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Intramolecular oxidative palladium-​catalyzed diamination reactions of alkenyl sulfamates: an efficient synthesis of [1,​2,​5]​thiadiazolo-​fused piperazinones 1-gen-2016 Chiacchio, U; Broggini, G; Romeo, R; Gazzola, S; Giofre, S; Gabriele, B; Mancuso, R; Floresta, G; Zagni, C; Chiacchio, M
Synthesis and evaluation of haloperidol metabolite II prodrugs as anticancer agents 1-gen-2017 Dichiara, Maria; Amata, Emanuele; Rescifina, Antonio; Prezzavento, Orazio; Floresta, Giuseppe; Parenti, Carmela; Pittalà, Valeria; Marrazzo, Agostino
Hyphenated 3D-QSAR statistical model-scaffold hopping analysis for the identification of potentially potent and selective sigma-2 receptor ligands 1-gen-2017 Floresta, Giuseppe; Rescifina, Antonio; Marrazzo, Agostino; Dichiara, Maria; Pistarà, Venerando; Pittalà, Valeria; Prezzavento, Orazio; Amata, Emanuele
The Search for Potent, Small-Molecule HDACIs in Cancer Treatment: A Decade After Vorinostat 1-gen-2017 Zagni, Chiara; Floresta, Giuseppe; Monciino, Giulia; Rescifina, Antonio
Sigma-2 receptor ligands QSAR model dataset 1-gen-2017 Rescifina, Antonio; Floresta, Giuseppe; Marrazzo, Agostino; Parenti, Carmela; Prezzavento, Orazio; Nastasi, Giovanni; Dichiara, Maria; Amata, Emanuele
Adipocyte fatty acid binding protein 4 (FABP4) inhibitors. A comprehensive systematic review 1-gen-2017 Floresta, Giuseppe; Pistarà, Venerando; Amata, Emanuele; Dichiara, Maria; Marrazzo, Agostino; Prezzavento, Orazio; Rescifina, Antonio
γ-Cyclodextrin as a Catalyst for the Synthesis of 2-Methyl-3,5-diarylisoxazolidines in Water 1-gen-2017 Floresta, Giuseppe; Talotta, Carmen; Gaeta, Carmine; De Rosa, Margherita; Chiacchio, Ugo; Neri, Placido; Rescifina, Antonio
Development of a Sigma-2 Receptor affinity filter through a Monte Carlo based QSAR analysis 1-gen-2017 Rescifina, Antonio; Floresta, Giuseppe; Marrazzo, Agostino; Parenti, Carmela; Prezzavento, Orazio; Nastasi, Giovanni; Dichiara, Maria; Amata, Emanuele
Potholing of the hydrophobic heme oxygenase-1 western region for the search of potent and selective imidazole-based inhibitors 1-gen-2018 Salerno, Loredana; Amata, Emanuele; Romeo, Giuseppe; Marrazzo, Agostino; Floresta, Giuseppe; Modica Maria, N.; Greish Khaled, F.; Sorrenti, Valeria; Rescifina, Antonio; Pittalà, Valeria
Rosmarinic acid amides: synthesis, α-glucosidase inhibition and enzyme binding mode 1-gen-2018 Cardullo, N.; Catinella, G.; Floresta, G.; Rosselli, S.; Rescifina, A.; Bruno, M.; Tringali, C. file da validare
Potholing of the hydrophobic heme oxygenase-1 western region for the search of potent and selective imidazole-based inhibitors 1-gen-2018 Salerno, Loredana; Amata, Emanuele; Romeo, Giuseppe; Marrazzo, Agostino; Prezzavento, Orazio; Floresta, Giuseppe; Sorrenti, Valeria; Barbagallo, Ignazio; Rescifina, Antonio; Pittalà, Valeria
DNA intercalators based on (1,10-phenanthrolin-2-yl)isoxazolidin-5-yl core with better growth inhibition and selectivity than cisplatin upon head and neck squamous cells carcinoma 1-gen-2018 Varrica G., Maria; Zagni, Chiara; Mineo, Placido; Floresta, Giuseppe; Monciino, Giulia; Pistara, Venerando; Abbadessa, Antonio; Nicosia, Angelo; Castilho M., Rogerio; Amata, Emanuele; Rescifina, Antonio
The hexameric resorcinarene capsule as an artificial enzyme: Ruling the regio and stereochemistry of a 1,3-dipolar cycloaddition between nitrones and unsaturated aldehydes 1-gen-2018 La Manna, Pellegrino; De Rosa, Margherita; Talotta, Carmen; Gaeta, Carmine; Soriente, Annunziata; Floresta, Giuseppe; Rescifina, Antonio; Neri, Placido
Identification of Potentially Potent Heme Oxygenase 1 Inhibitors through 3D-QSAR Coupled to Scaffold-Hopping Analysis 1-gen-2018 Floresta, Giuseppe; Amata, Emanuele; Dichiara, Maria; Marrazzo, Agostino; Salerno, Loredana; Romeo, Giuseppe; Prezzavento, Orazio; Pittalà, Valeria; Rescifina, Antonio
A structure-and ligand-based virtual screening of a database of “small” marine natural products for the identification of “blue” sigma-2 receptor ligands 1-gen-2018 Floresta, Giuseppe; Amata, Emanuele; Barbaraci, Carla; Gentile, Davide; Turnaturi, Rita; Marrazzo, Agostino; Rescifina, Antonio
Targeting heme Oxygenase-1 with hybrid compounds to overcome Imatinib resistance in chronic myeloid leukemia cell lines 1-gen-2018 Sorrenti, Valeria; Pittalà, Valeria; Romeo, Giuseppe; Amata, Emanuele; Dichiara, Maria; Marrazzo, Agostino; Turnaturi, Rita; Prezzavento, Orazio; Barbagallo, Ignazio; Vanella, Luca; Rescifina, Antonio; Floresta, Giuseppe; Tibullo, Daniele; DI RAIMONDO, Francesco; Intagliata, Sebastiano; Salerno, Loredana
Targeting the hydrophobic heme oxygenase-1 western region for the identification of novel and selective azole-based inhibitors. 1-gen-2018 Dichiara, M; Modica, Mn; Leonardi, C; Margani, F; Ciaffaglione, V; Fallica, An; Floresta, G; Gentile, D; Cosenza, J; Pittalà, V. file da validare
Discovery of high-affinity cannabinoid receptors ligands through a 3D-QSAR ushered by scaffold-hopping analysis 1-gen-2018 Floresta, G.; Apirakkan, O.; Rescifina, A.; Abbate, V.
Novel structural insight into inhibitors of heme oxygenase-1 (ho-1) by new imidazole-based compounds: Biochemical and in vitro anticancer activity evaluation 1-gen-2018 Greish F., Khaled; Salerno, Loredana; Zahrani Reem, Al; Amata, Emanuele; Modica, Maria Nunziata; Romeo, Giuseppe; Marrazzo, Agostino; Prezzavento, Orazio; Sorrenti, Valeria; Rescifina, Antonio; Floresta, Giuseppe; Intagliata, Sebastiano; Pittalà, Valeria
Novel Sigma-1 receptor antagonists: From opioids to small molecules: What is new? 1-gen-2018 Arena, Emanuela; Dichiara, Maria; Floresta, Giuseppe; Parenti, Carmela; Marrazzo, Agostino; Pittalà, Valeria; Amata, Emanuele; Prezzavento, Orazio
Mostrati risultati da 1 a 20 di 121
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