Sfoglia per Autore
Methoctramine-related polymethylene tetraamines. 4(1)-chirality effect on M2 muscarinic receptor blocking activity
file da validare1991-01-01 Giardina, D.; Marrazzo, A.; Marucci, G.; Grazia Piloni, M.; Quaglia, W.
Synthesis, physical properties ans toxicological studies of L-pyroglutamic and L-glutamic acid esters of acetamininophen as potentially useful prodrugs
file da validare1995-01-01 Bousquet, E; Tirendi, S; Spadaro, Angelo; Marrazzo, Agostino; Puglisi, Giovanni
Selective Ligands for Sigma1 Receptors with Agonist or Antagonist Properties
file da validare1995-01-01 Ronsisvalle, G.; Marrazzo, Agostino; Prezzavento, Orazio; Pittala', Valeria; Pappalardo, M. S.; Vittorio, F.; Spampinato, S.
New developments in opioid receptors ligands
file da validare1995-01-01 Ronsisvalle, G; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Marrazzo, Agostino; Vittorio, F; Pappalardo, Ms; Bousquet, E.
CCB, a novel specific kappa opioid agonist, which discriminates between opioid and sigma 1 recognition sites
1995-01-01 Ronsisvalle, Giuseppe; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Marrazzo, Agostino; Vittorio, F; Gomez Vidal, Ja; Carboni, L; Spampinato, S.
Synthesis and antimicrobial evaluation of 4-phenyl-3-isoquinolinoyl-hydrazones
file da validare1995-01-01 Vittorio, F; Ronsisvalle, G; Marrazzo, Agostino; Blandino, Giovanna
Progettazione, Sintesi e Profilo Farmacologico di Ligandi Sigma-Selettivi
file da validare1996-01-01 Ronsisvalle, Giuseppe; Marrazzo, Agostino; Pittala', Valeria
PEPTIDOMIMETICS OF THE KAPPA-OPIOID RECEPTOR. A HYBRID MPCB /PEPTIDE LIGAND (MPCB-RRI) BINDS KAPPA CLONED RECEPTOR WITH NANOMOLAR AFFINITY
file da validare1996-01-01 Ronsisvalle, Giuseppe; PAPPALARDO M., S; Carboni, L; Vittorio, F; Pasquinucci, Lorella Giuseppina; Marrazzo, Agostino; Cacciaguerra, S; Spampinato, S.
Synthesis, physical properties, toxicological studies and bioavailability of L-pyroglutamic and L-glutamic acid esters of paracetamol as potentially useful prodrugs
file da validare1996-01-01 Bousquet, E; Marrazzo, Agostino; Puglisi, Giovanni; Spadaro, Angelo; Tirendi, S.
SYNTHESIS OF (+)-(1'R,2'S) AND (1'S,2'R)-6,11-DIMETHYL-1,2,3,4,5,6-HEXAHYDRO-3-[[2'-(ALKOXYCARBONYL)-2'-PHENYLCYCLOPROPYL]METHYL]-2,6-METHANO-3-BENZAZOCIN-8-OL. COMPARISON OF THE AFFINITIES FOR SIGMA 1 AND OPIOID RECEPTORS WITHIN THE DIASTEREOISOMERIC MPCB AND CCB
file da validare1997-01-01 Ronsisvalle, Giuseppe; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Pappalardo, Ms; Marrazzo, Agostino; Vittorio, F; Carboni, L; Spampinato, S.
(+)-cis-N-ethyleneamino-N-normetazocine derivatives. Novel and selective sigma ligands with antagonist properties
1998-01-01 Ronsisvalle, G; Marrazzo, Agostino; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Vittorio, F; Pittala', Valeria; Pappalardo, Ms; Cacciaguerra, S; Spampinato, S.
Synthesis of (+) and (−)-cis-2-[(1-adamantylamino)-methyl]-1-phenylcyclopropane derivatives as probe for sigma-1 and sigma-2 binding sites
file da validare2000-01-01 Marrazzo, A; Prezzavento, O.; Vittorio, Franco; Pappalardo, M. S.; Ronsisvalle, G
Nonpeptide Analogues of Dynorphin A(1-8): Design, Synthesis, and Pharmacological Evaluation of k-Selective Agonists
2000-01-01 Ronsisvalle, G; Pasquinucci, Lorella Giuseppina; Pittala', Valeria; Marrazzo, A; Prezzavento, Orazio; DI TORO, R; Falcucci, B; Spampinato, S.
Specific kappa opioid receptor agonists
file da validare2000-01-01 Ronsisvalle, G; Marrazzo, A; Pasquinucci, L; Prezzavento, Orazio; Pappalardo, M; Vittorio, F.
Synthesis and pharmacological evaluation of potent and enantioselective sigma-1 and sigma-2 ligands
file da validare2000-01-01 Marrazzo, Agostino; Prezzavento, Orazio; Ronsisvalle, G.
Substituted 1-phenyl-2-cyclopropylmethylamines with high affinity and selectivity for sigma sites
2000-01-01 Ronsisvalle, Giuseppe; Marrazzo, Agostino; Falcucci, B; DI TORO, D; Spampinato, S; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina
Methyl 1-phenyl-2-{[(2,6,6-trimethylbicyclo[3.1.1]hept-3-yl)amino]methyl}cyclopropane-carboxylate diastereoisomers as potent and enantioselective sigma-1 and sigma-2 ligands
file da validare2001-01-01 Ronsisvalle, G; Marrazzo, Agostino; Panebianco, A; Prezzavento, Orazio
Synthesis and pharmacological evaluation of potent and enantioselective sigma-1 and sigma-2 ligands
2001-01-01 Marrazzo, Agostino; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Vittorio, F; Ronsisvalle, Giuseppe
Synthesis and binding affinity of cis-(–)- and cis-(+)-N-ethyleneamino-N-nordeoxymetazocine and cis-(–)-N-normetazocine analogues at σ1, σ2 and κ opioid receptors
2001-01-01 Ronsisvalle, G; Prezzavento, O; Marrazzo, Agostino; Vittorio, F; Bousquet, E; DI TORO, R; Spampinato, S.
Opioid and sigma receptor studies. New developments in the design of selective sigma ligands
2001-01-01 Ronsisvalle, G; Marrazzo, A; Prezzavento, O; Cagnotto, A; Mennini, T; Parenti, C; Scoto, Giovanna Maria
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Methoctramine-related polymethylene tetraamines. 4(1)-chirality effect on M2 muscarinic receptor blocking activity | 1-gen-1991 | Giardina, D.; Marrazzo, A.; Marucci, G.; Grazia Piloni, M.; Quaglia, W. | file da validare |
| Synthesis, physical properties ans toxicological studies of L-pyroglutamic and L-glutamic acid esters of acetamininophen as potentially useful prodrugs | 1-gen-1995 | Bousquet, E; Tirendi, S; Spadaro, Angelo; Marrazzo, Agostino; Puglisi, Giovanni | file da validare |
| Selective Ligands for Sigma1 Receptors with Agonist or Antagonist Properties | 1-gen-1995 | Ronsisvalle, G.; Marrazzo, Agostino; Prezzavento, Orazio; Pittala', Valeria; Pappalardo, M. S.; Vittorio, F.; Spampinato, S. | file da validare |
| New developments in opioid receptors ligands | 1-gen-1995 | Ronsisvalle, G; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Marrazzo, Agostino; Vittorio, F; Pappalardo, Ms; Bousquet, E. | file da validare |
| CCB, a novel specific kappa opioid agonist, which discriminates between opioid and sigma 1 recognition sites | 1-gen-1995 | Ronsisvalle, Giuseppe; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Marrazzo, Agostino; Vittorio, F; Gomez Vidal, Ja; Carboni, L; Spampinato, S. | |
| Synthesis and antimicrobial evaluation of 4-phenyl-3-isoquinolinoyl-hydrazones | 1-gen-1995 | Vittorio, F; Ronsisvalle, G; Marrazzo, Agostino; Blandino, Giovanna | file da validare |
| Progettazione, Sintesi e Profilo Farmacologico di Ligandi Sigma-Selettivi | 1-gen-1996 | Ronsisvalle, Giuseppe; Marrazzo, Agostino; Pittala', Valeria | file da validare |
| PEPTIDOMIMETICS OF THE KAPPA-OPIOID RECEPTOR. A HYBRID MPCB /PEPTIDE LIGAND (MPCB-RRI) BINDS KAPPA CLONED RECEPTOR WITH NANOMOLAR AFFINITY | 1-gen-1996 | Ronsisvalle, Giuseppe; PAPPALARDO M., S; Carboni, L; Vittorio, F; Pasquinucci, Lorella Giuseppina; Marrazzo, Agostino; Cacciaguerra, S; Spampinato, S. | file da validare |
| Synthesis, physical properties, toxicological studies and bioavailability of L-pyroglutamic and L-glutamic acid esters of paracetamol as potentially useful prodrugs | 1-gen-1996 | Bousquet, E; Marrazzo, Agostino; Puglisi, Giovanni; Spadaro, Angelo; Tirendi, S. | file da validare |
| SYNTHESIS OF (+)-(1'R,2'S) AND (1'S,2'R)-6,11-DIMETHYL-1,2,3,4,5,6-HEXAHYDRO-3-[[2'-(ALKOXYCARBONYL)-2'-PHENYLCYCLOPROPYL]METHYL]-2,6-METHANO-3-BENZAZOCIN-8-OL. COMPARISON OF THE AFFINITIES FOR SIGMA 1 AND OPIOID RECEPTORS WITHIN THE DIASTEREOISOMERIC MPCB AND CCB | 1-gen-1997 | Ronsisvalle, Giuseppe; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Pappalardo, Ms; Marrazzo, Agostino; Vittorio, F; Carboni, L; Spampinato, S. | file da validare |
| (+)-cis-N-ethyleneamino-N-normetazocine derivatives. Novel and selective sigma ligands with antagonist properties | 1-gen-1998 | Ronsisvalle, G; Marrazzo, Agostino; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Vittorio, F; Pittala', Valeria; Pappalardo, Ms; Cacciaguerra, S; Spampinato, S. | |
| Synthesis of (+) and (−)-cis-2-[(1-adamantylamino)-methyl]-1-phenylcyclopropane derivatives as probe for sigma-1 and sigma-2 binding sites | 1-gen-2000 | Marrazzo, A; Prezzavento, O.; Vittorio, Franco; Pappalardo, M. S.; Ronsisvalle, G | file da validare |
| Nonpeptide Analogues of Dynorphin A(1-8): Design, Synthesis, and Pharmacological Evaluation of k-Selective Agonists | 1-gen-2000 | Ronsisvalle, G; Pasquinucci, Lorella Giuseppina; Pittala', Valeria; Marrazzo, A; Prezzavento, Orazio; DI TORO, R; Falcucci, B; Spampinato, S. | |
| Specific kappa opioid receptor agonists | 1-gen-2000 | Ronsisvalle, G; Marrazzo, A; Pasquinucci, L; Prezzavento, Orazio; Pappalardo, M; Vittorio, F. | file da validare |
| Synthesis and pharmacological evaluation of potent and enantioselective sigma-1 and sigma-2 ligands | 1-gen-2000 | Marrazzo, Agostino; Prezzavento, Orazio; Ronsisvalle, G. | file da validare |
| Substituted 1-phenyl-2-cyclopropylmethylamines with high affinity and selectivity for sigma sites | 1-gen-2000 | Ronsisvalle, Giuseppe; Marrazzo, Agostino; Falcucci, B; DI TORO, D; Spampinato, S; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina | |
| Methyl 1-phenyl-2-{[(2,6,6-trimethylbicyclo[3.1.1]hept-3-yl)amino]methyl}cyclopropane-carboxylate diastereoisomers as potent and enantioselective sigma-1 and sigma-2 ligands | 1-gen-2001 | Ronsisvalle, G; Marrazzo, Agostino; Panebianco, A; Prezzavento, Orazio | file da validare |
| Synthesis and pharmacological evaluation of potent and enantioselective sigma-1 and sigma-2 ligands | 1-gen-2001 | Marrazzo, Agostino; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Vittorio, F; Ronsisvalle, Giuseppe | |
| Synthesis and binding affinity of cis-(–)- and cis-(+)-N-ethyleneamino-N-nordeoxymetazocine and cis-(–)-N-normetazocine analogues at σ1, σ2 and κ opioid receptors | 1-gen-2001 | Ronsisvalle, G; Prezzavento, O; Marrazzo, Agostino; Vittorio, F; Bousquet, E; DI TORO, R; Spampinato, S. | |
| Opioid and sigma receptor studies. New developments in the design of selective sigma ligands | 1-gen-2001 | Ronsisvalle, G; Marrazzo, A; Prezzavento, O; Cagnotto, A; Mennini, T; Parenti, C; Scoto, Giovanna Maria |
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