FLORESTA, GIUSEPPE
FLORESTA, GIUSEPPE
SCIENZE DEL FARMACO E DELLA SALUTE (DSFS) (Department of Drug and Health Sciences)
1,2-Dibenzoylhydrazine as a Multi-Inhibitor Compound: A Morphological and Docking Study
file da validare2023-01-01 Patamia, Vincenzo; Floresta, Giuseppe; Zagni, Chiara; Pistara', Venerando; Punzo, Francesco; Rescifina, Antonio
3D-QSAR assisted identification of FABP4 inhibitors: An effective scaffold hopping analysis/QSAR evaluation
2019-01-01 Floresta, G.; Cilibrizzi, A.; Abbate, V.; Spampinato, A.; Zagni, C.; Rescifina, A.
[1]Benzothieno[3,2-d]pyrimidine derivatives as ligands for the serotonergic 5-HT7 receptor
2019-01-01 Romeo, Giuseppe; Salerno, Loredana; Pittalà, Valeria; Candido, Marialuisa; Intagliata, Sebastiano; Amata, Emanuele; Salmona, Mario; Cagnotto, Alfredo; Rescifina, Antonio; Floresta, Giuseppe; Modica, Maria Nunziata
A hexameric resorcinarene capsule as a hydrogen bonding catalyst in the conjugate addition of pyrroles and indoles to nitroalkenes
2019-01-01 Gambaro, S.; De Rosa, M.; Soriente, A.; Talotta, C.; Floresta, G.; Rescifina, A.; Gaeta, C.; Neri, P.
A pseudouridine isoxazolidinyl nucleoside analogue structural analysis: A morphological approach
2018-01-01 Floresta, Giuseppe; Pistara', Venerando; Christensen E., Kirsten; Amata, Emanuele; Marrazzo, Agostino; Gentile, Davide; Rescifina, Antonio; Punzo, Francesco
A Rare Natural Benzo[k,l]xanthene as a Turn-Off Fluorescent Sensor for Cu2+ Ion
file da validare2020-01-01 Floresta, Giuseppe; Cardullo, Nunzio; Spatafora, Carmela; Rescifina, Antonio; Tringali, Corrado
A structure-and ligand-based virtual screening of a database of “small” marine natural products for the identification of “blue” sigma-2 receptor ligands
2018-01-01 Floresta, Giuseppe; Amata, Emanuele; Barbaraci, Carla; Gentile, Davide; Turnaturi, Rita; Marrazzo, Agostino; Rescifina, Antonio
Adipocyte fatty acid binding protein 4 (FABP4) inhibitors. A comprehensive systematic review
2017-01-01 Floresta, Giuseppe; Pistarà, Venerando; Amata, Emanuele; Dichiara, Maria; Marrazzo, Agostino; Prezzavento, Orazio; Rescifina, Antonio
Adipocyte fatty acid binding protein 4 (FABP4) inhibitors. An update from 2017 to early 2022
file da validare2022-01-01 Floresta, G.; Patamia, V.; Zagni, C.; Rescifina, A.
Ammidi dell’acido rosmarinico come potenziali agenti antidiabetici
2019-01-01 Muccilli, V; Cardullo, N; Catinella, G; Floresta, G; Rosselli, S; Rescifina, A; Bruno, M; Tringali., C
An integrated pharmacophore/docking/3D-QSAR approach to screening a large library of products in search of future botulinum neurotoxin a inhibitors
2020-01-01 Gentile, D.; Floresta, G.; Patamia, V.; Chiaramonte, R.; Mauro, G. L.; Rescifina, A.; Vecchio, M.
An Overview of PDE4 Inhibitors in Clinical Trials: 2010 to Early 2022
2022-01-01 Crocetti, L.; Floresta, G.; Cilibrizzi, A.; Giovannoni, M. P.
Artificial Intelligence Technologies for COVID-19 De Novo Drug Design
file da validare2022-01-01 Floresta, G.; Zagni, C.; Gentile, D.; Patamia, V.; Rescifina, A.
Carbamoyl-Decorated Cyclodextrins for Carbon Dioxide Adsorption
file da validare2023-01-01 Patamia, Vincenzo; Tomarchio, Rosario; Fiorenza, Roberto; Zagni, Chiara; Scire', Salvatore; Floresta, Giuseppe; Rescifina, Antonio
Chromatograpic resolution of phenylethanolic-azole racemic compounds highlighted stereoselective inhibition of heme oxygenase-1 by (R)-enantiomers
2020-01-01 Floresta, G.; Carotti, A.; Ianni, F.; Sorrenti, V.; Intagliata, S.; Rescifina, A.; Salerno, L.; Di Michele, A.; Sardella, R.; Pittala, V.
Computational tools in the discovery of FABP4 ligands: A statistical and molecular modeling approach
2019-01-01 Floresta, G.; Gentile, D.; Perrini, G.; Patamia, Vincenzo; Rescifina, A.
Computer-Assisted Design of Peptide-Based Radiotracers
file da validare2023-01-01 Patamia, Vincenzo; Zagni, Chiara; Brullo, Ilaria; Saccullo, Erika; Coco, Alessandro; Floresta, Giuseppe; Rescifina, Antonio
Cucurbit[7]uril as a catalytic nanoreactor for one-pot synthesis of isoxazolidines in water
2020-01-01 Gentile, Davide; Floresta, Giuseppe; Patamia, Vincenzo; Nicosia, Angelo; Mineo, Placido; Rescifina, Antonio
Design and synthesis of novel compounds as fatty acids binding protein inhibitors and as gallium-68 chelators for positron emission tomography
2018-11-09 Floresta, Giuseppe
Development of a Sigma-2 Receptor affinity filter through a Monte Carlo based QSAR analysis
2017-01-01 Rescifina, Antonio; Floresta, Giuseppe; Marrazzo, Agostino; Parenti, Carmela; Prezzavento, Orazio; Nastasi, Giovanni; Dichiara, Maria; Amata, Emanuele
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
1,2-Dibenzoylhydrazine as a Multi-Inhibitor Compound: A Morphological and Docking Study | 1-gen-2023 | Patamia, Vincenzo; Floresta, Giuseppe; Zagni, Chiara; Pistara', Venerando; Punzo, Francesco; Rescifina, Antonio | file da validare |
3D-QSAR assisted identification of FABP4 inhibitors: An effective scaffold hopping analysis/QSAR evaluation | 1-gen-2019 | Floresta, G.; Cilibrizzi, A.; Abbate, V.; Spampinato, A.; Zagni, C.; Rescifina, A. | |
[1]Benzothieno[3,2-d]pyrimidine derivatives as ligands for the serotonergic 5-HT7 receptor | 1-gen-2019 | Romeo, Giuseppe; Salerno, Loredana; Pittalà, Valeria; Candido, Marialuisa; Intagliata, Sebastiano; Amata, Emanuele; Salmona, Mario; Cagnotto, Alfredo; Rescifina, Antonio; Floresta, Giuseppe; Modica, Maria Nunziata | |
A hexameric resorcinarene capsule as a hydrogen bonding catalyst in the conjugate addition of pyrroles and indoles to nitroalkenes | 1-gen-2019 | Gambaro, S.; De Rosa, M.; Soriente, A.; Talotta, C.; Floresta, G.; Rescifina, A.; Gaeta, C.; Neri, P. | |
A pseudouridine isoxazolidinyl nucleoside analogue structural analysis: A morphological approach | 1-gen-2018 | Floresta, Giuseppe; Pistara', Venerando; Christensen E., Kirsten; Amata, Emanuele; Marrazzo, Agostino; Gentile, Davide; Rescifina, Antonio; Punzo, Francesco | |
A Rare Natural Benzo[k,l]xanthene as a Turn-Off Fluorescent Sensor for Cu2+ Ion | 1-gen-2020 | Floresta, Giuseppe; Cardullo, Nunzio; Spatafora, Carmela; Rescifina, Antonio; Tringali, Corrado | file da validare |
A structure-and ligand-based virtual screening of a database of “small” marine natural products for the identification of “blue” sigma-2 receptor ligands | 1-gen-2018 | Floresta, Giuseppe; Amata, Emanuele; Barbaraci, Carla; Gentile, Davide; Turnaturi, Rita; Marrazzo, Agostino; Rescifina, Antonio | |
Adipocyte fatty acid binding protein 4 (FABP4) inhibitors. A comprehensive systematic review | 1-gen-2017 | Floresta, Giuseppe; Pistarà, Venerando; Amata, Emanuele; Dichiara, Maria; Marrazzo, Agostino; Prezzavento, Orazio; Rescifina, Antonio | |
Adipocyte fatty acid binding protein 4 (FABP4) inhibitors. An update from 2017 to early 2022 | 1-gen-2022 | Floresta, G.; Patamia, V.; Zagni, C.; Rescifina, A. | file da validare |
Ammidi dell’acido rosmarinico come potenziali agenti antidiabetici | 1-gen-2019 | Muccilli, V; Cardullo, N; Catinella, G; Floresta, G; Rosselli, S; Rescifina, A; Bruno, M; Tringali., C | |
An integrated pharmacophore/docking/3D-QSAR approach to screening a large library of products in search of future botulinum neurotoxin a inhibitors | 1-gen-2020 | Gentile, D.; Floresta, G.; Patamia, V.; Chiaramonte, R.; Mauro, G. L.; Rescifina, A.; Vecchio, M. | |
An Overview of PDE4 Inhibitors in Clinical Trials: 2010 to Early 2022 | 1-gen-2022 | Crocetti, L.; Floresta, G.; Cilibrizzi, A.; Giovannoni, M. P. | |
Artificial Intelligence Technologies for COVID-19 De Novo Drug Design | 1-gen-2022 | Floresta, G.; Zagni, C.; Gentile, D.; Patamia, V.; Rescifina, A. | file da validare |
Carbamoyl-Decorated Cyclodextrins for Carbon Dioxide Adsorption | 1-gen-2023 | Patamia, Vincenzo; Tomarchio, Rosario; Fiorenza, Roberto; Zagni, Chiara; Scire', Salvatore; Floresta, Giuseppe; Rescifina, Antonio | file da validare |
Chromatograpic resolution of phenylethanolic-azole racemic compounds highlighted stereoselective inhibition of heme oxygenase-1 by (R)-enantiomers | 1-gen-2020 | Floresta, G.; Carotti, A.; Ianni, F.; Sorrenti, V.; Intagliata, S.; Rescifina, A.; Salerno, L.; Di Michele, A.; Sardella, R.; Pittala, V. | |
Computational tools in the discovery of FABP4 ligands: A statistical and molecular modeling approach | 1-gen-2019 | Floresta, G.; Gentile, D.; Perrini, G.; Patamia, Vincenzo; Rescifina, A. | |
Computer-Assisted Design of Peptide-Based Radiotracers | 1-gen-2023 | Patamia, Vincenzo; Zagni, Chiara; Brullo, Ilaria; Saccullo, Erika; Coco, Alessandro; Floresta, Giuseppe; Rescifina, Antonio | file da validare |
Cucurbit[7]uril as a catalytic nanoreactor for one-pot synthesis of isoxazolidines in water | 1-gen-2020 | Gentile, Davide; Floresta, Giuseppe; Patamia, Vincenzo; Nicosia, Angelo; Mineo, Placido; Rescifina, Antonio | |
Design and synthesis of novel compounds as fatty acids binding protein inhibitors and as gallium-68 chelators for positron emission tomography | 9-nov-2018 | Floresta, Giuseppe | |
Development of a Sigma-2 Receptor affinity filter through a Monte Carlo based QSAR analysis | 1-gen-2017 | Rescifina, Antonio; Floresta, Giuseppe; Marrazzo, Agostino; Parenti, Carmela; Prezzavento, Orazio; Nastasi, Giovanni; Dichiara, Maria; Amata, Emanuele |