MARRAZZO, Agostino
MARRAZZO, Agostino
SCIENZE DEL FARMACO E DELLA SALUTE (DSFS) (Department of Drug and Health Sciences)
(+)-and (−)-Phenazocine enantiomers: evaluation of their dual opioid agonist/σ1 antagonist properties and antinociceptive effects
2017-01-01 Prezzavento, Orazio; Arena, Emanuela; Sánchez-Fernández, Cristine; Turnaturi, Rita; Parenti, Carmela; Marrazzo, Agostino; Catalano, Roberto; Amata, Emanuele; Pasquinucci, Lorella; Cobos J., Enrique
(+)-cis-N-ethyleneamino-N-normetazocine derivatives. Novel and selective sigma ligands with antagonist properties
1998-01-01 Ronsisvalle, G; Marrazzo, Agostino; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Vittorio, F; Pittala', Valeria; Pappalardo, Ms; Cacciaguerra, S; Spampinato, S.
(+)-Methyl (1R,2S)-2-{[4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl]methyl}-1-phenylcyclopropanecarboxylate [(+)-MR200] Derivatives as Potent and Selective Sigma Receptor Ligands: Stereochemistry and Pharmacological Properties
2018-01-01 Amata, Emanuele; Rescifina, Antonio; Prezzavento, Orazio; Arena, Emanuela; Dichiara, Maria; Pittalà, Valeria; Montilla-Garcia, A ngeles; Punzo, Francesco; Merino, Pedro; Cobos J., Enrique; Marrazzo, Agostino
(+)-MR200 derivatives as potential new selective sigma ligands
file da validare2007-01-01 Marrazzo, Agostino; Ronsisvalle, Simone; Prezzavento, O; Vittorio, F; Ronsisvalle, Giuseppe
(+)-MR200 derivatives as potenzial new selective ligands
file da validare2007-01-01 Marrazzo, Agostino; Ronsisvalle, Simone; Prezzavento, Orazio; Franco, Vittorio; Giuseppe, Ronsisvalle
(+)-Mr200 derivatives: modifications on the amino moiety. In vitro and in vivo pharmacological evaluation
file da validare2008-01-01 Marrazzo, Agostino; Cobos, E. J.; Iemolo, A; Gonzàlez, L. G.; Prezzavento, Orazio; Parenti, Carmela; Aricò, G; Sanfilippo, M; Ronsisvalle, Simone; Scoto, Giovanna Maria
(+)-Pentazocine attenuates SH-SY5Y cell death, oxidative stress and microglial migration induced by conditioned medium from activated microglia
2017-01-01 Heiss, K; Raffaele, M; Vanella, L; Murabito, P; Prezzavento, O; Marrazzo, Agostino; Aricò, G; CASTRUCCIO CASTRACANI, Carlo; Barbagallo, IGNAZIO ALBERTO; Zappala', Agata; Avola, Roberto; LI VOLTI, Giovanni
(+)-Pentazocine reduces oxidative stress and apoptosis in microglia following hypoxia/reoxygenation injury
2016-01-01 Heiss, K; Vanella, Luca; Murabito, P; Prezzavento, Orazio; Marrazzo, Agostino; CASTRUCCIO CASTRACANI, Carlo; Barbagallo, IGNAZIO ALBERTO; Zappala', Agata; Arena, E; Astuto, Marinella; Giarratano, A; LI VOLTI, Giovanni
1-Phenyl-3azabicyclo[3.1.0]hexane derivatives as new ligands for sigma receptors
file da validare2004-01-01 Marrazzo, Agostino; Pappalardo, Andrea; Prezzavento, Orazio; Vittorio, F; Ronsisvalle, Giuseppe
4-Nitro-2,1,3-benzoxadiazole derivatives as potential fluorescent sigma receptor probes
2015-01-01 Schininà, Barbara; Martorana, Andrea; Colabufo Nicola, Antonio; Contino, Marialessandra; Niso, Mauro; Perrone Maria, Grazia; DE GUIDI, Guido; Catalfo, Alfio; Rappazzo, Giancarlo; Zuccarello, Elisa; Prezzavento, Orazio; Amata, Emanuele; Rescifina, Antonio; Marrazzo, Agostino
A new sigma ligand, (+/-)-PPCC, antagonizes kappa opioid receptor-mediated antinociceptive effect
2008-01-01 Prezzavento, Orazio; Parenti, Carmela; Marrazzo, Agostino; Ronsisvalle, Simone; Vittorio, F; Aricò, G; Scoto, Giovanna Maria; Ronsisvalle, Giuseppe
A new Sigma-1 Receptor antagonist in Chronic Pain Treatment: (+)-2R/S-LP2 effects in inflammatory and neuropathic pain
2022-01-01 Spoto, Salvatore; Pasquinucci, Lorella Giuseppina; Turnaturi, Rita; Costanzo, Giuliana; Chiechio, Santina; Vicario, Nunzio; Parenti, Rosalba; Marrazzo, Agostino; Amata, Emanuele; Parenti, Carmela
A novel adamantane derivative attenuates retinal ischemia-reperfusion damage in the rat retina through sigma1 receptors
2006-01-01 Bucolo, Claudio; Marrazzo, Agostino; Ronsisvalle, Simone; Ronsisvalle, Giuseppe; Cuzzocrea, S; Mazzon, E; Caputi, A; Drago, Filippo
A pseudouridine isoxazolidinyl nucleoside analogue structural analysis: A morphological approach
2018-01-01 Floresta, Giuseppe; Pistara', Venerando; Christensen E., Kirsten; Amata, Emanuele; Marrazzo, Agostino; Gentile, Davide; Rescifina, Antonio; Punzo, Francesco
A structure-and ligand-based virtual screening of a database of “small” marine natural products for the identification of “blue” sigma-2 receptor ligands
2018-01-01 Floresta, Giuseppe; Amata, Emanuele; Barbaraci, Carla; Gentile, Davide; Turnaturi, Rita; Marrazzo, Agostino; Rescifina, Antonio
Adipocyte fatty acid binding protein 4 (FABP4) inhibitors. A comprehensive systematic review
2017-01-01 Floresta, Giuseppe; Pistarà, Venerando; Amata, Emanuele; Dichiara, Maria; Marrazzo, Agostino; Prezzavento, Orazio; Rescifina, Antonio
Analgesici oppioidi
file da validare2024-01-01 Marrazzo, Agostino; Mollica, Adriano; Pasquinucci, Lorella; Turnaturi, Rita
Anti-amnesic and neuroprotective actions of the sigma-1 receptor agonist (-)-MR22 in rats with selective cholinergic lesion and amyloid infusion
2011-01-01 Antonini, V; Marrazzo, Agostino; Kleiner, G; Coradazzi, M; Ronsisvalle, Simone; Prezzavento, Orazio; Ronsisvalle, Giuseppe; Leanza, G.
Anti-amnesic properties of (+/-)-PPCC, a novel sigma receptor ligand, on cognitive dysfunction induced by selective cholinergic lesion in rats
2009-01-01 Antonini, V; Prezzavento, Orazio; Coradazzi, M; Marrazzo, Agostino; Ronsisvalle, Simone; Arena, E; Leanza, G.
Antiangiogenic Effect of (±)-Haloperidol Metabolite II Valproate Ester [(±)-MRJF22] in Human Microvascular Retinal Endothelial Cells
2016-01-01 Olivieri, Melania; Amata, Emanuele; Vinciguerra, Shila; Fiorito, Jole; Giurdanella, Giovanni; Drago, Filippo; Caporarello, Nunzia; Prezzavento, Orazio; Arena, Emanuela; Salerno, Loredana; Rescifina, Antonio; Lupo, Gabriella; Anfuso, CARMELINA DANIELA; Marrazzo, Agostino
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
(+)-and (−)-Phenazocine enantiomers: evaluation of their dual opioid agonist/σ1 antagonist properties and antinociceptive effects | 1-gen-2017 | Prezzavento, Orazio; Arena, Emanuela; Sánchez-Fernández, Cristine; Turnaturi, Rita; Parenti, Carmela; Marrazzo, Agostino; Catalano, Roberto; Amata, Emanuele; Pasquinucci, Lorella; Cobos J., Enrique | |
(+)-cis-N-ethyleneamino-N-normetazocine derivatives. Novel and selective sigma ligands with antagonist properties | 1-gen-1998 | Ronsisvalle, G; Marrazzo, Agostino; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Vittorio, F; Pittala', Valeria; Pappalardo, Ms; Cacciaguerra, S; Spampinato, S. | |
(+)-Methyl (1R,2S)-2-{[4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl]methyl}-1-phenylcyclopropanecarboxylate [(+)-MR200] Derivatives as Potent and Selective Sigma Receptor Ligands: Stereochemistry and Pharmacological Properties | 1-gen-2018 | Amata, Emanuele; Rescifina, Antonio; Prezzavento, Orazio; Arena, Emanuela; Dichiara, Maria; Pittalà, Valeria; Montilla-Garcia, A ngeles; Punzo, Francesco; Merino, Pedro; Cobos J., Enrique; Marrazzo, Agostino | |
(+)-MR200 derivatives as potential new selective sigma ligands | 1-gen-2007 | Marrazzo, Agostino; Ronsisvalle, Simone; Prezzavento, O; Vittorio, F; Ronsisvalle, Giuseppe | file da validare |
(+)-MR200 derivatives as potenzial new selective ligands | 1-gen-2007 | Marrazzo, Agostino; Ronsisvalle, Simone; Prezzavento, Orazio; Franco, Vittorio; Giuseppe, Ronsisvalle | file da validare |
(+)-Mr200 derivatives: modifications on the amino moiety. In vitro and in vivo pharmacological evaluation | 1-gen-2008 | Marrazzo, Agostino; Cobos, E. J.; Iemolo, A; Gonzàlez, L. G.; Prezzavento, Orazio; Parenti, Carmela; Aricò, G; Sanfilippo, M; Ronsisvalle, Simone; Scoto, Giovanna Maria | file da validare |
(+)-Pentazocine attenuates SH-SY5Y cell death, oxidative stress and microglial migration induced by conditioned medium from activated microglia | 1-gen-2017 | Heiss, K; Raffaele, M; Vanella, L; Murabito, P; Prezzavento, O; Marrazzo, Agostino; Aricò, G; CASTRUCCIO CASTRACANI, Carlo; Barbagallo, IGNAZIO ALBERTO; Zappala', Agata; Avola, Roberto; LI VOLTI, Giovanni | |
(+)-Pentazocine reduces oxidative stress and apoptosis in microglia following hypoxia/reoxygenation injury | 1-gen-2016 | Heiss, K; Vanella, Luca; Murabito, P; Prezzavento, Orazio; Marrazzo, Agostino; CASTRUCCIO CASTRACANI, Carlo; Barbagallo, IGNAZIO ALBERTO; Zappala', Agata; Arena, E; Astuto, Marinella; Giarratano, A; LI VOLTI, Giovanni | |
1-Phenyl-3azabicyclo[3.1.0]hexane derivatives as new ligands for sigma receptors | 1-gen-2004 | Marrazzo, Agostino; Pappalardo, Andrea; Prezzavento, Orazio; Vittorio, F; Ronsisvalle, Giuseppe | file da validare |
4-Nitro-2,1,3-benzoxadiazole derivatives as potential fluorescent sigma receptor probes | 1-gen-2015 | Schininà, Barbara; Martorana, Andrea; Colabufo Nicola, Antonio; Contino, Marialessandra; Niso, Mauro; Perrone Maria, Grazia; DE GUIDI, Guido; Catalfo, Alfio; Rappazzo, Giancarlo; Zuccarello, Elisa; Prezzavento, Orazio; Amata, Emanuele; Rescifina, Antonio; Marrazzo, Agostino | |
A new sigma ligand, (+/-)-PPCC, antagonizes kappa opioid receptor-mediated antinociceptive effect | 1-gen-2008 | Prezzavento, Orazio; Parenti, Carmela; Marrazzo, Agostino; Ronsisvalle, Simone; Vittorio, F; Aricò, G; Scoto, Giovanna Maria; Ronsisvalle, Giuseppe | |
A new Sigma-1 Receptor antagonist in Chronic Pain Treatment: (+)-2R/S-LP2 effects in inflammatory and neuropathic pain | 1-gen-2022 | Spoto, Salvatore; Pasquinucci, Lorella Giuseppina; Turnaturi, Rita; Costanzo, Giuliana; Chiechio, Santina; Vicario, Nunzio; Parenti, Rosalba; Marrazzo, Agostino; Amata, Emanuele; Parenti, Carmela | |
A novel adamantane derivative attenuates retinal ischemia-reperfusion damage in the rat retina through sigma1 receptors | 1-gen-2006 | Bucolo, Claudio; Marrazzo, Agostino; Ronsisvalle, Simone; Ronsisvalle, Giuseppe; Cuzzocrea, S; Mazzon, E; Caputi, A; Drago, Filippo | |
A pseudouridine isoxazolidinyl nucleoside analogue structural analysis: A morphological approach | 1-gen-2018 | Floresta, Giuseppe; Pistara', Venerando; Christensen E., Kirsten; Amata, Emanuele; Marrazzo, Agostino; Gentile, Davide; Rescifina, Antonio; Punzo, Francesco | |
A structure-and ligand-based virtual screening of a database of “small” marine natural products for the identification of “blue” sigma-2 receptor ligands | 1-gen-2018 | Floresta, Giuseppe; Amata, Emanuele; Barbaraci, Carla; Gentile, Davide; Turnaturi, Rita; Marrazzo, Agostino; Rescifina, Antonio | |
Adipocyte fatty acid binding protein 4 (FABP4) inhibitors. A comprehensive systematic review | 1-gen-2017 | Floresta, Giuseppe; Pistarà, Venerando; Amata, Emanuele; Dichiara, Maria; Marrazzo, Agostino; Prezzavento, Orazio; Rescifina, Antonio | |
Analgesici oppioidi | 1-gen-2024 | Marrazzo, Agostino; Mollica, Adriano; Pasquinucci, Lorella; Turnaturi, Rita | file da validare |
Anti-amnesic and neuroprotective actions of the sigma-1 receptor agonist (-)-MR22 in rats with selective cholinergic lesion and amyloid infusion | 1-gen-2011 | Antonini, V; Marrazzo, Agostino; Kleiner, G; Coradazzi, M; Ronsisvalle, Simone; Prezzavento, Orazio; Ronsisvalle, Giuseppe; Leanza, G. | |
Anti-amnesic properties of (+/-)-PPCC, a novel sigma receptor ligand, on cognitive dysfunction induced by selective cholinergic lesion in rats | 1-gen-2009 | Antonini, V; Prezzavento, Orazio; Coradazzi, M; Marrazzo, Agostino; Ronsisvalle, Simone; Arena, E; Leanza, G. | |
Antiangiogenic Effect of (±)-Haloperidol Metabolite II Valproate Ester [(±)-MRJF22] in Human Microvascular Retinal Endothelial Cells | 1-gen-2016 | Olivieri, Melania; Amata, Emanuele; Vinciguerra, Shila; Fiorito, Jole; Giurdanella, Giovanni; Drago, Filippo; Caporarello, Nunzia; Prezzavento, Orazio; Arena, Emanuela; Salerno, Loredana; Rescifina, Antonio; Lupo, Gabriella; Anfuso, CARMELINA DANIELA; Marrazzo, Agostino |