COSENTINO, GIUSEPPE
COSENTINO, GIUSEPPE
SCIENZE BIOMEDICHE E BIOTECNOLOGICHE
Design, Synthesis, and Cytotoxic Assessment of New Haloperidol Analogues as Potential Anticancer Compounds Targeting Sigma Receptors
2024-01-01 Zampieri, Daniele; Romano, Maurizio; Fortuna, Sara; Amata, Emanuele; Dichiara, Maria; Cosentino, Giuseppe; Marrazzo, Agostino; Grazia Mamolo, Maria
DESIGN, SYNTHESIS, MOLECULAR MODELING AND PHARMACOLOGICAL EVALUATION OF NOVEL DIAZABICYCLO[4.3.0]NONANE AND 2,7-DIAZASPIRO[3.5]NONANE AS SIGMA RECEPTORS LIGANDS
file da validare2023-01-01 Cosentino, G.; Dichiara, M.; Ambrosio, F. A.; Barbaraci, C.; González-Cano, R.; Costa, G.; Giordano, G.; Pasquinucci, L.; Marrazzo, A.; Cobos, E. J.; Alcaro, S.; Amata, E.
Designing drugs optimized for both blood-brain barrier permeation and intra-cerebral partition
file da validare2023-01-01 Dichiara, Maria; Cosentino, Giuseppe; Giordano, Giorgia; Pasquinucci, Lorella; Marrazzo, Agostino; Costanzo, Giuliana; Amata, Emanuele
Discovery and computational studies of piperidine/piperazine-based compounds endowed with sigma receptor affinity
2023-01-01 De Luca, L.; Lombardo, L.; Mirabile, S.; Marrazzo, A.; Dichiara, M.; Cosentino, G.; Amata, E.; Gitto, R.
Discovery of 3-(2-aminoethyl)-thiazolidine-2,4-diones as a novel chemotype of sigma-1 receptor ligands
2022-01-01 Elkholy, Nada; Abdelwaly, Ahmad; Mohamed, Karim; Amata, Emanuele; Lombino, Jessica; Cosentino, Giuseppe; Intagliata, Sebastiano; Helal A., Mohamed
Discovery of AD258 as a Sigma Receptor Ligand with Potent Antiallodynic Activity
2023-01-01 Dichiara, Maria; Ambrosio Francesca, Alessandra; Lee Sang, Min; Ruiz-Cantero M., Carmen; Lombino, Jessica; Coricello, Adriana; Costa, Giosuè; Shah, Dhara; Costanzo, Giuliana; Pasquinucci, Lorella Giuseppina; Son Kyung, No; Cosentino, Giuseppe; González-Cano, Rafael; Marrazzo, Agostino; Aakalu Vinay, Kumar; Cobos Enrique, J.; Alcaro, Stefano; Amata, Emanuele
Exploring Structural Requirements for Sigma-1 Receptor Linear Ligands: Experimental and Computational Approaches
2024-01-01 Lombardo, Lisa; Mirabile, Salvatore; Gitto, Rosaria; Cosentino, Giuseppe; Alcaro, Stefano; Dichiara, Maria; Marrazzo, Agostino; Amata, Emanuele; Ortuso, Francesco; De Luca, Laura
Investigation of Tau-Dependent Epigenetic Reprogramming in Alzheimer’s Disease
2024-01-01 Costanzo, G.; Coco, A.; Scarlatti, A.; Siano, G.; Cosentino, G.; Di Primio, C.; Amata, E.; Marrazzo, A.; Rescifina, A.; Pasquinucci, L.
Microscopic Evidence of the Behavior of pH-sensitive Food-grade Polymeric Delivery Systems
file da validare2023-01-01 Pignatello, Rosario; Carbone, Claudia; Rizzo, Salvatore; Cosentino, Giuseppe; Zingale, Elide; Bonaccorso, Angela; Petralia, Salvatore; Monforte, Francesca; Condorelli, Guglielmo G.
NOVEL N-NORMETAZOCINE DERIVATIVES WITH SIGMA-1 RECEPTOR ANTAGONIST PROFILE AS POTENTIAL ANALGESICS FOR INFLAMMATORY PAIN MANAGEMENT
file da validare2023-01-01 Costanzo, G.; Cosentino, G.; Patamia, V.; Turnaturi, R.; Parenti, C.; Rescifina, A.; Marrazzo, A.; Amata, E; Pasquinucci, L.
Synthesis and biological evaluation of novel σ1R ligands
2024-01-01 Costanzo, Giuliana; Cosentino, Giuseppe; Patamia, Vincenzo; Grasso, Margherita; Marrazzo, Agostino; Amata, Emanuele; Parenti, Carmela; Rescifina, Antonio; Pasquinucci, Lorella
SYNTHESIS, COMPUTATIONAL INSIGHTS, AND EVALUATION OF NOVEL SIGMA RECEPTORS LIGANDS
2023-01-01 Dichiara, M.; Ambrosio, F. A.; Barbaraci, C.; Shah, D.; Gonzàles-Cano, R.; Ruiz-Cantero, C.; Coricello, A.; Costa, G.; Lee, S. M.; Son, K. N.; Lombino, J.; Costanzo, G.; Cosentino, G.; Giordano, G.; Pasquinucci, L.; Marrazzo, A.; Aakalu, V. K.; Cobos, E. J.; Alcaro, S.; Amata, E.
Two‐Step Synthesis of Enantiomerically Pure Morphans from (R)‐Carvone
file da validare2024-01-01 Costanzo, Giuliana; Cosentino, Giuseppe; Pasquinucci, Lorella; Amata, Emanuele; Schepmann, Dirk; Wünsch, Bernhard
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Design, Synthesis, and Cytotoxic Assessment of New Haloperidol Analogues as Potential Anticancer Compounds Targeting Sigma Receptors | 1-gen-2024 | Zampieri, Daniele; Romano, Maurizio; Fortuna, Sara; Amata, Emanuele; Dichiara, Maria; Cosentino, Giuseppe; Marrazzo, Agostino; Grazia Mamolo, Maria | |
| DESIGN, SYNTHESIS, MOLECULAR MODELING AND PHARMACOLOGICAL EVALUATION OF NOVEL DIAZABICYCLO[4.3.0]NONANE AND 2,7-DIAZASPIRO[3.5]NONANE AS SIGMA RECEPTORS LIGANDS | 1-gen-2023 | Cosentino, G.; Dichiara, M.; Ambrosio, F. A.; Barbaraci, C.; González-Cano, R.; Costa, G.; Giordano, G.; Pasquinucci, L.; Marrazzo, A.; Cobos, E. J.; Alcaro, S.; Amata, E. | file da validare |
| Designing drugs optimized for both blood-brain barrier permeation and intra-cerebral partition | 1-gen-2023 | Dichiara, Maria; Cosentino, Giuseppe; Giordano, Giorgia; Pasquinucci, Lorella; Marrazzo, Agostino; Costanzo, Giuliana; Amata, Emanuele | file da validare |
| Discovery and computational studies of piperidine/piperazine-based compounds endowed with sigma receptor affinity | 1-gen-2023 | De Luca, L.; Lombardo, L.; Mirabile, S.; Marrazzo, A.; Dichiara, M.; Cosentino, G.; Amata, E.; Gitto, R. | |
| Discovery of 3-(2-aminoethyl)-thiazolidine-2,4-diones as a novel chemotype of sigma-1 receptor ligands | 1-gen-2022 | Elkholy, Nada; Abdelwaly, Ahmad; Mohamed, Karim; Amata, Emanuele; Lombino, Jessica; Cosentino, Giuseppe; Intagliata, Sebastiano; Helal A., Mohamed | |
| Discovery of AD258 as a Sigma Receptor Ligand with Potent Antiallodynic Activity | 1-gen-2023 | Dichiara, Maria; Ambrosio Francesca, Alessandra; Lee Sang, Min; Ruiz-Cantero M., Carmen; Lombino, Jessica; Coricello, Adriana; Costa, Giosuè; Shah, Dhara; Costanzo, Giuliana; Pasquinucci, Lorella Giuseppina; Son Kyung, No; Cosentino, Giuseppe; González-Cano, Rafael; Marrazzo, Agostino; Aakalu Vinay, Kumar; Cobos Enrique, J.; Alcaro, Stefano; Amata, Emanuele | |
| Exploring Structural Requirements for Sigma-1 Receptor Linear Ligands: Experimental and Computational Approaches | 1-gen-2024 | Lombardo, Lisa; Mirabile, Salvatore; Gitto, Rosaria; Cosentino, Giuseppe; Alcaro, Stefano; Dichiara, Maria; Marrazzo, Agostino; Amata, Emanuele; Ortuso, Francesco; De Luca, Laura | |
| Investigation of Tau-Dependent Epigenetic Reprogramming in Alzheimer’s Disease | 1-gen-2024 | Costanzo, G.; Coco, A.; Scarlatti, A.; Siano, G.; Cosentino, G.; Di Primio, C.; Amata, E.; Marrazzo, A.; Rescifina, A.; Pasquinucci, L. | |
| Microscopic Evidence of the Behavior of pH-sensitive Food-grade Polymeric Delivery Systems | 1-gen-2023 | Pignatello, Rosario; Carbone, Claudia; Rizzo, Salvatore; Cosentino, Giuseppe; Zingale, Elide; Bonaccorso, Angela; Petralia, Salvatore; Monforte, Francesca; Condorelli, Guglielmo G. | file da validare |
| NOVEL N-NORMETAZOCINE DERIVATIVES WITH SIGMA-1 RECEPTOR ANTAGONIST PROFILE AS POTENTIAL ANALGESICS FOR INFLAMMATORY PAIN MANAGEMENT | 1-gen-2023 | Costanzo, G.; Cosentino, G.; Patamia, V.; Turnaturi, R.; Parenti, C.; Rescifina, A.; Marrazzo, A.; Amata, E; Pasquinucci, L. | file da validare |
| Synthesis and biological evaluation of novel σ1R ligands | 1-gen-2024 | Costanzo, Giuliana; Cosentino, Giuseppe; Patamia, Vincenzo; Grasso, Margherita; Marrazzo, Agostino; Amata, Emanuele; Parenti, Carmela; Rescifina, Antonio; Pasquinucci, Lorella | |
| SYNTHESIS, COMPUTATIONAL INSIGHTS, AND EVALUATION OF NOVEL SIGMA RECEPTORS LIGANDS | 1-gen-2023 | Dichiara, M.; Ambrosio, F. A.; Barbaraci, C.; Shah, D.; Gonzàles-Cano, R.; Ruiz-Cantero, C.; Coricello, A.; Costa, G.; Lee, S. M.; Son, K. N.; Lombino, J.; Costanzo, G.; Cosentino, G.; Giordano, G.; Pasquinucci, L.; Marrazzo, A.; Aakalu, V. K.; Cobos, E. J.; Alcaro, S.; Amata, E. | |
| Two‐Step Synthesis of Enantiomerically Pure Morphans from (R)‐Carvone | 1-gen-2024 | Costanzo, Giuliana; Cosentino, Giuseppe; Pasquinucci, Lorella; Amata, Emanuele; Schepmann, Dirk; Wünsch, Bernhard | file da validare |