IRIS
RONSISVALLE, Giuseppe
 Distribuzione geografica
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Continente #
NA - Nord America 2.732
EU - Europa 1.576
AS - Asia 578
AF - Africa 198
OC - Oceania 4
Continente sconosciuto - Info sul continente non disponibili 3
SA - Sud America 1
Totale 5.092
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Nazione #
US - Stati Uniti d'America 2.553
UA - Ucraina 501
IE - Irlanda 467
CN - Cina 447
CA - Canada 179
DE - Germania 156
CI - Costa d'Avorio 150
RU - Federazione Russa 134
IT - Italia 108
SE - Svezia 88
VN - Vietnam 70
SN - Senegal 48
GB - Regno Unito 24
CH - Svizzera 22
BE - Belgio 17
IR - Iran 17
IN - India 15
FR - Francia 14
NL - Olanda 9
AT - Austria 8
CZ - Repubblica Ceca 8
GR - Grecia 8
LB - Libano 6
PL - Polonia 5
UZ - Uzbekistan 5
AU - Australia 3
EU - Europa 3
PK - Pakistan 3
SG - Singapore 3
ID - Indonesia 2
KR - Corea 2
TR - Turchia 2
TW - Taiwan 2
AL - Albania 1
BG - Bulgaria 1
DK - Danimarca 1
ES - Italia 1
FI - Finlandia 1
HK - Hong Kong 1
HU - Ungheria 1
IL - Israele 1
JP - Giappone 1
LV - Lettonia 1
NZ - Nuova Zelanda 1
PE - Perù 1
PH - Filippine 1
Totale 5.092
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Città #
Jacksonville 607
Chandler 566
Dublin 465
Nanjing 170
Abidjan 150
Toronto 147
Cambridge 132
Andover 130
Lawrence 129
Grafing 119
Ashburn 117
San Mateo 94
Boardman 85
Dong Ket 69
Des Moines 64
Catania 61
Wilmington 54
Nanchang 52
Shenyang 49
Dakar 48
Houston 47
Saint Petersburg 43
Ottawa 29
Jiaxing 28
Hebei 27
Bremen 26
Tianjin 26
Moscow 19
Changsha 18
Brussels 17
Norwalk 15
Ardabil 14
Kunming 12
Falls Church 11
Ningbo 11
Augusta 10
Den Haag 8
Jinan 8
Liberty Lake 8
Washington 8
Leawood 6
Ann Arbor 5
Beijing 5
Changchun 5
Hangzhou 5
Pune 5
Guangzhou 4
Prague 4
Seattle 4
Tappahannock 4
Zhengzhou 4
Fuzhou 3
Lahore 3
Lercara Friddi 3
Paris 3
Rome 3
Arklow 2
Bangalore 2
Bari 2
Ludwigshafen 2
Melbourne 2
Mountain View 2
Phoenix 2
Redwood City 2
San Francisco 2
Scarborough 2
Taipei 2
Vicenza 2
Amsterdam 1
Budapest 1
Canberra 1
Central 1
Chicago 1
Christchurch 1
Copenhagen 1
Florence 1
Frankfurt Am Main 1
Frankfurt am Main 1
Ghisalba 1
Guidonia Montecelio 1
Haikou 1
Hanover 1
Helsinki 1
Ho Chi Minh City 1
Iligan City 1
Jinhua 1
Kiev 1
Kyiv 1
Lanzhou 1
Lima 1
London 1
Los Angeles 1
Lvov 1
Madrid 1
Messina 1
Misterbianco 1
Monzuno 1
Mumbai 1
New York 1
Newark 1
Totale 3.815
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Nome #
1-Phenyl-3azabicyclo[3.1.0]hexane derivatives as new ligands for sigma receptors 87
1,4-Benzothiazines. IV 86
Design, Synthesis and Antiinflammatory Activity of Novel g-Tocopherol Acetylsalicylic acid Ester Codrug 86
Antiproliferative activity of phenylbutyrate ester of haloperidol metabolite II [(±)-MRJF4] in prostate cancer cells 72
4-Quinazolinones: synthesis and reduction of prostaglandin E-2 production 68
CCB, a novel specific kappa opioid agonist, which discriminates between opioid and sigma 1 recognition sites 61
A novel adamantane derivative attenuates retinal ischemia-reperfusion damage in the rat retina through sigma1 receptors 58
The benzomorphan-based LP1 ligand is a suitable MOR/DOR agonist for chronic pain treatment 58
CCB - A novel analog of MPCB with high binding affinity and specific kappa opioid receptor agonist 58
An improved synthesis of the antimalarial di(4-acetylaminophenil)sulfone 56
The in vitro effect of a lyophilized extract of wine obtained from Jacquez grapes on human chondrocytes 55
Amidinobenzisothiazole derivatives with antidegenerative activity on cartilage 55
Conformational aspects of some odd-membered disulfide-bridged metacyclophanes derived from m-dimethoxybenzene 54
Antinociceptive profile of LP1, a non-peptide multitarget opioid ligand. 54
6-Hydroxy-1,2,3,4-tetrahydro-isoquinoline-3-caboxylic acid mimics active conformation of tyrosine in opioid peptides 53
A novel and selective sigma-1/2 receptor ligand (PO680C): Binding properties and expression of tissue transglutaminase 53
13C NMR of N-Heterocycles. Conformation of Phenothiazines and 2,3-diazaphenothiazines 52
SYNTHESIS OF (+)-(1'R,2'S) AND (1'S,2'R)-6,11-DIMETHYL-1,2,3,4,5,6-HEXAHYDRO-3-[[2'-(ALKOXYCARBONYL)-2'-PHENYLCYCLOPROPYL]METHYL]-2,6-METHANO-3-BENZAZOCIN-8-OL. COMPARISON OF THE AFFINITIES FOR SIGMA 1 AND OPIOID RECEPTORS WITHIN THE DIASTEREOISOMERIC MPCB AND CCB 52
2,3-Diazaphenothiazine. VII. Quaternization reactions 52
SYNTHESIS AND SPASMOLYTIC ACTIVITY OF 2-SUBSTITUTED THIENOPYRIMIDIN-4-ONE DERIVATIVES 51
Synthesis and inclusion properties of some 10,12,24,26-tetrasubstituted 3,5,17,19-tetranitro-1,8,15,22-tetrathia[1.1.1.1]metacyclophanes 51
Nonpeptide Analogues of Dynorphin A(1-8): Design, Synthesis, and Pharmacological Evaluation of k-Selective Agonists 50
Synthesis and antimicrobial evaluation of 4-phenyl-3-isoquinolinoyl-hidrazones 50
Substituted 1-phenyl-2-cyclopropylmethylamines with high affinity and selectivity for sigma sites 50
Solution conformation of bis(m-nitrophenyl)disulphide 49
(+)-cis-N-ethyleneamino-N-normetazocine derivatives. Novel and selective sigma ligands with antagonist properties 49
Effects of leflunomide on human cartilage 48
Protective effect of capparis spinosa on chondrocites 48
Multitarget opioid ligands in pain relief: New players in an old game 48
Synthesis and immunostimulating activity of a thioglycolipopeptide glycomimetic as a potential anticancer vaccine derived from Tn antigen 48
Synthesis and pharmacological evaluation of MRJF4 as new potential anticancer tool 48
Reaction of cyanothioacetamide with ethyl bromopyruvate and ethyl beta-chloroacetone oxalate. I. New synthesis of thieno[2,3-b]pyridines 48
Benzomorphan-based opioid ligands with mixed m agonist/d antagonist activity 48
Multitarget Opioid/Non-opioid Ligands: A Potential Approach in Pain Management 48
Non-peptide ligands for opioid receptors. Design of kappa-specific agonists 47
European Medicinal Chemistry Education: the trasformational accomplishments and challenges 47
Bivalent opioid-peptides synthesized from mu-selective monomers display preferential selectivity for delta-receptors 47
Stereoisomerisation precesses in cis-octahedral-bis-chelòate complexes: activation energies associated with the different rearrangement modes in the case of phenylchlorobis(benzoylacetato)tin 46
modeling of k-opioid receptor/agonists interactions using pharmacophore-based and docking simulations 45
Calorimetric study in the interactio of thienopyrimidine derivatives with phosphatidylcholine membranes 45
Neuroprotective effect of the new sigma receptor ligands cis-(+) and cis-(–)-PPCC 45
Intrastriatal administration of sigma ligands inhibits basal dopamine release in vivo 44
Synthesis and anti-measles virus activity of new isoquinolin-4-one derivatives 44
Synthesis, characterization and stereochemistry of bis(isobutyrylketonate) complexes of II group metals 44
Sintesi di 2,3-diazafenotiazine. Nota X. 44
Analysis of ecdysteroids by micellar electrokinetic chromatography with on-line preconcentration 44
Analysis of aliphatic amines in air samples by HPLC with electrochemical detection 44
Synthesis and antifungal activity of some amidrazone derivatives 43
Stereochemical studies on medicinal agents. 31. Synthesis and opioid antagonist potencies of naltrexamine bivalent ligands with conformationally restricted spacers 43
Conformational properties of diaryldisulphides from dipole moment studies 43
SIMULTANEOUS DETERMINATION OF AMPHETAMINE AND ONE OF ITS METABOLITES BY HPLC WITH ELECTROCHEMICAL DETECTION 43
Novel Sigma Receptor Ligands: Synthesis and Biological Profile 42
Synthesis and pharmacological properties of 2-nitro-3-substituted-aminobenzo b thiophenes and 1-substituted benzothieno 2,3-d imidazoles 42
Specific kappa opioid receptor agonists 42
Synthesis and spectral behaviour of pyridothienoisothiazole and pyridothienopyrimidine derivatives 42
Evaluation of (–)-MR22 a novel sigma-1 receptor ligand on lesion-induced memory dysfunctions in the rat 41
Opioid and sigma receptor studies. New developments in the design of selective sigma ligands 41
Opioid receptors - Development of selective peptidomimetics with agonist or antagonist activity 40
Stereochemistry of hindered cyclophanes. 40
Synthesis of substituted thieno[2,3-c]- and [3,2-d]isothiazoles 40
Hybrid bivalent ligands with opiate and enkephalines pharrmacophores 40
Opioid agonist and antagonist bivalent ligands as receptor probes 40
In-vitro evaluation of a new benzomorphan-based ligand 40
Synthesis and in vitro opioid receptor studies on benzomorphan-based compounds: LP1, a potent and long-acting antinociceptive 40
Synthesis of (+)- and (-)-cis-2-[(1-adamantylamino)-methyl]-1-phenylcyclopropane derivatives as high affinity probes for sigma1 and sigma2 binding sites 40
Calorimetric study on the interaction of thienopyrimidine derivatives with phosphatidylcholine membranes 39
Solution conformation of bis(o-nitrophenyl)disulfide 38
Synthesis of new P3CS derivatives and their mitogenic activity on in vitro mice slenocytes 38
Anti-amnesic and neuroprotective actions of the sigma-1 receptor agonist (-)-MR22 in rats with selective cholinergic lesion and amyloid infusion 38
Synthesis and biological activity of some di(nitrothienyl)- and di (acetylaminothienyl)sulfones 37
Synthesis of 5-substituted-3-phenacyloxime,1,2,4-oxadiazoles from ... 37
Synthesis and pharmacological properties of N-thienyl alkylenediamines 37
Different in vitro activity of flurbiprofen and its enantimers on human articular cartilage 37
Sigma receptor binding profile of a series of analgesic tropane derivatives 37
Design, Synthesis and antiinflammatory activity of novel gamma-tocopherol naproxen ester prodrug 36
A new sigma ligand, (+/-)-PPCC, antagonizes kappa opioid receptor-mediated antinociceptive effect 36
Determination of undecenylic and sorbic acids in cosmetic preparations by high performance electrochemical liquid chromatography with detection 36
Synthesis of substituted pyrimidines, pyrazole[3,4-d]pyrimidines and imidazo[4,5-d]pyrimidines and evaluation of their antifungal activity 36
Synthesis, spectral behaviour and microbiological properties of some di(nitrothienyl)sulfides. 35
Sintesi di ditienildisolfuri. II 35
Stereostructure-activity relationship of opioid agonist and antagonist bivalent ligands. Evidence for bridging between vicinal opioid receptors 35
Methanesulphonamide of 3,5-dihydro-4H-pyrimido[5,4-b]indol4-one and [1]Benzothieno[3,2-d]pirimidin-4(3H)-one derivatives as potential COX-2 inhibitors 35
Development of new benzomorphan LP1 analogues 35
Reactions between thiobenzamides and ethyl beta-chloroacetonoxalate. Synthesis of thiazole, thiazolooxazoline and thiazolopyridazine derivatives 34
Opioid agonist and antagonist bivalent ligands - the relationship between spacer length and selectivity at multiple opioid receptors 34
Irreversible sigma compounds 34
Effect of a new sigma ligand, (±)PPCC, on KOP receptor mediated analgesia 34
Conformation of thianthrene and 2,7-dichlorothianthrene partially oriented in a nematic phase 34
Neuroprotective effects of sigma-1 receptor agonists against beta-amyloid-induced toxicity 34
(+)-MR200 derivatives as potential new selective sigma ligands 33
Synthesis of (+) and (−)-cis-2-[(1-adamantylamino)-methyl]-1-phenylcyclopropane derivatives as probe for sigma-1 and sigma-2 binding sites 33
Sintesi di ditienildisolfuri 32
Design, synthesis, and SAR analysis of novel selective sigma(1) ligands 32
Pain management: new long-acting opioid ligands 32
In vitro evaluation of thiazolyl and benzothiazolyl Schiff bases on pig cartilage 31
Molecular solute conformation of di-2-pyridil disulfide from dipole moment studies 31
New selective sigma receptor ligands cis-(+) and cis-(−) PPCC: in vitro and in vivo studies 31
Selective inhibition of the NOP receptor in the ventrolateral peraqueductal gray attenuates the development and the expression of tolerance to morphine-induced antinociception in rats 31
New benzomorphan derivatives of MPCB as MOP and KOP receptor ligands 31
Simultaneous determination of phenytoin and dextromethorphan in urine by solid-phase extraction and HPLC-DAD 31
Totale 4.441
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Categoria #
all - tutte 15.383
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 15.383
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2018/201932 0 0 0 0 0 0 0 0 0 1 5 26
2019/2020815 306 41 71 20 72 2 107 4 75 7 78 32
2020/20211.035 3 77 124 2 209 17 115 1 191 1 191 104
2021/2022951 129 132 0 16 157 6 132 28 100 1 31 219
2022/20231.621 140 75 15 167 184 305 3 253 419 6 46 8
2023/2024448 43 119 25 38 17 151 7 41 4 3 0 0
Totale 5.244