GENTILE, DAVIDE
GENTILE, DAVIDE
SCIENZE DEL FARMACO E DELLA SALUTE (DSFS) (Department of Drug and Health Sciences)
A pseudouridine isoxazolidinyl nucleoside analogue structural analysis: A morphological approach
2018-01-01 Floresta, Giuseppe; Pistara', Venerando; Christensen E., Kirsten; Amata, Emanuele; Marrazzo, Agostino; Gentile, Davide; Rescifina, Antonio; Punzo, Francesco
A structure-and ligand-based virtual screening of a database of “small” marine natural products for the identification of “blue” sigma-2 receptor ligands
2018-01-01 Floresta, Giuseppe; Amata, Emanuele; Barbaraci, Carla; Gentile, Davide; Turnaturi, Rita; Marrazzo, Agostino; Rescifina, Antonio
An integrated pharmacophore/docking/3D-QSAR approach to screening a large library of products in search of future botulinum neurotoxin a inhibitors
file da validare2020-01-01 Gentile, D.; Floresta, G.; Patamia, V.; Chiaramonte, R.; Mauro, G. L.; Rescifina, A.; Vecchio, M.
Artificial Intelligence Technologies for COVID-19 De Novo Drug Design
file da validare2022-01-01 Floresta, G.; Zagni, C.; Gentile, D.; Patamia, V.; Rescifina, A.
Computational tools in the discovery of FABP4 ligands: A statistical and molecular modeling approach
2019-01-01 Floresta, G.; Gentile, D.; Perrini, G.; Patamia, Vincenzo; Rescifina, A.
Covalently immobilized catalase on functionalized graphene: Effect on the activity, immobilization efficiency, and tetramer stability
2018-01-01 Barreca, D.; Neri, G.; Scala, A.; Fazio, E.; Gentile, D.; Rescifina, A.; Piperno, A.
Cucurbit[7]uril as a catalytic nanoreactor for one-pot synthesis of isoxazolidines in water
2020-01-01 Gentile, Davide; Floresta, Giuseppe; Patamia, Vincenzo; Nicosia, Angelo; Mineo, Placido; Rescifina, Antonio
Design, synthesis, and pharmacological evaluation of NO donor-sigma receptors hybrids for the treatment of cancer
2018-01-01 Dichiara, Maria; Barbaraci, Carla; Gentile, Davide; Intagliata, Sebastiano; Pittalà, Valeria; Arena, Emanuelea; Fraix, Aurore; Farina, Giuseppe; Prezzavento, Orazio; Amata, Emanuele; Marrazzo, Agostino.
Fourfold filtered statistical/computational approach for the identification of imidazole compounds as HO-1 inhibitors from natural products
2019-01-01 Floresta, Giuseppe; Amata, Emanuele; Gentile, Davide; Romeo, Giuseppe; Marrazzo, Agostino; Pittalà, Valeria; Salerno, Loredana; Rescifina, Antonio
La modellistica molecolare applicata ai recettori Sigma-1 e Sigma-2: un excursus
2019-01-01 Floresta, Giuseppe; Gentile, Davide; Dichiara, Maria; Amata, Emanuele; Rescifina, Antonio; Marrazzo, Agostino
Morphing of ibogaine: A successful attempt into the search for sigma-2 receptor ligands
2019-01-01 Floresta, Giuseppe; Dichiara, Maria; Gentile, Davide; Prezzavento, Orazio; Marrazzo, Agostino; Rescifina, Antonio; Amata, Emanuele
Nanosponges based on self-assembled starfish-shaped cucurbit[6]urils functionalized with imidazolium arms
file da validare2021-01-01 Patamia, Vincenzo; Gentile, Davide; Fiorenza, Roberto; Muccilli, Vera; Mineo, Placido G.; Scirè, Salvatore; Rescifina, Antonio
Natural Substances in the Fight of SARS-CoV-2: A Critical Evaluation Resulting from the Cross-Fertilization of Molecular Modeling Data with the Pharmacological Aspects
file da validare2021-01-01 Gentile, Davide; Patamia, Vincenzo; Fuochi, Virginia; Furneri, Pio M; Rescifina, Antonio
New anti sars-cov-2 targets for quinoline derivatives chloroquine and hydroxychloroquine
2020-01-01 Gentile, D.; Fuochi, V.; Rescifina, A.; Furneri, P. M.
Nitric Oxide Photo-Donor Hybrids of Ciprofloxacin and Norfloxacin: A Shift in Activity from Antimicrobial to Anticancer Agents
file da validare2021-01-01 Fallica Antonino, Nicolò; Barbaraci, Carla; Amata, Emanuele; Pasquinucci, Lorella; Turnaturi, Rita; Dichiara, Maria; Intagliata, Sebastiano; Gariboldi Marzia, Bruna; Marras, Emanuela; Orlandi Viviana, Teresa; Ferroni, Claudia; Martini, Cecilia; Rescifina, Antonio; Gentile, Davide; Varchi, Greta; Marrazzo, Agostino
Progress in the development of selective heme oxygenase-1 inhibitors and their potential therapeutic application
2019-01-01 Salerno, Loredana; Floresta, Giuseppe; Ciaffaglione, Valeria; Gentile, Davide; Margani, Fatima; Turnaturi, Rita; Rescifina, Antonio; Pittalà, Valeria
Putative inhibitors of SARS-COV-2 main protease from a library of marine natural products: A virtual screening and molecular modeling study
2020-01-01 Gentile, D.; Patamia, V.; Scala, A.; Sciortino, M. T.; Piperno, A.; Rescifina, A.
Repurposing of FDA-Approved Drugs for Treating Iatrogenic Botulism: A Paired 3D-QSAR/Docking Approach†
2020-01-01 Floresta, G.; Patamia, V.; Gentile, D.; Molteni, F.; Santamato, A.; Rescifina, A.; Vecchio, M.
Sigma Receptor Ligands Carrying a Nitric Oxide Donor Nitrate Moiety: Synthesis, In Silico, and Biological Evaluation
2020-01-01 Amata, Emanuele; Dichiara, Maria; Gentile, Davide; Marrazzo, Agostino; Turnaturi, Rita; Arena, Emanuela; La Mantia, Alfonsina; Tomasello, Barbara; Acquaviva, Rosaria; DI GIACOMO, Claudia; Rescifina, Antonio; Prezzavento, Orazio
Structural and Molecular Insight into Piperazine and Piperidine Derivatives as Histamine H3 and Sigma-1 Receptor Antagonists with Promising Antinociceptive Properties
2022-01-01 Szczepańska, Katarzyna; Podlewska, Sabina; Dichiara, Maria; Gentile, Davide; Patamia, Vincenzo; Rosier, Niklas; Mönnich, Denise; Ruiz Cantero M., Carmen; Karcz, Tadeusz; Łażewska, Dorota; Siwek, Agata; Pockes, Steffen; Cobos J., Enrique; Marrazzo, Agostino; Stark, Holger; Rescifina, Antonio; Bojarski J., Andrzej; Amata, Emanuele; Kieć-Kononowicz, Katarkyna
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
A pseudouridine isoxazolidinyl nucleoside analogue structural analysis: A morphological approach | 1-gen-2018 | Floresta, Giuseppe; Pistara', Venerando; Christensen E., Kirsten; Amata, Emanuele; Marrazzo, Agostino; Gentile, Davide; Rescifina, Antonio; Punzo, Francesco | |
A structure-and ligand-based virtual screening of a database of “small” marine natural products for the identification of “blue” sigma-2 receptor ligands | 1-gen-2018 | Floresta, Giuseppe; Amata, Emanuele; Barbaraci, Carla; Gentile, Davide; Turnaturi, Rita; Marrazzo, Agostino; Rescifina, Antonio | |
An integrated pharmacophore/docking/3D-QSAR approach to screening a large library of products in search of future botulinum neurotoxin a inhibitors | 1-gen-2020 | Gentile, D.; Floresta, G.; Patamia, V.; Chiaramonte, R.; Mauro, G. L.; Rescifina, A.; Vecchio, M. | file da validare |
Artificial Intelligence Technologies for COVID-19 De Novo Drug Design | 1-gen-2022 | Floresta, G.; Zagni, C.; Gentile, D.; Patamia, V.; Rescifina, A. | file da validare |
Computational tools in the discovery of FABP4 ligands: A statistical and molecular modeling approach | 1-gen-2019 | Floresta, G.; Gentile, D.; Perrini, G.; Patamia, Vincenzo; Rescifina, A. | |
Covalently immobilized catalase on functionalized graphene: Effect on the activity, immobilization efficiency, and tetramer stability | 1-gen-2018 | Barreca, D.; Neri, G.; Scala, A.; Fazio, E.; Gentile, D.; Rescifina, A.; Piperno, A. | |
Cucurbit[7]uril as a catalytic nanoreactor for one-pot synthesis of isoxazolidines in water | 1-gen-2020 | Gentile, Davide; Floresta, Giuseppe; Patamia, Vincenzo; Nicosia, Angelo; Mineo, Placido; Rescifina, Antonio | |
Design, synthesis, and pharmacological evaluation of NO donor-sigma receptors hybrids for the treatment of cancer | 1-gen-2018 | Dichiara, Maria; Barbaraci, Carla; Gentile, Davide; Intagliata, Sebastiano; Pittalà, Valeria; Arena, Emanuelea; Fraix, Aurore; Farina, Giuseppe; Prezzavento, Orazio; Amata, Emanuele; Marrazzo, Agostino. | |
Fourfold filtered statistical/computational approach for the identification of imidazole compounds as HO-1 inhibitors from natural products | 1-gen-2019 | Floresta, Giuseppe; Amata, Emanuele; Gentile, Davide; Romeo, Giuseppe; Marrazzo, Agostino; Pittalà, Valeria; Salerno, Loredana; Rescifina, Antonio | |
La modellistica molecolare applicata ai recettori Sigma-1 e Sigma-2: un excursus | 1-gen-2019 | Floresta, Giuseppe; Gentile, Davide; Dichiara, Maria; Amata, Emanuele; Rescifina, Antonio; Marrazzo, Agostino | |
Morphing of ibogaine: A successful attempt into the search for sigma-2 receptor ligands | 1-gen-2019 | Floresta, Giuseppe; Dichiara, Maria; Gentile, Davide; Prezzavento, Orazio; Marrazzo, Agostino; Rescifina, Antonio; Amata, Emanuele | |
Nanosponges based on self-assembled starfish-shaped cucurbit[6]urils functionalized with imidazolium arms | 1-gen-2021 | Patamia, Vincenzo; Gentile, Davide; Fiorenza, Roberto; Muccilli, Vera; Mineo, Placido G.; Scirè, Salvatore; Rescifina, Antonio | file da validare |
Natural Substances in the Fight of SARS-CoV-2: A Critical Evaluation Resulting from the Cross-Fertilization of Molecular Modeling Data with the Pharmacological Aspects | 1-gen-2021 | Gentile, Davide; Patamia, Vincenzo; Fuochi, Virginia; Furneri, Pio M; Rescifina, Antonio | file da validare |
New anti sars-cov-2 targets for quinoline derivatives chloroquine and hydroxychloroquine | 1-gen-2020 | Gentile, D.; Fuochi, V.; Rescifina, A.; Furneri, P. M. | |
Nitric Oxide Photo-Donor Hybrids of Ciprofloxacin and Norfloxacin: A Shift in Activity from Antimicrobial to Anticancer Agents | 1-gen-2021 | Fallica Antonino, Nicolò; Barbaraci, Carla; Amata, Emanuele; Pasquinucci, Lorella; Turnaturi, Rita; Dichiara, Maria; Intagliata, Sebastiano; Gariboldi Marzia, Bruna; Marras, Emanuela; Orlandi Viviana, Teresa; Ferroni, Claudia; Martini, Cecilia; Rescifina, Antonio; Gentile, Davide; Varchi, Greta; Marrazzo, Agostino | file da validare |
Progress in the development of selective heme oxygenase-1 inhibitors and their potential therapeutic application | 1-gen-2019 | Salerno, Loredana; Floresta, Giuseppe; Ciaffaglione, Valeria; Gentile, Davide; Margani, Fatima; Turnaturi, Rita; Rescifina, Antonio; Pittalà, Valeria | |
Putative inhibitors of SARS-COV-2 main protease from a library of marine natural products: A virtual screening and molecular modeling study | 1-gen-2020 | Gentile, D.; Patamia, V.; Scala, A.; Sciortino, M. T.; Piperno, A.; Rescifina, A. | |
Repurposing of FDA-Approved Drugs for Treating Iatrogenic Botulism: A Paired 3D-QSAR/Docking Approach† | 1-gen-2020 | Floresta, G.; Patamia, V.; Gentile, D.; Molteni, F.; Santamato, A.; Rescifina, A.; Vecchio, M. | |
Sigma Receptor Ligands Carrying a Nitric Oxide Donor Nitrate Moiety: Synthesis, In Silico, and Biological Evaluation | 1-gen-2020 | Amata, Emanuele; Dichiara, Maria; Gentile, Davide; Marrazzo, Agostino; Turnaturi, Rita; Arena, Emanuela; La Mantia, Alfonsina; Tomasello, Barbara; Acquaviva, Rosaria; DI GIACOMO, Claudia; Rescifina, Antonio; Prezzavento, Orazio | |
Structural and Molecular Insight into Piperazine and Piperidine Derivatives as Histamine H3 and Sigma-1 Receptor Antagonists with Promising Antinociceptive Properties | 1-gen-2022 | Szczepańska, Katarzyna; Podlewska, Sabina; Dichiara, Maria; Gentile, Davide; Patamia, Vincenzo; Rosier, Niklas; Mönnich, Denise; Ruiz Cantero M., Carmen; Karcz, Tadeusz; Łażewska, Dorota; Siwek, Agata; Pockes, Steffen; Cobos J., Enrique; Marrazzo, Agostino; Stark, Holger; Rescifina, Antonio; Bojarski J., Andrzej; Amata, Emanuele; Kieć-Kononowicz, Katarkyna |