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Mostrati risultati da 1 a 20 di 24
Titolo Data di pubblicazione Autore(i) File
New synthetic approach to fused heterocycloquinazolines 1-gen-1999 Santagati, Andrea; Modica, M; MONS SCOLARO, L; Santagati, M. file da validare
Synthesis of new [1,3,4]thiadiazolo[3,2-a]thieno[2,3-a]pyrimidinone derivatives with antiinflammatory activity 1-gen-2000 Modica, Maria; Santagati, Maria; Santagati, Andrea; Cutuli, Vincenza; Mangano, Nunzio; Caruso, Antonella file da validare
High potent and selective arylpiperazine derivatives as ligands for the 5-HT1A receptor 1-gen-2000 Modica, Maria Nunziata; Santagati, M; Santagati, Andrea; Russo, F; Cagnotto, A; Goegan, M; Mennini, T. file da validare
New synthetic approaches to bridgehead nitrogen heterocycles derived from 3-amino-2,3-dihydro-5,6-dimethyl-2-thioxo-thieno[2,3-d]pyrimidin-4(1H)-one and its salts 1-gen-2000 Santagati, Andrea; Modica, Maria Nunziata; Santagati, Maria file da validare
Synthesis and pharmacological screening of 1,3,4-thiadiazino[2,3-b]quinazoline derivatives 1-gen-2000 Santagati, Andrea; Modica, Maria Nunziata; Santagati, M; Cutuli, V; Mangano, N. G.; Caruso, A. file da validare
Synthetic route to 4,5-dihydro-9H-pyrido[1,2-a]thieno[3,2-e]pyrimidine derivative through 1,3-dipolar cycloaddition 1-gen-2001 Santagati, Andrea; Granata, G; Santagati, M. file da validare
Synthesis of new thienotriazolopyrimidine and thienopyrimidotetrazine derivatives from bifunctional intermediates 1-gen-2001 Maria, Modica; Maria, Santagati; Santagati, Andrea file da validare
Thienopyrimidine derivatives prevent cartilage destruction in articular disease 1-gen-2001 Panico, Anna Maria; Cardile, Venera; Santagati, Andrea; Gentile, Barbara
Synthesis and activity of phenyl derivatives containing 5,6-dimethyl-thieno[2,3-d]pyrimidin-4-(1H)-one or 4H-pyrimido[5,4-b]indo-4-one. Heterocyclic system as potential non-steroidal anti-inflammatory drugs 1-gen-2002 Santagati, Andrea; Giuseppe, Granata; Maria, Santagati; Vincenza, Cutuli; NUNZIO GUIDO, Mangano; Antonella, Caruso file da validare
Calorimetric study on the interaction of thienopyrimidine derivatives with phosphatidylcholine membranes 1-gen-2003 Panico, Anna Maria; Santagati, A; Cardile, Venera; Urso, D; Gentile, B; Ronsisvalle, G.
Synthesis and effects on the COX-1 and COX-2 activity in Human Whole Blood ex vivo of derivatives containing the [1]benzothienol[3,2-d]pyrimidin-4-one heterocyclic system 1-gen-2003 Santagati, Andrea; Giuseppe, Granata; Marrazzo, Agostino; Maria, Santagati
Synthesis of potential selective COX-2 enzyme inhibitors derived from ethyl ester of 2-isothiocyanato-5-phenyl-3-thiophenecarboxylic acid 1-gen-2003 Santagati, A; Marrazzo, Agostino; Granata, G.
Methanesulphonamide of 3,5-dihydro-4H-pyrimido[5,4-b]indol4-one and [1]Benzothieno[3,2-d]pirimidin-4(3H)-one derivatives as potential COX-2 inhibitors 1-gen-2005 Barbagallo, Salvatore; Granata, Giuseppe; Perdicaro, A; Marrazzo, Agostino; Santagati, A; Ronsisvalle, G. file da validare
Synthetic Approaches to Bridgehead Nitrogen Methanesulfonamide Derivatives of 3-Amino-2-thioxo-2,3-dihydrothieno[2,3-d]pyrimidin-4(1H)-ones, Potential COX-2 Selective Inhibitors 1-gen-2006 Granata, G; Barbagallo, S; Perdicaro, A; Marrazzo, Agostino; Santagati, Andrea; Lombardo, L; Cardile, Venera
Molecular modelling of a novel class of N5-methanesulfonamide dihydrothienopyrimidinoners as potential dual COX-2 inhibitor/ 1-gen-2007 Santagati, Andrea; Giuseppwe, Granata; Cardile, Venera; Guccione, Salvatore; Laura, Giurato file da validare
Copper-Catalyzed Coupling Reaction of 2-Thioxo-4-quinazolinone and Thieno[3,2-d]pyrimidin-4-one Methane Sulphonamide with Aryl Iodide : Preparation of Potential COX-2 Selective Inhibitors 1-gen-2008 Antonio, Perdicaro; Giuseppe, Granata; Marrazzo, Agostino; Santagati, Andrea
Inhibition of iNOS and COX-2 in human whole blood ex vivo and monocyte-macrophage J774 cells by a new group of aminothiopyrimidone derivatives 1-gen-2009 Cardile, Venera; Lombardo, L; Granata, G; Perdicaro, A; Balazy, M; Santagati, A.
Sulfonilamidothiopyrimidone and thiopyrimidone derivatives as selective COX-2 inhibitors: Synthesis, biological evaluation, and docking studies 1-gen-2012 Livia, Basile; Susana, Álvarez; Almudena, Blanco; Santagati, Andrea; Giuseppe, Granata; Patrizia Di, Pietro; Guccione, Salvatore; Ma Ángeles Muñoz, Fernandez file da validare
Cyclooxygenase-2 and cancer : development of vew fluorescent inhibitors of cox-2 for cancer detection 1-gen-2013 Mariarita, Barone; Santagati, Andrea; Alfio, Catalfo; DE GUIDI, Guido; Cardile, Venera file da validare
Synthesis and biological evaluation of new benzo-thieno[3,2-d]pyrimidin-4-one sulphonamide thio-derivatives as potential selective cyclooxygenase-2 inhibitors 1-gen-2013 Barone, M; Graziano, ADRIANA CAROL; Marrazzo, Agostino; Gemmellaro, P; Santagati, Andrea; Cardile, Venera
Mostrati risultati da 1 a 20 di 24
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