Sfoglia per Autore
C-5'-Triazolyl-2'-oxa-3'-aza-4'a-carbanucleosides: Synthesis and biological evaluation
2015-01-01 Romeo, Roberto; Carnovale, Caterina; Giofrè V., Salvatore; Chiacchio, MARIA ASSUNTA ROSSELLA; Garozzo, Adriana; Amata, Emanuele; Romeo, Giovanni; Chiacchio, Ugo
Evaluation of pyrrolidine and pyrazolone derivatives as inhibitors of trypanosomal phosphodiesterase B1 (TbrPDEB1)
2015-01-01 Amata, Emanuele; Bland D., Nicholas; Campbell K., Robert; Pollastri P., Michael
Protozoan Parasite Growth Inhibitors Discovered by Cross-Screening Yield Potent Scaffolds for Lead Discovery
2015-01-01 Devine, William; Woodring L., Jennifer; Swaminathan, Uma; Amata, Emanuele; Gautam, Patel; Erath, Jessey; Roncal E., Norma; Lee J., Patricia; Leed E., Susan; Rodriguez, Ana; Mensa-Wilmot, Kojo; Sciotti J., Richard; Pollastri P., Michael
Identification of “Preferred” Human Kinase Inhibitors for Human African Trypanosomiasis Through a Statistical Analysis-Driven Approach
file da validare2016-01-01 Amata, Emanuele; Pollastri Michael, P.
Heme Oxygenase-1 Inhibition: A Novel Strategy for the Design of Azole-Based Antitumour Agents
file da validare2016-01-01 Pittalà, Valeria; Romeo, Giuseppe; Marrazzo, Agostino; Amata, Emanuele; DI GIACOMO, Claudia; Sorrenti, Valeria; Salerno, Loredana
Haloperidol Metabolite II Valproate Ester: Antiangiogenic Activity in Human Microvascular Retinal Endothelial Cells
file da validare2016-01-01 Marrazzo, Agostino; Amata, Emanuele; Olivieri, Melania; Prezzavento, Orazio; Arena, Emanuela; Romeo, Giuseppe; Pittalà, Valeria; Salerno, Loredana; Anfuso, CARMELINA DANIELA
Identification of Novel Lead Compounds for Sleeping Sickness via Preferred Lead Repurposing
file da validare2016-01-01 Amata, Emanuele; Pollastri Michael, P.
Novel selective ligands for the serotonergic 5-HT7 receptor: tricyclic derivatives Bearing the pyrimido-4(3H)-one ring
file da validare2016-01-01 Romeo, Giuseppe; Pittala', Valeria; Salerno, Loredana; MODICA Maria, N; Candido, Margherita; Intagliata, Sebastiano; Marrazzo, Agostino; Amata, Emanuele; Cagnotto, A; Salmona, M; Siracusa, Maria Angela
Caspase-3 activation in human melanoma A375 cell line by a novel selective sigma-2 agonist
2016-01-01 Ronsisvalle, Simone; Aricò, Giuseppina; Cova, ANNA MARIA; Blanco, Palma; Amata, Emanuele; Pappalardo, Maria Sebastiana; Pasquinucci, Lorella; Spadaro, Angelo; Ronsisvalle, Nicole
Antiangiogenic Effect of (±)-Haloperidol Metabolite II Valproate Ester [(±)-MRJF22] in Human Microvascular Retinal Endothelial Cells
2016-01-01 Olivieri, Melania; Amata, Emanuele; Vinciguerra, Shila; Fiorito, Jole; Giurdanella, Giovanni; Drago, Filippo; Caporarello, Nunzia; Prezzavento, Orazio; Arena, Emanuela; Salerno, Loredana; Rescifina, Antonio; Lupo, Gabriella; Anfuso, CARMELINA DANIELA; Marrazzo, Agostino
Identification of “Preferred” Human Kinase Inhibitors for Sleeping Sickness Lead Discovery. Are Some Kinases Better than Others for Inhibitor Repurposing?
2016-01-01 Amata, Emanuele; Xi, Hualin; Colmenarejo, Gonzalo; Gonzalez-Diaz, Rosario; Cordon-Obras, Carlos; Berlanga, Manuela; Manzano, Pilar; Erath, Jessey; Roncal E., Norma; Lee J., Patricia; Leed E., Susan; Rodriguez, Ana; Sciotti J., Richard; Navarro, Miguel; Pollastri, P. Michael.
Composti inorganici [Cap. 6]
2017-01-01 Amata, Emanuele; Dichiara, Maria
Targeting Heme Oxygenase-1 to Overcome Imatinib Resistance in Chronic Myeloid Leukemia
file da validare2017-01-01 Salerno, Loredana; Pittalà, Valeria; Modica Maria, N.; Amata, Emanuele; Prezzavento, Orazio; Marrazzo, Agostino; Sorrenti, Valeria; Vanella, Luca; Greish, K.; Romeo, Giuseppe
Development of Sigma Receptors Nitric Oxide Photodonor Ligands with Antiproliferative Activity
file da validare2017-01-01 Amata, Emanuele; Marrazzo, Agostino; Dichiara, Maria; Arena, Emanuela; Russo, Marina; Fraix, Aurore; Modica Maria, N.; Pittalà, Valeria; Sortino, Salvatore; Prezzavento, Orazio
Tumor Targeting Sigma Receptor Ligands: Development of New Molecular Hybrids as Anticancer Therapeutics
file da validare2017-01-01 Dichiara, Maria; Amata, Emanuele; Prezzavento, Orazio; Arena, Emanuela; Sortino, Salvatore; Fraix, Aurore; Marrazzo, Agostino; Arico', Giuseppina
Synthesis of Novel Benzylpiperazine Derivatives as Ligands for the σ1 Receptor
file da validare2017-01-01 Romeo, Giuseppe; Salerno, Loredana; Bonanno, Federica; Pittalà, Valeria; Modica, Marian; Siracusa, Maria Angela; Marrazzo, Agostino; Amata, Emanuele; Arena, Emanuela; Prezzavento, Orazio
(+)-and (−)-Phenazocine enantiomers: evaluation of their dual opioid agonist/σ1 antagonist properties and antinociceptive effects
2017-01-01 Prezzavento, Orazio; Arena, Emanuela; Sánchez-Fernández, Cristine; Turnaturi, Rita; Parenti, Carmela; Marrazzo, Agostino; Catalano, Roberto; Amata, Emanuele; Pasquinucci, Lorella; Cobos J., Enrique
Heme Oxygenase-1: A new druggable target in the management of chronic and acute myeloid leukemia
2017-01-01 Salerno, Loredana; Romeo, Giuseppe; Modica, Maria Nunziata; Amata, Emanuele; Sorrenti, Valeria; Barbagallo, Ignazio; Pittalà, Valeria
Hyphenated 3D-QSAR statistical model-scaffold hopping analysis for the identification of potentially potent and selective sigma-2 receptor ligands
2017-01-01 Floresta, Giuseppe; Rescifina, Antonio; Marrazzo, Agostino; Dichiara, Maria; Pistarà, Venerando; Pittalà, Valeria; Prezzavento, Orazio; Amata, Emanuele
Adipocyte fatty acid binding protein 4 (FABP4) inhibitors. A comprehensive systematic review
2017-01-01 Floresta, Giuseppe; Pistarà, Venerando; Amata, Emanuele; Dichiara, Maria; Marrazzo, Agostino; Prezzavento, Orazio; Rescifina, Antonio
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
C-5'-Triazolyl-2'-oxa-3'-aza-4'a-carbanucleosides: Synthesis and biological evaluation | 1-gen-2015 | Romeo, Roberto; Carnovale, Caterina; Giofrè V., Salvatore; Chiacchio, MARIA ASSUNTA ROSSELLA; Garozzo, Adriana; Amata, Emanuele; Romeo, Giovanni; Chiacchio, Ugo | |
Evaluation of pyrrolidine and pyrazolone derivatives as inhibitors of trypanosomal phosphodiesterase B1 (TbrPDEB1) | 1-gen-2015 | Amata, Emanuele; Bland D., Nicholas; Campbell K., Robert; Pollastri P., Michael | |
Protozoan Parasite Growth Inhibitors Discovered by Cross-Screening Yield Potent Scaffolds for Lead Discovery | 1-gen-2015 | Devine, William; Woodring L., Jennifer; Swaminathan, Uma; Amata, Emanuele; Gautam, Patel; Erath, Jessey; Roncal E., Norma; Lee J., Patricia; Leed E., Susan; Rodriguez, Ana; Mensa-Wilmot, Kojo; Sciotti J., Richard; Pollastri P., Michael | |
Identification of “Preferred” Human Kinase Inhibitors for Human African Trypanosomiasis Through a Statistical Analysis-Driven Approach | 1-gen-2016 | Amata, Emanuele; Pollastri Michael, P. | file da validare |
Heme Oxygenase-1 Inhibition: A Novel Strategy for the Design of Azole-Based Antitumour Agents | 1-gen-2016 | Pittalà, Valeria; Romeo, Giuseppe; Marrazzo, Agostino; Amata, Emanuele; DI GIACOMO, Claudia; Sorrenti, Valeria; Salerno, Loredana | file da validare |
Haloperidol Metabolite II Valproate Ester: Antiangiogenic Activity in Human Microvascular Retinal Endothelial Cells | 1-gen-2016 | Marrazzo, Agostino; Amata, Emanuele; Olivieri, Melania; Prezzavento, Orazio; Arena, Emanuela; Romeo, Giuseppe; Pittalà, Valeria; Salerno, Loredana; Anfuso, CARMELINA DANIELA | file da validare |
Identification of Novel Lead Compounds for Sleeping Sickness via Preferred Lead Repurposing | 1-gen-2016 | Amata, Emanuele; Pollastri Michael, P. | file da validare |
Novel selective ligands for the serotonergic 5-HT7 receptor: tricyclic derivatives Bearing the pyrimido-4(3H)-one ring | 1-gen-2016 | Romeo, Giuseppe; Pittala', Valeria; Salerno, Loredana; MODICA Maria, N; Candido, Margherita; Intagliata, Sebastiano; Marrazzo, Agostino; Amata, Emanuele; Cagnotto, A; Salmona, M; Siracusa, Maria Angela | file da validare |
Caspase-3 activation in human melanoma A375 cell line by a novel selective sigma-2 agonist | 1-gen-2016 | Ronsisvalle, Simone; Aricò, Giuseppina; Cova, ANNA MARIA; Blanco, Palma; Amata, Emanuele; Pappalardo, Maria Sebastiana; Pasquinucci, Lorella; Spadaro, Angelo; Ronsisvalle, Nicole | |
Antiangiogenic Effect of (±)-Haloperidol Metabolite II Valproate Ester [(±)-MRJF22] in Human Microvascular Retinal Endothelial Cells | 1-gen-2016 | Olivieri, Melania; Amata, Emanuele; Vinciguerra, Shila; Fiorito, Jole; Giurdanella, Giovanni; Drago, Filippo; Caporarello, Nunzia; Prezzavento, Orazio; Arena, Emanuela; Salerno, Loredana; Rescifina, Antonio; Lupo, Gabriella; Anfuso, CARMELINA DANIELA; Marrazzo, Agostino | |
Identification of “Preferred” Human Kinase Inhibitors for Sleeping Sickness Lead Discovery. Are Some Kinases Better than Others for Inhibitor Repurposing? | 1-gen-2016 | Amata, Emanuele; Xi, Hualin; Colmenarejo, Gonzalo; Gonzalez-Diaz, Rosario; Cordon-Obras, Carlos; Berlanga, Manuela; Manzano, Pilar; Erath, Jessey; Roncal E., Norma; Lee J., Patricia; Leed E., Susan; Rodriguez, Ana; Sciotti J., Richard; Navarro, Miguel; Pollastri, P. Michael. | |
Composti inorganici [Cap. 6] | 1-gen-2017 | Amata, Emanuele; Dichiara, Maria | |
Targeting Heme Oxygenase-1 to Overcome Imatinib Resistance in Chronic Myeloid Leukemia | 1-gen-2017 | Salerno, Loredana; Pittalà, Valeria; Modica Maria, N.; Amata, Emanuele; Prezzavento, Orazio; Marrazzo, Agostino; Sorrenti, Valeria; Vanella, Luca; Greish, K.; Romeo, Giuseppe | file da validare |
Development of Sigma Receptors Nitric Oxide Photodonor Ligands with Antiproliferative Activity | 1-gen-2017 | Amata, Emanuele; Marrazzo, Agostino; Dichiara, Maria; Arena, Emanuela; Russo, Marina; Fraix, Aurore; Modica Maria, N.; Pittalà, Valeria; Sortino, Salvatore; Prezzavento, Orazio | file da validare |
Tumor Targeting Sigma Receptor Ligands: Development of New Molecular Hybrids as Anticancer Therapeutics | 1-gen-2017 | Dichiara, Maria; Amata, Emanuele; Prezzavento, Orazio; Arena, Emanuela; Sortino, Salvatore; Fraix, Aurore; Marrazzo, Agostino; Arico', Giuseppina | file da validare |
Synthesis of Novel Benzylpiperazine Derivatives as Ligands for the σ1 Receptor | 1-gen-2017 | Romeo, Giuseppe; Salerno, Loredana; Bonanno, Federica; Pittalà, Valeria; Modica, Marian; Siracusa, Maria Angela; Marrazzo, Agostino; Amata, Emanuele; Arena, Emanuela; Prezzavento, Orazio | file da validare |
(+)-and (−)-Phenazocine enantiomers: evaluation of their dual opioid agonist/σ1 antagonist properties and antinociceptive effects | 1-gen-2017 | Prezzavento, Orazio; Arena, Emanuela; Sánchez-Fernández, Cristine; Turnaturi, Rita; Parenti, Carmela; Marrazzo, Agostino; Catalano, Roberto; Amata, Emanuele; Pasquinucci, Lorella; Cobos J., Enrique | |
Heme Oxygenase-1: A new druggable target in the management of chronic and acute myeloid leukemia | 1-gen-2017 | Salerno, Loredana; Romeo, Giuseppe; Modica, Maria Nunziata; Amata, Emanuele; Sorrenti, Valeria; Barbagallo, Ignazio; Pittalà, Valeria | |
Hyphenated 3D-QSAR statistical model-scaffold hopping analysis for the identification of potentially potent and selective sigma-2 receptor ligands | 1-gen-2017 | Floresta, Giuseppe; Rescifina, Antonio; Marrazzo, Agostino; Dichiara, Maria; Pistarà, Venerando; Pittalà, Valeria; Prezzavento, Orazio; Amata, Emanuele | |
Adipocyte fatty acid binding protein 4 (FABP4) inhibitors. A comprehensive systematic review | 1-gen-2017 | Floresta, Giuseppe; Pistarà, Venerando; Amata, Emanuele; Dichiara, Maria; Marrazzo, Agostino; Prezzavento, Orazio; Rescifina, Antonio |
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