Sfoglia per Autore
Intramolecular oxidative palladium-catalyzed diamination reactions of alkenyl sulfamates: an efficient synthesis of [1,2,5]thiadiazolo-fused piperazinones
2016-01-01 Chiacchio, U; Broggini, G; Romeo, R; Gazzola, S; Giofre, S; Gabriele, B; Mancuso, R; Floresta, G; Zagni, C; Chiacchio, M
γ-Cyclodextrin as a Catalyst for the Synthesis of 2-Methyl-3,5-diarylisoxazolidines in Water
2017-01-01 Floresta, Giuseppe; Talotta, Carmen; Gaeta, Carmine; De Rosa, Margherita; Chiacchio, Ugo; Neri, Placido; Rescifina, Antonio
The Search for Potent, Small-Molecule HDACIs in Cancer Treatment: A Decade After Vorinostat
2017-01-01 Zagni, Chiara; Floresta, Giuseppe; Monciino, Giulia; Rescifina, Antonio
Development of a Sigma-2 Receptor affinity filter through a Monte Carlo based QSAR analysis
2017-01-01 Rescifina, Antonio; Floresta, Giuseppe; Marrazzo, Agostino; Parenti, Carmela; Prezzavento, Orazio; Nastasi, Giovanni; Dichiara, Maria; Amata, Emanuele
Synthesis and evaluation of haloperidol metabolite II prodrugs as anticancer agents
2017-01-01 Dichiara, Maria; Amata, Emanuele; Rescifina, Antonio; Prezzavento, Orazio; Floresta, Giuseppe; Parenti, Carmela; Pittalà, Valeria; Marrazzo, Agostino
Adipocyte fatty acid binding protein 4 (FABP4) inhibitors. A comprehensive systematic review
2017-01-01 Floresta, Giuseppe; Pistarà, Venerando; Amata, Emanuele; Dichiara, Maria; Marrazzo, Agostino; Prezzavento, Orazio; Rescifina, Antonio
Sigma-2 receptor ligands QSAR model dataset
2017-01-01 Rescifina, Antonio; Floresta, Giuseppe; Marrazzo, Agostino; Parenti, Carmela; Prezzavento, Orazio; Nastasi, Giovanni; Dichiara, Maria; Amata, Emanuele
Hyphenated 3D-QSAR statistical model-scaffold hopping analysis for the identification of potentially potent and selective sigma-2 receptor ligands
2017-01-01 Floresta, Giuseppe; Rescifina, Antonio; Marrazzo, Agostino; Dichiara, Maria; Pistarà, Venerando; Pittalà, Valeria; Prezzavento, Orazio; Amata, Emanuele
Potholing of the hydrophobic heme oxygenase-1 western region for the search of potent and selective imidazole-based inhibitors
2018-01-01 Salerno, Loredana; Amata, Emanuele; Romeo, Giuseppe; Marrazzo, Agostino; Floresta, Giuseppe; Modica Maria, N.; Greish Khaled, F.; Sorrenti, Valeria; Rescifina, Antonio; Pittalà, Valeria
Rosmarinic acid amides: synthesis, α-glucosidase inhibition and enzyme binding mode
file da validare2018-01-01 Cardullo, N.; Catinella, G.; Floresta, G.; Rosselli, S.; Rescifina, A.; Bruno, M.; Tringali, C.
Targeting the hydrophobic heme oxygenase-1 western region for the identification of novel and selective azole-based inhibitors.
file da validare2018-01-01 Dichiara, M; Modica, Mn; Leonardi, C; Margani, F; Ciaffaglione, V; Fallica, An; Floresta, G; Gentile, D; Cosenza, J; Pittalà, V.
Identification of Potentially Potent Heme Oxygenase 1 Inhibitors through 3D-QSAR Coupled to Scaffold-Hopping Analysis
2018-01-01 Floresta, Giuseppe; Amata, Emanuele; Dichiara, Maria; Marrazzo, Agostino; Salerno, Loredana; Romeo, Giuseppe; Prezzavento, Orazio; Pittalà, Valeria; Rescifina, Antonio
Potholing of the hydrophobic heme oxygenase-1 western region for the search of potent and selective imidazole-based inhibitors
2018-01-01 Salerno, Loredana; Amata, Emanuele; Romeo, Giuseppe; Marrazzo, Agostino; Prezzavento, Orazio; Floresta, Giuseppe; Sorrenti, Valeria; Barbagallo, Ignazio; Rescifina, Antonio; Pittalà, Valeria
DNA intercalators based on (1,10-phenanthrolin-2-yl)isoxazolidin-5-yl core with better growth inhibition and selectivity than cisplatin upon head and neck squamous cells carcinoma
2018-01-01 Varrica G., Maria; Zagni, Chiara; Mineo, Placido; Floresta, Giuseppe; Monciino, Giulia; Pistara, Venerando; Abbadessa, Antonio; Nicosia, Angelo; Castilho M., Rogerio; Amata, Emanuele; Rescifina, Antonio
Mild Friedel–Crafts Reactions inside a Hexameric Resorcinarene Capsule: C−Cl Bond Activation through Hydrogen Bonding to Bridging Water Molecules
2018-01-01 La Manna, Pellegrino; Talotta, Carmen; Floresta, Giuseppe; De Rosa, Margherita; Soriente, Annunziata; Rescifina, Antonio; Gaeta, Carmine; Neri, Placido
The hexameric resorcinarene capsule as an artificial enzyme: Ruling the regio and stereochemistry of a 1,3-dipolar cycloaddition between nitrones and unsaturated aldehydes
2018-01-01 La Manna, Pellegrino; De Rosa, Margherita; Talotta, Carmen; Gaeta, Carmine; Soriente, Annunziata; Floresta, Giuseppe; Rescifina, Antonio; Neri, Placido
Development of new HO-1 inhibitors by a thorough scaffold-hopping analysis
2018-01-01 Floresta, G; Pittalà, V; Sorrenti, V; Romeo, G; Salerno, L; Rescifina, A.
Targeting heme Oxygenase-1 with hybrid compounds to overcome Imatinib resistance in chronic myeloid leukemia cell lines
2018-01-01 Sorrenti, Valeria; Pittalà, Valeria; Romeo, Giuseppe; Amata, Emanuele; Dichiara, Maria; Marrazzo, Agostino; Turnaturi, Rita; Prezzavento, Orazio; Barbagallo, Ignazio; Vanella, Luca; Rescifina, Antonio; Floresta, Giuseppe; Tibullo, Daniele; DI RAIMONDO, Francesco; Intagliata, Sebastiano; Salerno, Loredana
A pseudouridine isoxazolidinyl nucleoside analogue structural analysis: A morphological approach
2018-01-01 Floresta, Giuseppe; Pistara', Venerando; Christensen E., Kirsten; Amata, Emanuele; Marrazzo, Agostino; Gentile, Davide; Rescifina, Antonio; Punzo, Francesco
A structure-and ligand-based virtual screening of a database of “small” marine natural products for the identification of “blue” sigma-2 receptor ligands
2018-01-01 Floresta, Giuseppe; Amata, Emanuele; Barbaraci, Carla; Gentile, Davide; Turnaturi, Rita; Marrazzo, Agostino; Rescifina, Antonio
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Intramolecular oxidative palladium-catalyzed diamination reactions of alkenyl sulfamates: an efficient synthesis of [1,2,5]thiadiazolo-fused piperazinones | 1-gen-2016 | Chiacchio, U; Broggini, G; Romeo, R; Gazzola, S; Giofre, S; Gabriele, B; Mancuso, R; Floresta, G; Zagni, C; Chiacchio, M | |
γ-Cyclodextrin as a Catalyst for the Synthesis of 2-Methyl-3,5-diarylisoxazolidines in Water | 1-gen-2017 | Floresta, Giuseppe; Talotta, Carmen; Gaeta, Carmine; De Rosa, Margherita; Chiacchio, Ugo; Neri, Placido; Rescifina, Antonio | |
The Search for Potent, Small-Molecule HDACIs in Cancer Treatment: A Decade After Vorinostat | 1-gen-2017 | Zagni, Chiara; Floresta, Giuseppe; Monciino, Giulia; Rescifina, Antonio | |
Development of a Sigma-2 Receptor affinity filter through a Monte Carlo based QSAR analysis | 1-gen-2017 | Rescifina, Antonio; Floresta, Giuseppe; Marrazzo, Agostino; Parenti, Carmela; Prezzavento, Orazio; Nastasi, Giovanni; Dichiara, Maria; Amata, Emanuele | |
Synthesis and evaluation of haloperidol metabolite II prodrugs as anticancer agents | 1-gen-2017 | Dichiara, Maria; Amata, Emanuele; Rescifina, Antonio; Prezzavento, Orazio; Floresta, Giuseppe; Parenti, Carmela; Pittalà, Valeria; Marrazzo, Agostino | |
Adipocyte fatty acid binding protein 4 (FABP4) inhibitors. A comprehensive systematic review | 1-gen-2017 | Floresta, Giuseppe; Pistarà, Venerando; Amata, Emanuele; Dichiara, Maria; Marrazzo, Agostino; Prezzavento, Orazio; Rescifina, Antonio | |
Sigma-2 receptor ligands QSAR model dataset | 1-gen-2017 | Rescifina, Antonio; Floresta, Giuseppe; Marrazzo, Agostino; Parenti, Carmela; Prezzavento, Orazio; Nastasi, Giovanni; Dichiara, Maria; Amata, Emanuele | |
Hyphenated 3D-QSAR statistical model-scaffold hopping analysis for the identification of potentially potent and selective sigma-2 receptor ligands | 1-gen-2017 | Floresta, Giuseppe; Rescifina, Antonio; Marrazzo, Agostino; Dichiara, Maria; Pistarà, Venerando; Pittalà, Valeria; Prezzavento, Orazio; Amata, Emanuele | |
Potholing of the hydrophobic heme oxygenase-1 western region for the search of potent and selective imidazole-based inhibitors | 1-gen-2018 | Salerno, Loredana; Amata, Emanuele; Romeo, Giuseppe; Marrazzo, Agostino; Floresta, Giuseppe; Modica Maria, N.; Greish Khaled, F.; Sorrenti, Valeria; Rescifina, Antonio; Pittalà, Valeria | |
Rosmarinic acid amides: synthesis, α-glucosidase inhibition and enzyme binding mode | 1-gen-2018 | Cardullo, N.; Catinella, G.; Floresta, G.; Rosselli, S.; Rescifina, A.; Bruno, M.; Tringali, C. | file da validare |
Targeting the hydrophobic heme oxygenase-1 western region for the identification of novel and selective azole-based inhibitors. | 1-gen-2018 | Dichiara, M; Modica, Mn; Leonardi, C; Margani, F; Ciaffaglione, V; Fallica, An; Floresta, G; Gentile, D; Cosenza, J; Pittalà, V. | file da validare |
Identification of Potentially Potent Heme Oxygenase 1 Inhibitors through 3D-QSAR Coupled to Scaffold-Hopping Analysis | 1-gen-2018 | Floresta, Giuseppe; Amata, Emanuele; Dichiara, Maria; Marrazzo, Agostino; Salerno, Loredana; Romeo, Giuseppe; Prezzavento, Orazio; Pittalà, Valeria; Rescifina, Antonio | |
Potholing of the hydrophobic heme oxygenase-1 western region for the search of potent and selective imidazole-based inhibitors | 1-gen-2018 | Salerno, Loredana; Amata, Emanuele; Romeo, Giuseppe; Marrazzo, Agostino; Prezzavento, Orazio; Floresta, Giuseppe; Sorrenti, Valeria; Barbagallo, Ignazio; Rescifina, Antonio; Pittalà, Valeria | |
DNA intercalators based on (1,10-phenanthrolin-2-yl)isoxazolidin-5-yl core with better growth inhibition and selectivity than cisplatin upon head and neck squamous cells carcinoma | 1-gen-2018 | Varrica G., Maria; Zagni, Chiara; Mineo, Placido; Floresta, Giuseppe; Monciino, Giulia; Pistara, Venerando; Abbadessa, Antonio; Nicosia, Angelo; Castilho M., Rogerio; Amata, Emanuele; Rescifina, Antonio | |
Mild Friedel–Crafts Reactions inside a Hexameric Resorcinarene Capsule: C−Cl Bond Activation through Hydrogen Bonding to Bridging Water Molecules | 1-gen-2018 | La Manna, Pellegrino; Talotta, Carmen; Floresta, Giuseppe; De Rosa, Margherita; Soriente, Annunziata; Rescifina, Antonio; Gaeta, Carmine; Neri, Placido | |
The hexameric resorcinarene capsule as an artificial enzyme: Ruling the regio and stereochemistry of a 1,3-dipolar cycloaddition between nitrones and unsaturated aldehydes | 1-gen-2018 | La Manna, Pellegrino; De Rosa, Margherita; Talotta, Carmen; Gaeta, Carmine; Soriente, Annunziata; Floresta, Giuseppe; Rescifina, Antonio; Neri, Placido | |
Development of new HO-1 inhibitors by a thorough scaffold-hopping analysis | 1-gen-2018 | Floresta, G; Pittalà, V; Sorrenti, V; Romeo, G; Salerno, L; Rescifina, A. | |
Targeting heme Oxygenase-1 with hybrid compounds to overcome Imatinib resistance in chronic myeloid leukemia cell lines | 1-gen-2018 | Sorrenti, Valeria; Pittalà, Valeria; Romeo, Giuseppe; Amata, Emanuele; Dichiara, Maria; Marrazzo, Agostino; Turnaturi, Rita; Prezzavento, Orazio; Barbagallo, Ignazio; Vanella, Luca; Rescifina, Antonio; Floresta, Giuseppe; Tibullo, Daniele; DI RAIMONDO, Francesco; Intagliata, Sebastiano; Salerno, Loredana | |
A pseudouridine isoxazolidinyl nucleoside analogue structural analysis: A morphological approach | 1-gen-2018 | Floresta, Giuseppe; Pistara', Venerando; Christensen E., Kirsten; Amata, Emanuele; Marrazzo, Agostino; Gentile, Davide; Rescifina, Antonio; Punzo, Francesco | |
A structure-and ligand-based virtual screening of a database of “small” marine natural products for the identification of “blue” sigma-2 receptor ligands | 1-gen-2018 | Floresta, Giuseppe; Amata, Emanuele; Barbaraci, Carla; Gentile, Davide; Turnaturi, Rita; Marrazzo, Agostino; Rescifina, Antonio |
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