Sfoglia per Autore
A new heterocyclic ring system: synthesis of pyrazolo[3',4':4,5]pyrimido-[2,1-a]phthalazine derivatives
file da validare1992-01-01 Santagati, M; Santagati, A; Modica, Maria Nunziata; Russo, F.
Synthesis of piperazinyl-alkylthiothieno[2,3-d]pyrimidine derivatives and serotonergic activity avaluation
file da validare1992-01-01 Modica, Maria Nunziata; Santagati, M; Santagati, A; Russo, F.
Synthesis of 2,3,5,6,7,8-hexahydro-3-amino-thioxo[1]benzothieno[2,3-d]-pyrimidin-4(1H)-one and derivatives of the new heterocyclic system 7,8,9,10-tetrahydro-3H,11H-[1]benzothieno[2',3':4,5]pyrimido[2,1-b][1,3,4]-thiadiazin-11-one
file da validare1993-01-01 Santagati, A; Santagati, M; Modica, Maria Nunziata
Synthesis and pharmacological properties of benzothiazole, 1,3,4-oxadiazole and 1,3,4-thiadiazole derivatives
file da validare1994-01-01 Santagati, M; Modica, Maria Nunziata; Santagati, A; Russo, F; Caruso, A; Cutuli, V; DI PIETRO, E; AMICO ROXAS, M.
Synthesis of 2,3-dihydro-3-amino-6-phenyl-2-thioxothieno[2,3-d]pyrimidin-4(1H)-one and of potential antiinflammatory agents 2-aryl-7-phenyl-3H,9H-pyrimido[2,1-b]thieno[2',3':4,5][1,3,4]thiadiazin-9-ones
file da validare1994-01-01 Santagati, A; Modica, Maria Nunziata; Santagati, M; Caruso, A; Cutuli, V.
Study on the tachykinins antagonist effect of combinatorial functionalized heterocycle replacements in tryciclic pyrimidine derivatives
file da validare1994-01-01 Guccione, Salvatore; Modica, Maria Nunziata; Shaw, D; UCCELLO BARRETTA, G; Santagati, A; Santagati, M.
Bridgehead nitrogen heterocycles derived from the potassium salt of 2,3,5,6,7,8-hexahydro-3-amino-2-thioxo-[1]benzothieno[2,3-d]pyrimidin-4(1H)-one
file da validare1994-01-01 Santagati, A; Modica, Maria Nunziata; Santagati, M.
Synthesis and pharmacological properties of thieno[2',3':4,5]pyrimido[2,1-b][1,3,4]thiadiazine derivatives
file da validare1995-01-01 Santagati, A; Modica, Maria Nunziata; Santagati, M; Cutuli, V; Amore, D; Caruso, A.
CoMFA contributions to a binding mode for NK2 receptor antagonists
file da validare1995-01-01 Guccione, Salvatore; Santagati, M; Santagati, A; Modica, Maria Nunziata; UCCELLO BARRETTA, G; Langer, T; Russo, F.
Potential of indole skeleton containing heterocycles as antagonists at the neurokinin (NK) receptor system
file da validare1995-01-01 Modica, Maria Nunziata; Santagati, A; Santagati, M; MONSU’ SCOLARO, L; Guccione, Salvatore; Russo, F.
Synthesis and NK-2 antagonist effect of 1,6-diphenyl-pyrazolo [3, 4-d]-thiazolo[3,2-a]4H-pyrimidin-4-one
file da validare1996-01-01 Guccione, Salvatore; Modica, Maria Nunziata; J., Longmore; D., Shaw; G., UCCELLO BARRETTA; A., Santagati; M., Santagati; F., Russo
Synthesis of aminothienopyrimidine and thienotriazolopyrimidine derivatives as potential anticonvulsant agents
file da validare1996-01-01 Santagati, M; Modica, Maria Nunziata; Santagati, A; Russo, F; Spampinato, S.
[[(Arylpiperazinyl)alkylthio]thieno[2,3-d]pyrimidinone derivatives as high-affinity, selective 5-HT1A receptor ligands
file da validare1997-01-01 Modica, Maria Nunziata; Santagati, M; Russo, F; Parotti, L; DE GIOIA, L; Selvaggini, C; Salmona, M; Mennini, T.
Synthesis of 1-phenyl-6-arilsubstituted pyrazolopyrimidothiazole as antagonists at the NK-2 receptors
file da validare1997-01-01 Russo, F; Longmore, J; Modica, Maria Nunziata; Santagati, M; Santagati, A; Guccione, Salvatore
Building a model of interaction at the NK-2 receptors: polycondensed heterocycles containing the pyrimidoindole skeleton
file da validare1998-01-01 Santagati, A; Longmore, J; Guccione, Salvatore; Langer, T; Tonnel, E; Modica, Maria Nunziata; Santagati, M; MONSU’ SCOLARO, L; Russo, F.
5-HT1A receptors mapping by conformational analysis (2D NOESY/MM) and ”three way modelling” (HASL, CoMFA, PARM)
file da validare1998-01-01 Santagati, M; Doweyko, A; Santagati, A; Modica, Maria Nunziata; Guccione, Salvatore; Chen, H. M.; Uccello Barretta, G; Balzano, F.
5-HT1A receptors mapping by conformational analysis (2D NOESY/MM) and "tree way modelling" (HASL, CoMFA, PARM)
file da validare1998-01-01 Santagati, M; Doweyko, A; Santagati, A; Modica, Maria Nunziata; Guccione, Salvatore; Chen, H; Russo, F; UCCELLO BARRETTA, G; Balzano, F.
Application of PARM to constructing and comparing 5-HT1A and alfa1 receptor models
file da validare1998-01-01 Santagati, M; Chen, H; Santagati, A; Modica, Maria Nunziata; Guccione, Salvatore; Uccello Barretta, G; Balzano, F.
Application of Parm to constructing and comparing 5-HT1A and alfa1 receptor models
file da validare1998-01-01 Santagati, M; Chen, H; Santagati, A; Modica, Maria Nunziata; Guccione, Salvatore; Russo, F; UCCELLO BARRETTA, G; Balzano, F.
Receptor modeling using " Multiconformer" alignment: comparison of HASL and CoMFA in the analysis of 5-HT1A thienopyrimidinone ligands
file da validare1999-01-01 Guccione, Salvatore; Doweyko, A. M.; Chen, H; Modica, Maria Nunziata; Santagati, M; Santagati, A; UCCELLO BARRETTA, G; Balzano, F.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
A new heterocyclic ring system: synthesis of pyrazolo[3',4':4,5]pyrimido-[2,1-a]phthalazine derivatives | 1-gen-1992 | Santagati, M; Santagati, A; Modica, Maria Nunziata; Russo, F. | file da validare |
Synthesis of piperazinyl-alkylthiothieno[2,3-d]pyrimidine derivatives and serotonergic activity avaluation | 1-gen-1992 | Modica, Maria Nunziata; Santagati, M; Santagati, A; Russo, F. | file da validare |
Synthesis of 2,3,5,6,7,8-hexahydro-3-amino-thioxo[1]benzothieno[2,3-d]-pyrimidin-4(1H)-one and derivatives of the new heterocyclic system 7,8,9,10-tetrahydro-3H,11H-[1]benzothieno[2',3':4,5]pyrimido[2,1-b][1,3,4]-thiadiazin-11-one | 1-gen-1993 | Santagati, A; Santagati, M; Modica, Maria Nunziata | file da validare |
Synthesis and pharmacological properties of benzothiazole, 1,3,4-oxadiazole and 1,3,4-thiadiazole derivatives | 1-gen-1994 | Santagati, M; Modica, Maria Nunziata; Santagati, A; Russo, F; Caruso, A; Cutuli, V; DI PIETRO, E; AMICO ROXAS, M. | file da validare |
Synthesis of 2,3-dihydro-3-amino-6-phenyl-2-thioxothieno[2,3-d]pyrimidin-4(1H)-one and of potential antiinflammatory agents 2-aryl-7-phenyl-3H,9H-pyrimido[2,1-b]thieno[2',3':4,5][1,3,4]thiadiazin-9-ones | 1-gen-1994 | Santagati, A; Modica, Maria Nunziata; Santagati, M; Caruso, A; Cutuli, V. | file da validare |
Study on the tachykinins antagonist effect of combinatorial functionalized heterocycle replacements in tryciclic pyrimidine derivatives | 1-gen-1994 | Guccione, Salvatore; Modica, Maria Nunziata; Shaw, D; UCCELLO BARRETTA, G; Santagati, A; Santagati, M. | file da validare |
Bridgehead nitrogen heterocycles derived from the potassium salt of 2,3,5,6,7,8-hexahydro-3-amino-2-thioxo-[1]benzothieno[2,3-d]pyrimidin-4(1H)-one | 1-gen-1994 | Santagati, A; Modica, Maria Nunziata; Santagati, M. | file da validare |
Synthesis and pharmacological properties of thieno[2',3':4,5]pyrimido[2,1-b][1,3,4]thiadiazine derivatives | 1-gen-1995 | Santagati, A; Modica, Maria Nunziata; Santagati, M; Cutuli, V; Amore, D; Caruso, A. | file da validare |
CoMFA contributions to a binding mode for NK2 receptor antagonists | 1-gen-1995 | Guccione, Salvatore; Santagati, M; Santagati, A; Modica, Maria Nunziata; UCCELLO BARRETTA, G; Langer, T; Russo, F. | file da validare |
Potential of indole skeleton containing heterocycles as antagonists at the neurokinin (NK) receptor system | 1-gen-1995 | Modica, Maria Nunziata; Santagati, A; Santagati, M; MONSU’ SCOLARO, L; Guccione, Salvatore; Russo, F. | file da validare |
Synthesis and NK-2 antagonist effect of 1,6-diphenyl-pyrazolo [3, 4-d]-thiazolo[3,2-a]4H-pyrimidin-4-one | 1-gen-1996 | Guccione, Salvatore; Modica, Maria Nunziata; J., Longmore; D., Shaw; G., UCCELLO BARRETTA; A., Santagati; M., Santagati; F., Russo | file da validare |
Synthesis of aminothienopyrimidine and thienotriazolopyrimidine derivatives as potential anticonvulsant agents | 1-gen-1996 | Santagati, M; Modica, Maria Nunziata; Santagati, A; Russo, F; Spampinato, S. | file da validare |
[[(Arylpiperazinyl)alkylthio]thieno[2,3-d]pyrimidinone derivatives as high-affinity, selective 5-HT1A receptor ligands | 1-gen-1997 | Modica, Maria Nunziata; Santagati, M; Russo, F; Parotti, L; DE GIOIA, L; Selvaggini, C; Salmona, M; Mennini, T. | file da validare |
Synthesis of 1-phenyl-6-arilsubstituted pyrazolopyrimidothiazole as antagonists at the NK-2 receptors | 1-gen-1997 | Russo, F; Longmore, J; Modica, Maria Nunziata; Santagati, M; Santagati, A; Guccione, Salvatore | file da validare |
Building a model of interaction at the NK-2 receptors: polycondensed heterocycles containing the pyrimidoindole skeleton | 1-gen-1998 | Santagati, A; Longmore, J; Guccione, Salvatore; Langer, T; Tonnel, E; Modica, Maria Nunziata; Santagati, M; MONSU’ SCOLARO, L; Russo, F. | file da validare |
5-HT1A receptors mapping by conformational analysis (2D NOESY/MM) and ”three way modelling” (HASL, CoMFA, PARM) | 1-gen-1998 | Santagati, M; Doweyko, A; Santagati, A; Modica, Maria Nunziata; Guccione, Salvatore; Chen, H. M.; Uccello Barretta, G; Balzano, F. | file da validare |
5-HT1A receptors mapping by conformational analysis (2D NOESY/MM) and "tree way modelling" (HASL, CoMFA, PARM) | 1-gen-1998 | Santagati, M; Doweyko, A; Santagati, A; Modica, Maria Nunziata; Guccione, Salvatore; Chen, H; Russo, F; UCCELLO BARRETTA, G; Balzano, F. | file da validare |
Application of PARM to constructing and comparing 5-HT1A and alfa1 receptor models | 1-gen-1998 | Santagati, M; Chen, H; Santagati, A; Modica, Maria Nunziata; Guccione, Salvatore; Uccello Barretta, G; Balzano, F. | file da validare |
Application of Parm to constructing and comparing 5-HT1A and alfa1 receptor models | 1-gen-1998 | Santagati, M; Chen, H; Santagati, A; Modica, Maria Nunziata; Guccione, Salvatore; Russo, F; UCCELLO BARRETTA, G; Balzano, F. | file da validare |
Receptor modeling using " Multiconformer" alignment: comparison of HASL and CoMFA in the analysis of 5-HT1A thienopyrimidinone ligands | 1-gen-1999 | Guccione, Salvatore; Doweyko, A. M.; Chen, H; Modica, Maria Nunziata; Santagati, M; Santagati, A; UCCELLO BARRETTA, G; Balzano, F. | file da validare |
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