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Titolo Data di pubblicazione Autore(i) File
C-5'-Triazolyl-2'-oxa-3'-aza-4'a-carbanucleosides: Synthesis and biological evaluation 1-gen-2015 Romeo, Roberto; Carnovale, Caterina; Giofrè V., Salvatore; Chiacchio, MARIA ASSUNTA ROSSELLA; Garozzo, Adriana; Amata, Emanuele; Romeo, Giovanni; Chiacchio, Ugo
Evaluation of pyrrolidine and pyrazolone derivatives as inhibitors of trypanosomal phosphodiesterase B1 (TbrPDEB1) 1-gen-2015 Amata, Emanuele; Bland D., Nicholas; Campbell K., Robert; Pollastri P., Michael
Protozoan Parasite Growth Inhibitors Discovered by Cross-Screening Yield Potent Scaffolds for Lead Discovery 1-gen-2015 Devine, William; Woodring L., Jennifer; Swaminathan, Uma; Amata, Emanuele; Gautam, Patel; Erath, Jessey; Roncal E., Norma; Lee J., Patricia; Leed E., Susan; Rodriguez, Ana; Mensa-Wilmot, Kojo; Sciotti J., Richard; Pollastri P., Michael
Identification of “Preferred” Human Kinase Inhibitors for Human African Trypanosomiasis Through a Statistical Analysis-Driven Approach 1-gen-2016 Amata, Emanuele; Pollastri Michael, P. file da validare
Heme Oxygenase-1 Inhibition: A Novel Strategy for the Design of Azole-Based Antitumour Agents 1-gen-2016 Pittalà, Valeria; Romeo, Giuseppe; Marrazzo, Agostino; Amata, Emanuele; DI GIACOMO, Claudia; Sorrenti, Valeria; Salerno, Loredana file da validare
Haloperidol Metabolite II Valproate Ester: Antiangiogenic Activity in Human Microvascular Retinal Endothelial Cells 1-gen-2016 Marrazzo, Agostino; Amata, Emanuele; Olivieri, Melania; Prezzavento, Orazio; Arena, Emanuela; Romeo, Giuseppe; Pittalà, Valeria; Salerno, Loredana; Anfuso, CARMELINA DANIELA file da validare
Identification of Novel Lead Compounds for Sleeping Sickness via Preferred Lead Repurposing 1-gen-2016 Amata, Emanuele; Pollastri Michael, P. file da validare
Novel selective ligands for the serotonergic 5-HT7 receptor: tricyclic derivatives Bearing the pyrimido-4(3H)-one ring 1-gen-2016 Romeo, Giuseppe; Pittala', Valeria; Salerno, Loredana; MODICA Maria, N; Candido, Margherita; Intagliata, Sebastiano; Marrazzo, Agostino; Amata, Emanuele; Cagnotto, A; Salmona, M; Siracusa, Maria Angela file da validare
Caspase-3 activation in human melanoma A375 cell line by a novel selective sigma-2 agonist 1-gen-2016 Ronsisvalle, Simone; Aricò, Giuseppina; Cova, ANNA MARIA; Blanco, Palma; Amata, Emanuele; Pappalardo, Maria Sebastiana; Pasquinucci, Lorella; Spadaro, Angelo; Ronsisvalle, Nicole
Antiangiogenic Effect of (±)-Haloperidol Metabolite II Valproate Ester [(±)-MRJF22] in Human Microvascular Retinal Endothelial Cells 1-gen-2016 Olivieri, Melania; Amata, Emanuele; Vinciguerra, Shila; Fiorito, Jole; Giurdanella, Giovanni; Drago, Filippo; Caporarello, Nunzia; Prezzavento, Orazio; Arena, Emanuela; Salerno, Loredana; Rescifina, Antonio; Lupo, Gabriella; Anfuso, CARMELINA DANIELA; Marrazzo, Agostino
Identification of “Preferred” Human Kinase Inhibitors for Sleeping Sickness Lead Discovery. Are Some Kinases Better than Others for Inhibitor Repurposing? 1-gen-2016 Amata, Emanuele; Xi, Hualin; Colmenarejo, Gonzalo; Gonzalez-Diaz, Rosario; Cordon-Obras, Carlos; Berlanga, Manuela; Manzano, Pilar; Erath, Jessey; Roncal E., Norma; Lee J., Patricia; Leed E., Susan; Rodriguez, Ana; Sciotti J., Richard; Navarro, Miguel; Pollastri, P. Michael.
Composti inorganici [Cap. 6] 1-gen-2017 Amata, Emanuele; Dichiara, Maria
Targeting Heme Oxygenase-1 to Overcome Imatinib Resistance in Chronic Myeloid Leukemia 1-gen-2017 Salerno, Loredana; Pittalà, Valeria; Modica Maria, N.; Amata, Emanuele; Prezzavento, Orazio; Marrazzo, Agostino; Sorrenti, Valeria; Vanella, Luca; Greish, K.; Romeo, Giuseppe file da validare
Development of Sigma Receptors Nitric Oxide Photodonor Ligands with Antiproliferative Activity 1-gen-2017 Amata, Emanuele; Marrazzo, Agostino; Dichiara, Maria; Arena, Emanuela; Russo, Marina; Fraix, Aurore; Modica Maria, N.; Pittalà, Valeria; Sortino, Salvatore; Prezzavento, Orazio file da validare
Tumor Targeting Sigma Receptor Ligands: Development of New Molecular Hybrids as Anticancer Therapeutics 1-gen-2017 Dichiara, Maria; Amata, Emanuele; Prezzavento, Orazio; Arena, Emanuela; Sortino, Salvatore; Fraix, Aurore; Marrazzo, Agostino; Arico', Giuseppina file da validare
Synthesis of Novel Benzylpiperazine Derivatives as Ligands for the σ1 Receptor 1-gen-2017 Romeo, Giuseppe; Salerno, Loredana; Bonanno, Federica; Pittalà, Valeria; Modica, Marian; Siracusa, Maria Angela; Marrazzo, Agostino; Amata, Emanuele; Arena, Emanuela; Prezzavento, Orazio file da validare
(+)-and (−)-Phenazocine enantiomers: evaluation of their dual opioid agonist/σ1 antagonist properties and antinociceptive effects 1-gen-2017 Prezzavento, Orazio; Arena, Emanuela; Sánchez-Fernández, Cristine; Turnaturi, Rita; Parenti, Carmela; Marrazzo, Agostino; Catalano, Roberto; Amata, Emanuele; Pasquinucci, Lorella; Cobos J., Enrique
Heme Oxygenase-1: A new druggable target in the management of chronic and acute myeloid leukemia 1-gen-2017 Salerno, Loredana; Romeo, Giuseppe; Modica, Maria Nunziata; Amata, Emanuele; Sorrenti, Valeria; Barbagallo, Ignazio; Pittalà, Valeria
Hyphenated 3D-QSAR statistical model-scaffold hopping analysis for the identification of potentially potent and selective sigma-2 receptor ligands 1-gen-2017 Floresta, Giuseppe; Rescifina, Antonio; Marrazzo, Agostino; Dichiara, Maria; Pistarà, Venerando; Pittalà, Valeria; Prezzavento, Orazio; Amata, Emanuele
Adipocyte fatty acid binding protein 4 (FABP4) inhibitors. A comprehensive systematic review 1-gen-2017 Floresta, Giuseppe; Pistarà, Venerando; Amata, Emanuele; Dichiara, Maria; Marrazzo, Agostino; Prezzavento, Orazio; Rescifina, Antonio
Mostrati risultati da 21 a 40 di 117
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