AMATA, EMANUELE
AMATA, EMANUELE
SCIENZE DEL FARMACO E DELLA SALUTE (DSFS) (Department of Drug and Health Sciences)
[1]Benzothieno[3,2-d]pyrimidine derivatives as ligands for the serotonergic 5-HT7 receptor
2019-01-01 Romeo, G.; Salerno, L.; Pittalà, V.; Candido, M.; Intagliata, S.; Amata, E.; Salmona, M.; Cagnotto, A.; Rescifina, A.; Floresta, G.; Modica, M. N.
4-Nitro-2,1,3-benzoxadiazole derivatives as potential fluorescent sigma receptor probes
2015-01-01 Schinina', Barbara; Martorana, Andrea; Colabufo Nicola, Antonio; Contino, Marialessandra; Niso, Mauro; Perrone Maria, Grazia; DE GUIDI, Guido; Catalfo, Alfio; Rappazzo, Giancarlo; Zuccarello, Elisa; Prezzavento, Orazio; Amata, Emanuele; Rescifina, Antonio; Marrazzo, Agostino
Adipocyte fatty acid binding protein 4 (FABP4) inhibitors. A comprehensive systematic review
2017-01-01 Floresta, Giuseppe; Pistarà, Venerando; Amata, Emanuele; Dichiara, Maria; Marrazzo, Agostino; Prezzavento, Orazio; Rescifina, Antonio
(+)-and (−)-Phenazocine enantiomers: evaluation of their dual opioid agonist/σ1 antagonist properties and antinociceptive effects
2017-01-01 Prezzavento, Orazio; Arena, Emanuela; Sánchez-Fernández, Cristine; Turnaturi, Rita; Parenti, Carmela; Marrazzo, Agostino; Catalano, Roberto; Amata, Emanuele; Pasquinucci, Lorella; Cobos J., Enrique
Antiangiogenic Effect of (±)-Haloperidol Metabolite II Valproate Ester [(±)-MRJF22] in Human Microvascular Retinal Endothelial Cells
2016-01-01 Olivieri, Melania; Amata, Emanuele; Vinciguerra, Shila; Fiorito, Jole; Giurdanella, Giovanni; Drago, Filippo; Caporarello, Nunzia; Prezzavento, Orazio; Arena, Emanuela; Salerno, Loredana; Rescifina, Antonio; Lupo, Gabriella; Anfuso, CARMELINA DANIELA; Marrazzo, Agostino
Antioxidant activity of (+)-Pentazocine on activated microglia
2015-01-01 Marrazzo, Agostino; Heiss, Kathrin; Prezzavento, Orazio; Arena, Emanuela; Amata, Emanuele; LI VOLTI, Giovanni
Antioxidant properties and pharmacokinetic studies of new selective σ1 bifunctional ligands
2015-01-01 Marrazzo, Agostino; Arena, Emanuela; Cacciatore, Ivana; Cerasa Laura, S.; Amata, Emanuele; Pittala', Valeria; Pasquinucci, Lorella Giuseppina; Turkez, Hasan; Di Stefano, Antonio; Prezzavento, Orazio
Antitrypanosomal lead discovery: Identification of a ligand-efficient inhibitor of Trypanosoma cruzi CYP51 and parasite growth
2013-01-01 Andriani, Grasiella; Amata, Emanuele; Beatty, Joel; Clements, Zeke; Coffey J., Brian; Courtemanche, Gilles; Devine, William; Erath, Jessey; Juda E., Cristin; Wawrzak, Zdzislaw; Wood T., Jodianne; Lepesheva L., Galina; Rodriguez, Ana; Pollastri P., Michael
C-5'-Triazolyl-2'-oxa-3'-aza-4'a-carbanucleosides: Synthesis and biological evaluation
2015-01-01 Romeo, Roberto; Carnovale, Caterina; Giofrè V., Salvatore; Chiacchio, MARIA ASSUNTA ROSSELLA; Garozzo, Adriana; Amata, Emanuele; Romeo, Giovanni; Chiacchio, Ugo
Caspase-3 activation in human melanoma A375 cell line by a novel selective sigma-2 agonist
2016-01-01 Ronsisvalle, Simone; Arico, Giuseppina; Cova, ANNA MARIA; Blanco, Palma; Amata, Emanuele; Pappalardo, Maria Sebastiana; Pasquinucci, Lorella; Spadaro, Angelo; Ronsisvalle, Nicole
CNS permeability parameters determination through a statistical analysis driven approach
2019-01-01 Dichiara, Maria; Marrazzo, Agostino; Amata, Emanuele
Combination of heme oxygenase-1 inhibition and sigma receptor modulation for anticancer activity
2021-01-01 Romeo, G.; Ciaffaglione, V.; Amata, E.; Dichiara, M.; Calabrese, L.; Vanella, L.; Sorrenti, V.; Grosso, S.; D'Amico, A. G.; D'Agata, V.; Intagliata, S.; Salerno, L.
Composti inorganici [Cap. 6]
2017-01-01 Amata, Emanuele; Dichiara, Maria
Comprehensive data on a 2D-QSAR model for Heme Oxygenase isoform 1 inhibitors
2017-01-01 Amata, Emanuele; Marrazzo, Agostino; Dichiara, Maria; Modica Maria, N.; Salerno, Loredana; Prezzavento, Orazio; Nastasi, Giovanni; Rescifina, Antonio; Romeo, Giuseppe; Pittalà, Valeria
Design and synthesis of new benzomorphan LP1 analogues, an opioid ligand with low development of tolerance
2009-01-01 Amata, Emanuele
Design, synthesis, and pharmacological evaluation of NO donor-sigma receptors hybrids for the treatment of cancer
2018-01-01 Dichiara, Maria; Barbaraci, Carla; Gentile, Davide; Intagliata, Sebastiano; Pittalà, Valeria; Arena, Emanuelea; Fraix, Aurore; Farina, Giuseppe; Prezzavento, Orazio; Amata, Emanuele; Marrazzo, Agostino.
Development of a Sigma-2 Receptor affinity filter through a Monte Carlo based QSAR analysis
2017-01-01 Rescifina, Antonio; Floresta, Giuseppe; Marrazzo, Agostino; Parenti, Carmela; Prezzavento, Orazio; Nastasi, Giovanni; Dichiara, Maria; Amata, Emanuele
Development of new benzomorphan LP1 analogues
2008-01-01 Pasquinucci, Lorella Giuseppina; Amata, Emanuele; Ronsisvalle, Giuseppe
Development of NO-releasing sigma receptor hybrids as anticancer agents
2019-01-01 Dichiara, Maria; Acquaviva, Rosaria; La Mantia, Alfonsina; DI GIACOMO, Claudia; Arena, Emanuele; Floresta, Giuseppe; Marrazzo, Agostino; Amata, Emanuele; Prezzavento, Orazio
Development of novel H2S-donor sigma receptor hybrids for the management of pain.
2019-01-01 Dichiara, Maria; Pitino, Cristina; Barbaraci, Carla; Artacho-Cordón, A.; Cobos Enrique, J; Marrazzo, Agostino; Amata, Emanuele
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| [1]Benzothieno[3,2-d]pyrimidine derivatives as ligands for the serotonergic 5-HT7 receptor | 1-gen-2019 | Romeo, G.; Salerno, L.; Pittalà, V.; Candido, M.; Intagliata, S.; Amata, E.; Salmona, M.; Cagnotto, A.; Rescifina, A.; Floresta, G.; Modica, M. N. | |
| 4-Nitro-2,1,3-benzoxadiazole derivatives as potential fluorescent sigma receptor probes | 1-gen-2015 | Schinina', Barbara; Martorana, Andrea; Colabufo Nicola, Antonio; Contino, Marialessandra; Niso, Mauro; Perrone Maria, Grazia; DE GUIDI, Guido; Catalfo, Alfio; Rappazzo, Giancarlo; Zuccarello, Elisa; Prezzavento, Orazio; Amata, Emanuele; Rescifina, Antonio; Marrazzo, Agostino | |
| Adipocyte fatty acid binding protein 4 (FABP4) inhibitors. A comprehensive systematic review | 1-gen-2017 | Floresta, Giuseppe; Pistarà, Venerando; Amata, Emanuele; Dichiara, Maria; Marrazzo, Agostino; Prezzavento, Orazio; Rescifina, Antonio | |
| (+)-and (−)-Phenazocine enantiomers: evaluation of their dual opioid agonist/σ1 antagonist properties and antinociceptive effects | 1-gen-2017 | Prezzavento, Orazio; Arena, Emanuela; Sánchez-Fernández, Cristine; Turnaturi, Rita; Parenti, Carmela; Marrazzo, Agostino; Catalano, Roberto; Amata, Emanuele; Pasquinucci, Lorella; Cobos J., Enrique | |
| Antiangiogenic Effect of (±)-Haloperidol Metabolite II Valproate Ester [(±)-MRJF22] in Human Microvascular Retinal Endothelial Cells | 1-gen-2016 | Olivieri, Melania; Amata, Emanuele; Vinciguerra, Shila; Fiorito, Jole; Giurdanella, Giovanni; Drago, Filippo; Caporarello, Nunzia; Prezzavento, Orazio; Arena, Emanuela; Salerno, Loredana; Rescifina, Antonio; Lupo, Gabriella; Anfuso, CARMELINA DANIELA; Marrazzo, Agostino | |
| Antioxidant activity of (+)-Pentazocine on activated microglia | 1-gen-2015 | Marrazzo, Agostino; Heiss, Kathrin; Prezzavento, Orazio; Arena, Emanuela; Amata, Emanuele; LI VOLTI, Giovanni | |
| Antioxidant properties and pharmacokinetic studies of new selective σ1 bifunctional ligands | 1-gen-2015 | Marrazzo, Agostino; Arena, Emanuela; Cacciatore, Ivana; Cerasa Laura, S.; Amata, Emanuele; Pittala', Valeria; Pasquinucci, Lorella Giuseppina; Turkez, Hasan; Di Stefano, Antonio; Prezzavento, Orazio | |
| Antitrypanosomal lead discovery: Identification of a ligand-efficient inhibitor of Trypanosoma cruzi CYP51 and parasite growth | 1-gen-2013 | Andriani, Grasiella; Amata, Emanuele; Beatty, Joel; Clements, Zeke; Coffey J., Brian; Courtemanche, Gilles; Devine, William; Erath, Jessey; Juda E., Cristin; Wawrzak, Zdzislaw; Wood T., Jodianne; Lepesheva L., Galina; Rodriguez, Ana; Pollastri P., Michael | |
| C-5'-Triazolyl-2'-oxa-3'-aza-4'a-carbanucleosides: Synthesis and biological evaluation | 1-gen-2015 | Romeo, Roberto; Carnovale, Caterina; Giofrè V., Salvatore; Chiacchio, MARIA ASSUNTA ROSSELLA; Garozzo, Adriana; Amata, Emanuele; Romeo, Giovanni; Chiacchio, Ugo | |
| Caspase-3 activation in human melanoma A375 cell line by a novel selective sigma-2 agonist | 1-gen-2016 | Ronsisvalle, Simone; Arico, Giuseppina; Cova, ANNA MARIA; Blanco, Palma; Amata, Emanuele; Pappalardo, Maria Sebastiana; Pasquinucci, Lorella; Spadaro, Angelo; Ronsisvalle, Nicole | |
| CNS permeability parameters determination through a statistical analysis driven approach | 1-gen-2019 | Dichiara, Maria; Marrazzo, Agostino; Amata, Emanuele | |
| Combination of heme oxygenase-1 inhibition and sigma receptor modulation for anticancer activity | 1-gen-2021 | Romeo, G.; Ciaffaglione, V.; Amata, E.; Dichiara, M.; Calabrese, L.; Vanella, L.; Sorrenti, V.; Grosso, S.; D'Amico, A. G.; D'Agata, V.; Intagliata, S.; Salerno, L. | |
| Composti inorganici [Cap. 6] | 1-gen-2017 | Amata, Emanuele; Dichiara, Maria | |
| Comprehensive data on a 2D-QSAR model for Heme Oxygenase isoform 1 inhibitors | 1-gen-2017 | Amata, Emanuele; Marrazzo, Agostino; Dichiara, Maria; Modica Maria, N.; Salerno, Loredana; Prezzavento, Orazio; Nastasi, Giovanni; Rescifina, Antonio; Romeo, Giuseppe; Pittalà, Valeria | |
| Design and synthesis of new benzomorphan LP1 analogues, an opioid ligand with low development of tolerance | 1-gen-2009 | Amata, Emanuele | |
| Design, synthesis, and pharmacological evaluation of NO donor-sigma receptors hybrids for the treatment of cancer | 1-gen-2018 | Dichiara, Maria; Barbaraci, Carla; Gentile, Davide; Intagliata, Sebastiano; Pittalà, Valeria; Arena, Emanuelea; Fraix, Aurore; Farina, Giuseppe; Prezzavento, Orazio; Amata, Emanuele; Marrazzo, Agostino. | |
| Development of a Sigma-2 Receptor affinity filter through a Monte Carlo based QSAR analysis | 1-gen-2017 | Rescifina, Antonio; Floresta, Giuseppe; Marrazzo, Agostino; Parenti, Carmela; Prezzavento, Orazio; Nastasi, Giovanni; Dichiara, Maria; Amata, Emanuele | |
| Development of new benzomorphan LP1 analogues | 1-gen-2008 | Pasquinucci, Lorella Giuseppina; Amata, Emanuele; Ronsisvalle, Giuseppe | |
| Development of NO-releasing sigma receptor hybrids as anticancer agents | 1-gen-2019 | Dichiara, Maria; Acquaviva, Rosaria; La Mantia, Alfonsina; DI GIACOMO, Claudia; Arena, Emanuele; Floresta, Giuseppe; Marrazzo, Agostino; Amata, Emanuele; Prezzavento, Orazio | |
| Development of novel H2S-donor sigma receptor hybrids for the management of pain. | 1-gen-2019 | Dichiara, Maria; Pitino, Cristina; Barbaraci, Carla; Artacho-Cordón, A.; Cobos Enrique, J; Marrazzo, Agostino; Amata, Emanuele |