Sfoglia per Autore
CCB - A novel analog of MPCB with high binding affinity and specific kappa opioid receptor agonist
file da validare1994-01-01 Ronsisvalle, Giuseppe; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Carboni, L; Pistacchio, E; Spampinato, S.
New developments in opioid receptors ligands
file da validare1995-01-01 Ronsisvalle, G; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Marrazzo, Agostino; Vittorio, F; Pappalardo, Ms; Bousquet, E.
Selective Ligands for Sigma1 Receptors with Agonist or Antagonist Properties
file da validare1995-01-01 Ronsisvalle, G.; Marrazzo, Agostino; Prezzavento, Orazio; Pittala', Valeria; Pappalardo, M. S.; Vittorio, F.; Spampinato, S.
CCB, a novel specific kappa opioid agonist, which discriminates between opioid and sigma 1 recognition sites
1995-01-01 Ronsisvalle, Giuseppe; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Marrazzo, Agostino; Vittorio, F; Gomez Vidal, Ja; Carboni, L; Spampinato, S.
SYNTHESIS OF (+)-(1'R,2'S) AND (1'S,2'R)-6,11-DIMETHYL-1,2,3,4,5,6-HEXAHYDRO-3-[[2'-(ALKOXYCARBONYL)-2'-PHENYLCYCLOPROPYL]METHYL]-2,6-METHANO-3-BENZAZOCIN-8-OL. COMPARISON OF THE AFFINITIES FOR SIGMA 1 AND OPIOID RECEPTORS WITHIN THE DIASTEREOISOMERIC MPCB AND CCB
file da validare1997-01-01 Ronsisvalle, Giuseppe; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Pappalardo, Ms; Marrazzo, Agostino; Vittorio, F; Carboni, L; Spampinato, S.
(+)-cis-N-ethyleneamino-N-normetazocine derivatives. Novel and selective sigma ligands with antagonist properties
1998-01-01 Ronsisvalle, G; Marrazzo, Agostino; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Vittorio, F; Pittala', Valeria; Pappalardo, Ms; Cacciaguerra, S; Spampinato, S.
SYNTHESIS AND SPAMOLYTIC ACTIVITY OF 2-SUBSTITUTED THIENOPYRIMIDIN-4-ONE DERIVATIVES
file da validare2000-01-01 Santagati, N. A.; Prezzavento, Orazio; Ronsisvalle, G; Spampinato, S.
Synthesis of (+) and (−)-cis-2-[(1-adamantylamino)-methyl]-1-phenylcyclopropane derivatives as probe for sigma-1 and sigma-2 binding sites
file da validare2000-01-01 Marrazzo, A; Prezzavento, O.; Vittorio, Franco; Pappalardo, M. S.; Ronsisvalle, G
Nonpeptide Analogues of Dynorphin A(1-8): Design, Synthesis, and Pharmacological Evaluation of k-Selective Agonists
2000-01-01 Ronsisvalle, G; Pasquinucci, Lorella Giuseppina; Pittala', Valeria; Marrazzo, A; Prezzavento, Orazio; DI TORO, R; Falcucci, B; Spampinato, S.
Substituted 1-phenyl-2-cyclopropylmethylamines with high affinity and selectivity for sigma sites
2000-01-01 Ronsisvalle, Giuseppe; Marrazzo, Agostino; Falcucci, B; DI TORO, D; Spampinato, S; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina
Specific kappa opioid receptor agonists
file da validare2000-01-01 Ronsisvalle, G; Marrazzo, A; Pasquinucci, L; Prezzavento, Orazio; Pappalardo, M; Vittorio, F.
Synthesis and pharmacological evaluation of potent and enantioselective sigma-1 and sigma-2 ligands
file da validare2000-01-01 Marrazzo, Agostino; Prezzavento, Orazio; Ronsisvalle, G.
NOVEL 1-PHENYL-2-{[(2,6,6-TRIMETHYLBICYCLO[3.1.1]HEPT-3-YL)AMINO]METHYL}CYCLOPROPANECARBOXYLATE DIASTEREOISOMERS AS POTENT AND ENANTIOSELECTIVE SIGMA-1 AND SIGMA-2 LIGANDS
file da validare2001-01-01 Ronsisvalle, G; Marrazzo, Agostino; Panebianco, A; Prezzavento, Orazio
Methyl 1-phenyl-2-{[(2,6,6-trimethylbicyclo[3.1.1]hept-3-yl)amino]methyl}cyclopropane-carboxylate diastereoisomers as potent and enantioselective sigma-1 and sigma-2 ligands
file da validare2001-01-01 Ronsisvalle, G; Marrazzo, Agostino; Panebianco, A; Prezzavento, Orazio
Novel methyl-2-[4-[(4-hydroxy-4-phenylpiperidin-1-yl)methyl]-1-phenylcyclopropane-carboxylate derivatives as sigma-1 and sigma-2 receptor ligands
file da validare2001-01-01 Prezzavento, O; Massimino, M; Marrazzo, Agostino; Pasquinucci, Lorella Giuseppina; Ronsisvalle, G.
SYNTHESIS OF BNIT AN ISOTHIOCYANATE DERIVATIVE OF N-BENZYL-NORMETAZOCINE AS ACYLANT AGENT FOR σ1 RECEPTOR
file da validare2001-01-01 Prezzavento, Orazio; Massimino, M; Marrazzo, Agostino; Ronsisvalle, G.
Synthesis and pharmacological evaluation of potent and enantioselective sigma-1 and sigma-2 ligands
2001-01-01 Marrazzo, Agostino; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Vittorio, F; Ronsisvalle, Giuseppe
SYNTHESIS AND BINDING AFFINITY OF CIS-(-)- AND CIS-(+)-N-ETHYLENEAMINO-N-NORDEOXYMETAZOCINE AND CIS(-)-N-NORMETAZOCINE ANALOGUES AT SIGMA-1, SIGMA-2 AND KAPPA OPIOID RECEPTORS
file da validare2001-01-01 Ronsisvalle, G; Prezzavento, Orazio; Marrazzo, Agostino; Vittorio, F; Bousquet, E; DI TORO, R; Spampinato, S.
Opioid and sigma receptor studies. New developments in the design of selective sigma ligands
2001-01-01 Ronsisvalle, G; Marrazzo, A; Prezzavento, O; Cagnotto, A; Mennini, T; Parenti, C; Scoto, Giovanna Maria
Benzyl-tropanyl esters and ethers of phenoxypropionic acid as novel sigma receptor ligands
file da validare2002-01-01 Romanelli, M. N.; Dei, S; Gualtieri, F; Scapecchi, S; Teodori, E; Prezzavento, Orazio; Ronsisvalle, G.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
CCB - A novel analog of MPCB with high binding affinity and specific kappa opioid receptor agonist | 1-gen-1994 | Ronsisvalle, Giuseppe; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Carboni, L; Pistacchio, E; Spampinato, S. | file da validare |
New developments in opioid receptors ligands | 1-gen-1995 | Ronsisvalle, G; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Marrazzo, Agostino; Vittorio, F; Pappalardo, Ms; Bousquet, E. | file da validare |
Selective Ligands for Sigma1 Receptors with Agonist or Antagonist Properties | 1-gen-1995 | Ronsisvalle, G.; Marrazzo, Agostino; Prezzavento, Orazio; Pittala', Valeria; Pappalardo, M. S.; Vittorio, F.; Spampinato, S. | file da validare |
CCB, a novel specific kappa opioid agonist, which discriminates between opioid and sigma 1 recognition sites | 1-gen-1995 | Ronsisvalle, Giuseppe; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Marrazzo, Agostino; Vittorio, F; Gomez Vidal, Ja; Carboni, L; Spampinato, S. | |
SYNTHESIS OF (+)-(1'R,2'S) AND (1'S,2'R)-6,11-DIMETHYL-1,2,3,4,5,6-HEXAHYDRO-3-[[2'-(ALKOXYCARBONYL)-2'-PHENYLCYCLOPROPYL]METHYL]-2,6-METHANO-3-BENZAZOCIN-8-OL. COMPARISON OF THE AFFINITIES FOR SIGMA 1 AND OPIOID RECEPTORS WITHIN THE DIASTEREOISOMERIC MPCB AND CCB | 1-gen-1997 | Ronsisvalle, Giuseppe; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Pappalardo, Ms; Marrazzo, Agostino; Vittorio, F; Carboni, L; Spampinato, S. | file da validare |
(+)-cis-N-ethyleneamino-N-normetazocine derivatives. Novel and selective sigma ligands with antagonist properties | 1-gen-1998 | Ronsisvalle, G; Marrazzo, Agostino; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Vittorio, F; Pittala', Valeria; Pappalardo, Ms; Cacciaguerra, S; Spampinato, S. | |
SYNTHESIS AND SPAMOLYTIC ACTIVITY OF 2-SUBSTITUTED THIENOPYRIMIDIN-4-ONE DERIVATIVES | 1-gen-2000 | Santagati, N. A.; Prezzavento, Orazio; Ronsisvalle, G; Spampinato, S. | file da validare |
Synthesis of (+) and (−)-cis-2-[(1-adamantylamino)-methyl]-1-phenylcyclopropane derivatives as probe for sigma-1 and sigma-2 binding sites | 1-gen-2000 | Marrazzo, A; Prezzavento, O.; Vittorio, Franco; Pappalardo, M. S.; Ronsisvalle, G | file da validare |
Nonpeptide Analogues of Dynorphin A(1-8): Design, Synthesis, and Pharmacological Evaluation of k-Selective Agonists | 1-gen-2000 | Ronsisvalle, G; Pasquinucci, Lorella Giuseppina; Pittala', Valeria; Marrazzo, A; Prezzavento, Orazio; DI TORO, R; Falcucci, B; Spampinato, S. | |
Substituted 1-phenyl-2-cyclopropylmethylamines with high affinity and selectivity for sigma sites | 1-gen-2000 | Ronsisvalle, Giuseppe; Marrazzo, Agostino; Falcucci, B; DI TORO, D; Spampinato, S; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina | |
Specific kappa opioid receptor agonists | 1-gen-2000 | Ronsisvalle, G; Marrazzo, A; Pasquinucci, L; Prezzavento, Orazio; Pappalardo, M; Vittorio, F. | file da validare |
Synthesis and pharmacological evaluation of potent and enantioselective sigma-1 and sigma-2 ligands | 1-gen-2000 | Marrazzo, Agostino; Prezzavento, Orazio; Ronsisvalle, G. | file da validare |
NOVEL 1-PHENYL-2-{[(2,6,6-TRIMETHYLBICYCLO[3.1.1]HEPT-3-YL)AMINO]METHYL}CYCLOPROPANECARBOXYLATE DIASTEREOISOMERS AS POTENT AND ENANTIOSELECTIVE SIGMA-1 AND SIGMA-2 LIGANDS | 1-gen-2001 | Ronsisvalle, G; Marrazzo, Agostino; Panebianco, A; Prezzavento, Orazio | file da validare |
Methyl 1-phenyl-2-{[(2,6,6-trimethylbicyclo[3.1.1]hept-3-yl)amino]methyl}cyclopropane-carboxylate diastereoisomers as potent and enantioselective sigma-1 and sigma-2 ligands | 1-gen-2001 | Ronsisvalle, G; Marrazzo, Agostino; Panebianco, A; Prezzavento, Orazio | file da validare |
Novel methyl-2-[4-[(4-hydroxy-4-phenylpiperidin-1-yl)methyl]-1-phenylcyclopropane-carboxylate derivatives as sigma-1 and sigma-2 receptor ligands | 1-gen-2001 | Prezzavento, O; Massimino, M; Marrazzo, Agostino; Pasquinucci, Lorella Giuseppina; Ronsisvalle, G. | file da validare |
SYNTHESIS OF BNIT AN ISOTHIOCYANATE DERIVATIVE OF N-BENZYL-NORMETAZOCINE AS ACYLANT AGENT FOR σ1 RECEPTOR | 1-gen-2001 | Prezzavento, Orazio; Massimino, M; Marrazzo, Agostino; Ronsisvalle, G. | file da validare |
Synthesis and pharmacological evaluation of potent and enantioselective sigma-1 and sigma-2 ligands | 1-gen-2001 | Marrazzo, Agostino; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Vittorio, F; Ronsisvalle, Giuseppe | |
SYNTHESIS AND BINDING AFFINITY OF CIS-(-)- AND CIS-(+)-N-ETHYLENEAMINO-N-NORDEOXYMETAZOCINE AND CIS(-)-N-NORMETAZOCINE ANALOGUES AT SIGMA-1, SIGMA-2 AND KAPPA OPIOID RECEPTORS | 1-gen-2001 | Ronsisvalle, G; Prezzavento, Orazio; Marrazzo, Agostino; Vittorio, F; Bousquet, E; DI TORO, R; Spampinato, S. | file da validare |
Opioid and sigma receptor studies. New developments in the design of selective sigma ligands | 1-gen-2001 | Ronsisvalle, G; Marrazzo, A; Prezzavento, O; Cagnotto, A; Mennini, T; Parenti, C; Scoto, Giovanna Maria | |
Benzyl-tropanyl esters and ethers of phenoxypropionic acid as novel sigma receptor ligands | 1-gen-2002 | Romanelli, M. N.; Dei, S; Gualtieri, F; Scapecchi, S; Teodori, E; Prezzavento, Orazio; Ronsisvalle, G. | file da validare |
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