Sfoglia per Autore
Synthesis and antimicrobial evaluation of 4-phenyl-3-isoquinolinoyl-hydrazones
file da validare1995-01-01 Vittorio, F; Ronsisvalle, G; Marrazzo, Agostino; Blandino, Giovanna
CCB, a novel specific kappa opioid agonist, which discriminates between opioid and sigma 1 recognition sites
1995-01-01 Ronsisvalle, Giuseppe; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Marrazzo, Agostino; Vittorio, F; Gomez Vidal, Ja; Carboni, L; Spampinato, S.
Selective Ligands for Sigma1 Receptors with Agonist or Antagonist Properties
file da validare1995-01-01 Ronsisvalle, G.; Marrazzo, Agostino; Prezzavento, Orazio; Pittala', Valeria; Pappalardo, M. S.; Vittorio, F.; Spampinato, S.
New developments in opioid receptors ligands
file da validare1995-01-01 Ronsisvalle, G; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Marrazzo, Agostino; Vittorio, F; Pappalardo, Ms; Bousquet, E.
Synthesis, physical properties ans toxicological studies of L-pyroglutamic and L-glutamic acid esters of acetamininophen as potentially useful prodrugs
file da validare1995-01-01 Bousquet, E; Tirendi, S; Spadaro, Angelo; Marrazzo, Agostino; Puglisi, Giovanni
PEPTIDOMIMETICS OF THE KAPPA-OPIOID RECEPTOR. A HYBRID MPCB /PEPTIDE LIGAND (MPCB-RRI) BINDS KAPPA CLONED RECEPTOR WITH NANOMOLAR AFFINITY
file da validare1996-01-01 Ronsisvalle, Giuseppe; PAPPALARDO M., S; Carboni, L; Vittorio, F; Pasquinucci, Lorella Giuseppina; Marrazzo, Agostino; Cacciaguerra, S; Spampinato, S.
Synthesis, physical properties, toxicological studies and bioavailability of L-pyroglutamic and L-glutamic acid esters of paracetamol as potentially useful prodrugs
file da validare1996-01-01 Bousquet, E; Marrazzo, Agostino; Puglisi, Giovanni; Spadaro, Angelo; Tirendi, S.
Progettazione, Sintesi e Profilo Farmacologico di Ligandi Sigma-Selettivi
file da validare1996-01-01 Ronsisvalle, Giuseppe; Marrazzo, Agostino; Pittala', Valeria
SYNTHESIS OF (+)-(1'R,2'S) AND (1'S,2'R)-6,11-DIMETHYL-1,2,3,4,5,6-HEXAHYDRO-3-[[2'-(ALKOXYCARBONYL)-2'-PHENYLCYCLOPROPYL]METHYL]-2,6-METHANO-3-BENZAZOCIN-8-OL. COMPARISON OF THE AFFINITIES FOR SIGMA 1 AND OPIOID RECEPTORS WITHIN THE DIASTEREOISOMERIC MPCB AND CCB
file da validare1997-01-01 Ronsisvalle, Giuseppe; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Pappalardo, Ms; Marrazzo, Agostino; Vittorio, F; Carboni, L; Spampinato, S.
(+)-cis-N-ethyleneamino-N-normetazocine derivatives. Novel and selective sigma ligands with antagonist properties
1998-01-01 Ronsisvalle, G; Marrazzo, Agostino; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Vittorio, F; Pittala', Valeria; Pappalardo, Ms; Cacciaguerra, S; Spampinato, S.
Synthesis and pharmacological evaluation of potent and enantioselective sigma-1 and sigma-2 ligands
file da validare2000-01-01 Marrazzo, Agostino; Prezzavento, Orazio; Ronsisvalle, G.
Synthesis of (+) and (−)-cis-2-[(1-adamantylamino)-methyl]-1-phenylcyclopropane derivatives as probe for sigma-1 and sigma-2 binding sites
file da validare2000-01-01 Marrazzo, A; Prezzavento, O.; Vittorio, Franco; Pappalardo, M. S.; Ronsisvalle, G
Nonpeptide Analogues of Dynorphin A(1-8): Design, Synthesis, and Pharmacological Evaluation of k-Selective Agonists
2000-01-01 Ronsisvalle, G; Pasquinucci, Lorella Giuseppina; Pittala', Valeria; Marrazzo, A; Prezzavento, Orazio; DI TORO, R; Falcucci, B; Spampinato, S.
Substituted 1-phenyl-2-cyclopropylmethylamines with high affinity and selectivity for sigma sites
2000-01-01 Ronsisvalle, Giuseppe; Marrazzo, Agostino; Falcucci, B; DI TORO, D; Spampinato, S; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina
Specific kappa opioid receptor agonists
file da validare2000-01-01 Ronsisvalle, G; Marrazzo, A; Pasquinucci, L; Prezzavento, Orazio; Pappalardo, M; Vittorio, F.
Methyl 1-phenyl-2-{[(2,6,6-trimethylbicyclo[3.1.1]hept-3-yl)amino]methyl}cyclopropane-carboxylate diastereoisomers as potent and enantioselective sigma-1 and sigma-2 ligands
file da validare2001-01-01 Ronsisvalle, G; Marrazzo, Agostino; Panebianco, A; Prezzavento, Orazio
Novel methyl-2-[4-[(4-hydroxy-4-phenylpiperidin-1-yl)methyl]-1-phenylcyclopropane-carboxylate derivatives as sigma-1 and sigma-2 receptor ligands
file da validare2001-01-01 Prezzavento, O; Massimino, M; Marrazzo, Agostino; Pasquinucci, Lorella Giuseppina; Ronsisvalle, G.
Specific kappa opioid receptor agonists
2001-01-01 Ronsisvalle, Giuseppe; Marrazzo, Agostino; Pasquinucci, Lorella Giuseppina; Prezzavento, O; Pappalardo, M; Vittorio, F.
Opioid and sigma receptor studies. New developments in the design of selective sigma ligands
2001-01-01 Ronsisvalle, G; Marrazzo, A; Prezzavento, O; Cagnotto, A; Mennini, T; Parenti, C; Scoto, Giovanna Maria
PHARMACOLOGICAL EVALUATION OF POTENT SIGMA LIGANDS IN β-AMYLOID INDUCED NEURODEGENERATION
file da validare2001-01-01 Ferrara, G; Marrazzo, Agostino; Copani, Agata Graziella; Prezzavento, O; Ronsisvalle, G.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Synthesis and antimicrobial evaluation of 4-phenyl-3-isoquinolinoyl-hydrazones | 1-gen-1995 | Vittorio, F; Ronsisvalle, G; Marrazzo, Agostino; Blandino, Giovanna | file da validare |
CCB, a novel specific kappa opioid agonist, which discriminates between opioid and sigma 1 recognition sites | 1-gen-1995 | Ronsisvalle, Giuseppe; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Marrazzo, Agostino; Vittorio, F; Gomez Vidal, Ja; Carboni, L; Spampinato, S. | |
Selective Ligands for Sigma1 Receptors with Agonist or Antagonist Properties | 1-gen-1995 | Ronsisvalle, G.; Marrazzo, Agostino; Prezzavento, Orazio; Pittala', Valeria; Pappalardo, M. S.; Vittorio, F.; Spampinato, S. | file da validare |
New developments in opioid receptors ligands | 1-gen-1995 | Ronsisvalle, G; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Marrazzo, Agostino; Vittorio, F; Pappalardo, Ms; Bousquet, E. | file da validare |
Synthesis, physical properties ans toxicological studies of L-pyroglutamic and L-glutamic acid esters of acetamininophen as potentially useful prodrugs | 1-gen-1995 | Bousquet, E; Tirendi, S; Spadaro, Angelo; Marrazzo, Agostino; Puglisi, Giovanni | file da validare |
PEPTIDOMIMETICS OF THE KAPPA-OPIOID RECEPTOR. A HYBRID MPCB /PEPTIDE LIGAND (MPCB-RRI) BINDS KAPPA CLONED RECEPTOR WITH NANOMOLAR AFFINITY | 1-gen-1996 | Ronsisvalle, Giuseppe; PAPPALARDO M., S; Carboni, L; Vittorio, F; Pasquinucci, Lorella Giuseppina; Marrazzo, Agostino; Cacciaguerra, S; Spampinato, S. | file da validare |
Synthesis, physical properties, toxicological studies and bioavailability of L-pyroglutamic and L-glutamic acid esters of paracetamol as potentially useful prodrugs | 1-gen-1996 | Bousquet, E; Marrazzo, Agostino; Puglisi, Giovanni; Spadaro, Angelo; Tirendi, S. | file da validare |
Progettazione, Sintesi e Profilo Farmacologico di Ligandi Sigma-Selettivi | 1-gen-1996 | Ronsisvalle, Giuseppe; Marrazzo, Agostino; Pittala', Valeria | file da validare |
SYNTHESIS OF (+)-(1'R,2'S) AND (1'S,2'R)-6,11-DIMETHYL-1,2,3,4,5,6-HEXAHYDRO-3-[[2'-(ALKOXYCARBONYL)-2'-PHENYLCYCLOPROPYL]METHYL]-2,6-METHANO-3-BENZAZOCIN-8-OL. COMPARISON OF THE AFFINITIES FOR SIGMA 1 AND OPIOID RECEPTORS WITHIN THE DIASTEREOISOMERIC MPCB AND CCB | 1-gen-1997 | Ronsisvalle, Giuseppe; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Pappalardo, Ms; Marrazzo, Agostino; Vittorio, F; Carboni, L; Spampinato, S. | file da validare |
(+)-cis-N-ethyleneamino-N-normetazocine derivatives. Novel and selective sigma ligands with antagonist properties | 1-gen-1998 | Ronsisvalle, G; Marrazzo, Agostino; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina; Vittorio, F; Pittala', Valeria; Pappalardo, Ms; Cacciaguerra, S; Spampinato, S. | |
Synthesis and pharmacological evaluation of potent and enantioselective sigma-1 and sigma-2 ligands | 1-gen-2000 | Marrazzo, Agostino; Prezzavento, Orazio; Ronsisvalle, G. | file da validare |
Synthesis of (+) and (−)-cis-2-[(1-adamantylamino)-methyl]-1-phenylcyclopropane derivatives as probe for sigma-1 and sigma-2 binding sites | 1-gen-2000 | Marrazzo, A; Prezzavento, O.; Vittorio, Franco; Pappalardo, M. S.; Ronsisvalle, G | file da validare |
Nonpeptide Analogues of Dynorphin A(1-8): Design, Synthesis, and Pharmacological Evaluation of k-Selective Agonists | 1-gen-2000 | Ronsisvalle, G; Pasquinucci, Lorella Giuseppina; Pittala', Valeria; Marrazzo, A; Prezzavento, Orazio; DI TORO, R; Falcucci, B; Spampinato, S. | |
Substituted 1-phenyl-2-cyclopropylmethylamines with high affinity and selectivity for sigma sites | 1-gen-2000 | Ronsisvalle, Giuseppe; Marrazzo, Agostino; Falcucci, B; DI TORO, D; Spampinato, S; Prezzavento, Orazio; Pasquinucci, Lorella Giuseppina | |
Specific kappa opioid receptor agonists | 1-gen-2000 | Ronsisvalle, G; Marrazzo, A; Pasquinucci, L; Prezzavento, Orazio; Pappalardo, M; Vittorio, F. | file da validare |
Methyl 1-phenyl-2-{[(2,6,6-trimethylbicyclo[3.1.1]hept-3-yl)amino]methyl}cyclopropane-carboxylate diastereoisomers as potent and enantioselective sigma-1 and sigma-2 ligands | 1-gen-2001 | Ronsisvalle, G; Marrazzo, Agostino; Panebianco, A; Prezzavento, Orazio | file da validare |
Novel methyl-2-[4-[(4-hydroxy-4-phenylpiperidin-1-yl)methyl]-1-phenylcyclopropane-carboxylate derivatives as sigma-1 and sigma-2 receptor ligands | 1-gen-2001 | Prezzavento, O; Massimino, M; Marrazzo, Agostino; Pasquinucci, Lorella Giuseppina; Ronsisvalle, G. | file da validare |
Specific kappa opioid receptor agonists | 1-gen-2001 | Ronsisvalle, Giuseppe; Marrazzo, Agostino; Pasquinucci, Lorella Giuseppina; Prezzavento, O; Pappalardo, M; Vittorio, F. | |
Opioid and sigma receptor studies. New developments in the design of selective sigma ligands | 1-gen-2001 | Ronsisvalle, G; Marrazzo, A; Prezzavento, O; Cagnotto, A; Mennini, T; Parenti, C; Scoto, Giovanna Maria | |
PHARMACOLOGICAL EVALUATION OF POTENT SIGMA LIGANDS IN β-AMYLOID INDUCED NEURODEGENERATION | 1-gen-2001 | Ferrara, G; Marrazzo, Agostino; Copani, Agata Graziella; Prezzavento, O; Ronsisvalle, G. | file da validare |
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