuele; Scoto Giovanna, M.; Ronsisvalle, Giuseppe; Pasquinucci, Lorella | file da validare |
Evaluation of N-substitution in 6,7-benzomorphan compounds | 1-gen-2010 | Pasquinucci, Lorella; Prezzavento, Orazio; Marrazzo, Agostino; Amata, Emanuele; Ronsisvalle, Simone; Georgoussi, Zafiroula; Fourla, Danai-Dionysia; Scoto M., Giovanna; Parenti, Carmela; Aricò, Giuseppina; Ronsisvalle, Giuseppe | |
Synthesis and pharmacological evaluation of indole-based sigma receptor ligands | 1-gen-2011 | Mesangeau, Christophe; Amata, Emanuele; Alsharif, Walid; Seminerio J., Michael; Robson J., Matthew; Matsumoto R., Rae; Poupaert H., Jacques; McCurdy R., Christopher | |
Evaluation of human PDE4 inhibitors cilomilast and piclamilast as lead compounds for the treatment of human African trypanosomiasis (HAT) | 1-gen-2012 | Amata, Emanuele; Woodring, J; Ochiana, So; Bland, Nd; Gustafson, A; Campbell, Rk; Pollastri, Mp | file da validare |
Preparation and Evaluation of a Series of Indoles as Sigma Receptor Ligands | 1-gen-2012 | Alsharif, W; Mesangeau, C; Matsumoto, Rr; Seminerio, Mj; M., Robson M; Poupaert, Jh; Amata, Emanuele; Mccurdy, Cr | file da validare |
Neglected disease lead discovery: Profiling analogs of Lapatinib against the protozoan parasites that cause Chagas disease, leishmaniasis, and malaria | 1-gen-2012 | Amata, Emanuele; Devine, W; Mehta, N; Swaminathan, U; Rodriguez, A; Erath, J.; Andriani, G; Sciotti, R; Pollastri, Mp | file da validare |
Targeting Neglected Parasitic Diseases with Human EGFR Inhibitor Chemotypes | 1-gen-2013 | Woodring, J. L.; Patel, G.; Amata, Emanuele; Sciotti, R.; Rodriguez, A.; Pollastri, M. P. | file da validare |
Antitrypanosomal lead discovery: Identification of a ligand-efficient inhibitor of Trypanosoma cruzi CYP51 and parasite growth | 1-gen-2013 | Andriani, Grasiella; Amata, Emanuele; Beatty, Joel; Clements, Zeke; Coffey J., Brian; Courtemanche, Gilles; Devine, William; Erath, Jessey; Juda E., Cristin; Wawrzak, Zdzislaw; Wood T., Jodianne; Lepesheva L., Galina; Rodriguez, Ana; Pollastri P., Michael | |
Involvement of sigma 2 receptor on motor disorder | 1-gen-2014 | Aricò, G; Ronsisvalle, N; Cova, Am; Blanco, P; Amata, Emanuele; Parenti, Carmela; Ronsisvalle, Simone | file da validare |
Repurposing human PDE4 inhibitors for neglected tropical diseases: design, synthesis and evaluation of cilomilast analogues as Trypanosoma brucei PDEB1 inhibitors | 1-gen-2014 | Amata, Emanuele; Bland D., Nicholas; Hoyt T., Charles; Settimo, Luca; Campbell K., Robert; Pollastri P., Michael | file da validare |
Identification and characterization of hundreds of potent and selective inhibitors of Trypanosoma brucei growth from a kinase-targeted library screening campaign | 1-gen-2014 | Diaz, Rosario; Luengo-Arratta A., Sandra; Seixas D., João; Amata, Emanuele; Devine, William; Cordon-Obras, Carlos; Rojas-Barros L., Domingo; Jimenez, Elena; Ortega, Fatima; Crouch, Sabrinia; Colmenarejo, Gonzalo; Fiandor Jose, Maria; Martin Jose, Julio; Berlanga, Manuela; Gonzalez, Silvia; Manzano, Pilar; Navarro, Miguel; Pollastri P., Michael | |
Antioxidant activity of (+)-Pentazocine on activated microglia | 1-gen-2015 | Marrazzo, Agostino; Heiss, Kathrin; Prezzavento, Orazio; Arena, Emanuela; Amata, Emanuele; LI VOLTI, Giovanni | file da validare |
New 5-Ht7 Receptor Ligands As Potential Antidepressant Agents. | 1-gen-2015 | Romeo, Giuseppe; Modica, Maria Nunziata; Salerno, Loredana; Pittala', Valeria; Siracusa, Maria Angela; Intagliata, Sebastiano; Marrazzo, Agostino; Prezzavento, Orazio; Amata, Emanuele; Cagnotto, Alfredo; Salmona, Mario | file da validare |
Antioxidant properties and pharmacokinetic studies of new selective σ1 bifunctional ligands | 1-gen-2015 | Marrazzo, Agostino; Arena, Emanuela; Cacciatore, Ivana; Cerasa Laura, S.; Amata, Emanuele; Pittala', Valeria; Pasquinucci, Lorella Giuseppina; Turkez, Hasan; Di Stefano, Antonio; Prezzavento, Orazio | file da validare |
C-5'-Triazolyl-2'-oxa-3'-aza-4'a-carbanucleosides: Synthesis and biological evaluation | 1-gen-2015 | Romeo, Roberto; Carnovale, Caterina; Giofrè V., Salvatore; Chiacchio, MARIA ASSUNTA ROSSELLA; Garozzo, Adriana; Amata, Emanuele; Romeo, Giovanni; Chiacchio, Ugo |
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